Affinity DataKi: 450nMAssay Description:In vivo binding affinity fot cytosolic androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:In vivo binding affinity fot cytosolic androgen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 2.22E+3nMAssay Description:Antagonist activity at human recombinant GABAc rho-1 receptor expressed in Xenopus laevis oocytes assessed as inhibition of GABA-induced current by t...More data for this Ligand-Target Pair
Affinity DataIC50: 2.32E+3nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 3.90E+3nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 9.73E+3nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 1.04E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 1.35E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 1.42E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 1.56E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of [3H]-R-1881 binding to rat ventral prostrate cytosolic androgen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.99E+4nMAssay Description:Antagonist activity at human recombinant GABAc rho-1 receptor expressed in Xenopus laevis oocytes assessed as inhibition of GABA-induced current by t...More data for this Ligand-Target Pair
Affinity DataIC50: 2.21E+4nMAssay Description:Antagonist activity at human recombinant GABAc rho-2 receptor expressed in Xenopus laevis oocytes assessed as inhibition of GABA-induced current by t...More data for this Ligand-Target Pair
Affinity DataIC50: 2.74E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 2.97E+4nMAssay Description:Antagonist activity at human recombinant GABAc rho-1 receptor expressed in Xenopus laevis oocytes assessed as inhibition of GABA-induced current by t...More data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 3.59E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+4nMAssay Description:Antagonist activity at human recombinant GABAb 1b/2 receptor expressed in Xenopus laevis oocytes co-expressing GIRK1/4 assessed as inhibition of GABA...More data for this Ligand-Target Pair
Affinity DataIC50: 4.12E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 5.13E+4nMAssay Description:Antagonist activity at human recombinant GABAc rho-2 receptor expressed in Xenopus laevis oocytes assessed as inhibition of GABA-induced current by t...More data for this Ligand-Target Pair
Affinity DataIC50: 5.70E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 5.71E+4nMAssay Description:Antagonist activity at human recombinant GABAc rho-2 receptor expressed in Xenopus laevis oocytes assessed as inhibition of GABA-induced current by t...More data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+4nMAssay Description:Antagonist activity at human recombinant GABAc rho-1 receptor expressed in Xenopus laevis oocytes assessed as inhibition of GABA-induced current by t...More data for this Ligand-Target Pair
Affinity DataIC50: 6.25E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 5.08E+5nMAssay Description:Antagonist activity at human recombinant GABAA alpha1beta2gamma2L receptor expressed in Xenopus laevis oocytes assessed as inhibition of GABA-induced...More data for this Ligand-Target Pair
Affinity DataEC50: 5.00E+5nMAssay Description:Antagonist activity at human recombinant GABAb 1b/2 receptor expressed in Xenopus laevis oocytes co-expressing GIRK1/4 assessed as inhibition of GABA...More data for this Ligand-Target Pair