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Found 5 with Last Name = 'buskes' and Initial = 'mj'
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM10995((1R)-N-methyl-2,3-dihydro-1H-inden-1-amine | N-met...)
Affinity DataIC50:  200nMAssay Description:Inhibition of PDK1 (unknown origin) expressed in HEK293 cells using PDKtide as substrate after 10 mins by liquid scintillation counting in presence o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50049555(CHEMBL3311455)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of PDK1 (unknown origin) expressed in HEK293 cells using PDKtide as substrate after 10 mins by liquid scintillation counting in presence o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))TBA
LigandPNGBDBM50614737(CHEMBL2180750)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of IDH1 R132H mutant (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50049556(CHEMBL3311451)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of PDK1 (unknown origin) expressed in HEK293 cells using PDKtide as substrate after 10 mins by liquid scintillation counting in presence o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))TBA
LigandPNGBDBM50614738(CHEMBL2180749)
Affinity DataIC50: >1.10E+4nMAssay Description:Inhibition of IDH1 R132H mutant (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed