Compile Data Set for Download or QSAR
maximum 50k data
Found 109 with Last Name = 'butler' and Initial = 'hs'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265896(CHEMBL4070359)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of Adenosine A2A receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600005(CHEMBL5195268)
Affinity DataIC50:  30nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)
Affinity DataIC50:  45nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activityMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600003(CHEMBL5201228)
Affinity DataIC50:  55nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50050549(GSK2140944 | Gepotidacin)
Affinity DataIC50:  60nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activityMore data for this Ligand-Target Pair
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600006(CHEMBL5172158)
Affinity DataIC50:  90nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600007(CHEMBL5182200)
Affinity DataIC50:  105nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600004(CHEMBL5184104)
Affinity DataIC50:  220nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600009(CHEMBL5177076)
Affinity DataIC50:  340nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600008(CHEMBL5198597)
Affinity DataIC50:  460nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265895(CHEMBL4097537)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of phosphodiesterase 4D (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600011(CHEMBL5205047)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600007(CHEMBL5182200)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600010(CHEMBL5184352)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600003(CHEMBL5201228)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600013(CHEMBL5194618)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600018(CHEMBL5199405)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600014(CHEMBL5172094)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600012(CHEMBL5190832)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600017(CHEMBL5195721)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600003(CHEMBL5201228)
Affinity DataIC50:  1.44E+4nMAssay Description:Inhibition of human topoisomerase 2 assessed as reduction in decatenationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600015(CHEMBL5206169)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600004(CHEMBL5184104)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600016(CHEMBL5170129)
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50050549(GSK2140944 | Gepotidacin)
Affinity DataIC50:  5.52E+4nMAssay Description:Inhibition of human topoisomerase 2 assessed as reduction in decatenationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600005(CHEMBL5195268)
Affinity DataIC50:  7.28E+4nMAssay Description:Inhibition of human topoisomerase 2 assessed as reduction in decatenationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600007(CHEMBL5182200)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human topoisomerase 2 assessed as reduction in decatenationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50050549(GSK2140944 | Gepotidacin)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600006(CHEMBL5172158)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human topoisomerase 2 assessed as reduction in decatenationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600004(CHEMBL5184104)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human topoisomerase 2 assessed as reduction in decatenationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human topoisomerase 2 assessed as reduction in decatenationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600009(CHEMBL5177076)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600008(CHEMBL5198597)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600008(CHEMBL5198597)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human topoisomerase 2 assessed as reduction in decatenationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600006(CHEMBL5172158)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600005(CHEMBL5195268)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human ERG by Ionworks electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Redx Anti-Infectives

Curated by ChEMBL
LigandPNGBDBM50600009(CHEMBL5177076)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human topoisomerase 2 assessed as reduction in decatenationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265860(CHEMBL4082804)
Affinity DataEC50: >1.70E+4nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265862(CHEMBL4077507)
Affinity DataEC50:  640nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265865(CHEMBL4076190)
Affinity DataEC50:  260nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265868(CHEMBL4071228)
Affinity DataEC50: >1.70E+4nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265874(CHEMBL4085695)
Affinity DataEC50:  2.60E+3nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265875(CHEMBL4070273)
Affinity DataEC50:  720nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265876(CHEMBL4077353)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265877(CHEMBL4101071)
Affinity DataEC50:  710nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265878(CHEMBL4060517)
Affinity DataEC50:  990nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265879(CHEMBL4065429)
Affinity DataEC50: >1.70E+4nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265880(CHEMBL4076004)
Affinity DataEC50:  760nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265881(CHEMBL4065890)
Affinity DataEC50:  4.80E+3nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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