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Found 11 with Last Name = 'bugni' and Initial = 'ts'
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50252375(CHEMBL446072 | Spheciosterol sulfate C)
Affinity DataIC50:  110nMAssay Description:Inhibition of PKCzeta (unknown origin) by TR-FRET based lanthascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50252374(CHEMBL475118 | Spheciosterol sulfate B)
Affinity DataIC50:  530nMAssay Description:Inhibition of PKCzeta (unknown origin) by TR-FRET based lanthascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50252376(CHEMBL455091 | Topsentiasterol sulfate E)
Affinity DataIC50:  1.21E+3nMAssay Description:Inhibition of PKCzeta (unknown origin) by TR-FRET based lanthascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50252373(CHEMBL447723 | Spheciosterol sulfate A)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of PKCzeta (unknown origin) by TR-FRET based lanthascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50478130(CHEMBL271159)
Affinity DataEC50:  6.00E+3nMAssay Description:Inhibition of hypoxia-induced HIF1 transcriptional activation in human U251-HRE cells by luciferase reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50478131(CHEMBL270091)
Affinity DataEC50:  8.00E+3nMAssay Description:Inhibition of hypoxia-induced HIF1 transcriptional activation in human U251-HRE cells by luciferase reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50478132(CHEMBL259472)
Affinity DataEC50:  1.30E+4nMAssay Description:Inhibition of hypoxia-induced HIF1 transcriptional activation in human U251-HRE cells by luciferase reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor p65(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50252375(CHEMBL446072 | Spheciosterol sulfate C)
Affinity DataEC50:  1.20E+4nMAssay Description:Inhibition of IL1-induced NFkappaB P65 activation in human osteoarthritic primary chondrocytes preincubated 2 hrs before addition of IL1 by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor p65(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50252376(CHEMBL455091 | Topsentiasterol sulfate E)
Affinity DataEC50:  1.20E+4nMAssay Description:Inhibition of IL1-induced NFkappaB P65 activation in human osteoarthritic primary chondrocytes preincubated 2 hrs before addition of IL1 by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor p65(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50252373(CHEMBL447723 | Spheciosterol sulfate A)
Affinity DataEC50:  1.20E+4nMAssay Description:Inhibition of IL1-induced NFkappaB P65 activation in human osteoarthritic primary chondrocytes preincubated 2 hrs before addition of IL1 by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor p65(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50252374(CHEMBL475118 | Spheciosterol sulfate B)
Affinity DataEC50:  1.20E+4nMAssay Description:Inhibition of IL1-induced NFkappaB P65 activation in human osteoarthritic primary chondrocytes preincubated 2 hrs before addition of IL1 by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed