TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Coimbra
Curated by ChEMBL
University Of Coimbra
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as a substrate by Cornish-Bowden plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the free enzyme using S-butyrylthiocholine iodide as a substrate by Cor...More data for this Ligand-Target Pair
Affinity DataKi: 4.80E+3nMAssay Description:Mixed type inhibition of equine serum BuChE using S-butyrylthiocholine iodide as a substrate by Cornish-Bowden plot analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Coimbra
Curated by ChEMBL
University Of Coimbra
Curated by ChEMBL
Affinity DataKi: 6.10E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as a substrate by Cornish-Bowden plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6.70E+3nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the enzyme-substrate complex using S-butyrylthiocholine iodide as a sub...More data for this Ligand-Target Pair
Affinity DataKi: 7.20E+3nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the free enzyme using S-butyrylthiocholine iodide as a substrate by Cor...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Coimbra
Curated by ChEMBL
University Of Coimbra
Curated by ChEMBL
Affinity DataKi: 7.40E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as a substrate by Cornish-Bowden plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 9.00E+3nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the free enzyme using S-butyrylthiocholine iodide as a substrate by Cor...More data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the enzyme-substrate complex using S-butyrylthiocholine iodide as a sub...More data for this Ligand-Target Pair
Affinity DataKi: 1.37E+4nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the enzyme-substrate complex using S-butyrylthiocholine iodide as a sub...More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Mixed type inhibition of equine serum BuChE using S-butyrylthiocholine iodide as a substrate by Cornish-Bowden plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+4nMAssay Description:Mixed type inhibition of equine serum BuChE using S-butyrylthiocholine iodide as a substrate by Cornish-Bowden plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+4nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the free enzyme using S-butyrylthiocholine iodide as a substrate by Cor...More data for this Ligand-Target Pair
Affinity DataKi: 1.91E+4nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the enzyme-substrate complex using S-butyrylthiocholine iodide as a sub...More data for this Ligand-Target Pair
Affinity DataKi: 4.10E+4nMAssay Description:Reversible competitive inhibition of equine BuChE by Lineweaver-burk plot analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Coimbra
Curated by ChEMBL
University Of Coimbra
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as a substrate and measured upto 180 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of equine serum BuChEMore data for this Ligand-Target Pair
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of AChE in Swiss mouse brain homogenate using acetylthiocholine iodide as substrate by Ellman's assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Coimbra
Curated by ChEMBL
University Of Coimbra
Curated by ChEMBL
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine iodide as a substrate measured for 125 secs by DNTB reagent based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.89E+3nMAssay Description:Antagonistic affinity tested against isolated Rat Prostatic Vas Deferens Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.09E+3nMAssay Description:Antagonistic affinity tested against isolated Rat Spleen Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.24E+3nMAssay Description:Antagonistic affinity tested against isolated Rat Prostatic Vas Deferens Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.31E+3nMAssay Description:Antagonistic affinity tested against isolated Rat Spleen Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Coimbra
Curated by ChEMBL
University Of Coimbra
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as a substrate measured for 125 secs by DNTB reagent based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.76E+3nMAssay Description:Antagonistic affinity tested against isolated Rat Thoracic Aorta Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Coimbra
Curated by ChEMBL
University Of Coimbra
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine iodide as a substrate measured for 125 secs by DNTB reagent based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5.47E+3nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine iodide as a substrate measured for 125 secs by DNTB reagent based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.61E+3nMAssay Description:Inhibition of equine serum BuChE after 15 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 7.41E+3nMAssay Description:Inhibition of equine serum BuChEMore data for this Ligand-Target Pair
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 8.32E+3nMAssay Description:Antagonistic affinity tested against isolated Rat Spleen Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine iodide as a substrate measured for 125 secs by DNTB reagent based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.42E+4nMAssay Description:Antagonistic affinity tested against isolated Rat Prostate Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine iodide as a substrate measured for 125 secs by DNTB reagent based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.83E+4nMAssay Description:Inhibition of equine serum BuChEMore data for this Ligand-Target Pair
Affinity DataIC50: 1.93E+4nMAssay Description:Antagonistic affinity tested against isolated Rat Prostate Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine iodide as a substrate measured for 125 secs by DNTB reagent based Ellman's methodMore data for this Ligand-Target Pair