Affinity DataKi: 160nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 0.0650nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 0.570nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 0.850nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 6.5nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 73nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 89nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of human recombinant CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of human recombinant CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
TargetSodium/iodide cotransporter(Rattus norvegicus)
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Institut De Biologie Et De Technologies De Saclay (Ibitecs)
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:inhibition of sodium iodide symporter in rat FRTL5 cells after 1 hr by arsenic/cerium titration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of human recombinant CYP2C9More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of human recombinant CYP2B6More data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of human recombinant CYP2C9More data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of human recombinant CYP2B6More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant CYP2C8More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant CYP2C8More data for this Ligand-Target Pair
Affinity DataEC50: 23nMAssay Description:Inhibition of castor bean ricin-induced toxicity in human A549 cells assessed as protection against toxin-induced inhibition of protein biosynthesis ...More data for this Ligand-Target Pair
Affinity DataEC50: 3.20E+3nMAssay Description:Inhibition of castor bean ricin-induced toxicity in human A549 cells assessed as protection against toxin-induced inhibition of protein biosynthesis ...More data for this Ligand-Target Pair
Affinity DataEC50: 57nMAssay Description:Inhibition of castor bean ricin-induced toxicity in human A549 cells assessed as protection against toxin-induced inhibition of protein biosynthesis ...More data for this Ligand-Target Pair