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Found 161 with Last Name = 'burke' and Initial = 'aj'
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50577715(CHEMBL4866640)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as a substrate by Cornish-Bowden plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592320(CHEMBL5172319)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the free enzyme using S-butyrylthiocholine iodide as a substrate by Cor...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50577715(CHEMBL4866640)
Affinity DataKi:  4.80E+3nMAssay Description:Mixed type inhibition of equine serum BuChE using S-butyrylthiocholine iodide as a substrate by Cornish-Bowden plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50577730(CHEMBL4870225)
Affinity DataKi:  6.10E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as a substrate by Cornish-Bowden plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592320(CHEMBL5172319)
Affinity DataKi:  6.70E+3nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the enzyme-substrate complex using S-butyrylthiocholine iodide as a sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592312(CHEMBL5186546)
Affinity DataKi:  7.20E+3nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the free enzyme using S-butyrylthiocholine iodide as a substrate by Cor...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50577717(CHEMBL4858862)
Affinity DataKi:  7.40E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as a substrate by Cornish-Bowden plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592326(CHEMBL5187617)
Affinity DataKi:  9.00E+3nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the free enzyme using S-butyrylthiocholine iodide as a substrate by Cor...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592328(CHEMBL5179978)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the enzyme-substrate complex using S-butyrylthiocholine iodide as a sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592312(CHEMBL5186546)
Affinity DataKi:  1.37E+4nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the enzyme-substrate complex using S-butyrylthiocholine iodide as a sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50577717(CHEMBL4858862)
Affinity DataKi:  1.50E+4nMAssay Description:Mixed type inhibition of equine serum BuChE using S-butyrylthiocholine iodide as a substrate by Cornish-Bowden plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50577730(CHEMBL4870225)
Affinity DataKi:  1.80E+4nMAssay Description:Mixed type inhibition of equine serum BuChE using S-butyrylthiocholine iodide as a substrate by Cornish-Bowden plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592328(CHEMBL5179978)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the free enzyme using S-butyrylthiocholine iodide as a substrate by Cor...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592326(CHEMBL5187617)
Affinity DataKi:  1.91E+4nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the enzyme-substrate complex using S-butyrylthiocholine iodide as a sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50503819(CHEMBL4565335)
Affinity DataKi:  4.10E+4nMAssay Description:Reversible competitive inhibition of equine BuChE by Lineweaver-burk plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50592330(CHEMBL5193166)
Affinity DataIC50:  100nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as a substrate and measured upto 180 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50344826(1-(4-chlorobenzyl)-3-hydroxy-3-phenylindolin-2-one...)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of equine serum BuChEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  1.06E+3nMAssay Description:Inhibition of AChE in Swiss mouse brain homogenate using acetylthiocholine iodide as substrate by Ellman's assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50577715(CHEMBL4866640)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine iodide as a substrate measured for 125 secs by DNTB reagent based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50407439(CHEMBL5273857)
Affinity DataIC50:  1.89E+3nMAssay Description:Antagonistic affinity tested against isolated Rat Prostatic Vas Deferens Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  2.09E+3nMAssay Description:Antagonistic affinity tested against isolated Rat Spleen Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50407440(CHEMBL5286517)
Affinity DataIC50:  2.24E+3nMAssay Description:Antagonistic affinity tested against isolated Rat Prostatic Vas Deferens Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50407437(CHEMBL5274569)
Affinity DataIC50:  2.31E+3nMAssay Description:Antagonistic affinity tested against isolated Rat Spleen Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as a substrate measured for 125 secs by DNTB reagent based Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50407436(CHEMBL5287904)
Affinity DataIC50:  2.76E+3nMAssay Description:Antagonistic affinity tested against isolated Rat Thoracic Aorta Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592320(CHEMBL5172319)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592319(CHEMBL5184631)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  3.50E+3nMAssay Description:The inhibition assay of these compounds for AChE (electrophorus electricus) and BuChE (equine serum) were determined by the spectroscopic method desc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine iodide as a substrate measured for 125 secs by DNTB reagent based Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592323(CHEMBL5175872)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592312(CHEMBL5186546)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  5.47E+3nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50577730(CHEMBL4870225)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine iodide as a substrate measured for 125 secs by DNTB reagent based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592321(CHEMBL5201709)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50503820(CHEMBL4550082)
Affinity DataIC50:  6.61E+3nMAssay Description:Inhibition of equine serum BuChE after 15 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592309(CHEMBL5203011)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50503818(CHEMBL4593576)
Affinity DataIC50:  7.41E+3nMAssay Description:Inhibition of equine serum BuChEMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592326(CHEMBL5187617)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50407437(CHEMBL5274569)
Affinity DataIC50:  8.32E+3nMAssay Description:Antagonistic affinity tested against isolated Rat Spleen Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50577717(CHEMBL4858862)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine iodide as a substrate measured for 125 secs by DNTB reagent based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592328(CHEMBL5179978)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592314(CHEMBL5203069)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50407440(CHEMBL5286517)
Affinity DataIC50:  1.42E+4nMAssay Description:Antagonistic affinity tested against isolated Rat Prostate Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592305(CHEMBL5182078)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50577737(CHEMBL4853721)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine iodide as a substrate measured for 125 secs by DNTB reagent based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50592307(CHEMBL5198472)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of Equine serum BuChE using S-butyrylthiocholine iodide as a substrate and measured for 125 sec by DTNB based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50503819(CHEMBL4565335)
Affinity DataIC50:  1.83E+4nMAssay Description:Inhibition of equine serum BuChEMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  1.93E+4nMAssay Description:Antagonistic affinity tested against isolated Rat Prostate Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetCholinesterase(Equus caballus (Horse))
University Of £Vora

Curated by ChEMBL
LigandPNGBDBM50577719(CHEMBL4858873)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine iodide as a substrate measured for 125 secs by DNTB reagent based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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