Compile Data Set for Download or QSAR
maximum 50k data
Found 752 with Last Name = 'calbet' and Initial = 'm'
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211682(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}pyri...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211685(4'-(2-furyl)-N-pyridin-3-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211680(4'-(2-furyl)-N-pyrimidin-5-yl-4,5'-bipyrimidin-2'-...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211688(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}-1-m...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211679(4'-(2-furyl)-N-(1-oxidopyridin-3-yl)-4,5'-bipyrimi...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211684(4'-(2-furyl)-N-(2-methoxypyrimidin-5-yl)-4,5'-bipy...)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211687(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}nico...)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211681(4'-(2-furyl)-N-(6-methoxypyridin-3-yl)-4,5'-bipyri...)
Affinity DataKi:  115nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211686(4'-(2-furyl)-N-pyrazin-2-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211683(1-(cyclopropylmethyl)-5-{[4'-(2-furyl)-4,5'-bipyri...)
Affinity DataKi:  119nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211682(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}pyri...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211687(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}nico...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211685(4'-(2-furyl)-N-pyridin-3-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211683(1-(cyclopropylmethyl)-5-{[4'-(2-furyl)-4,5'-bipyri...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211681(4'-(2-furyl)-N-(6-methoxypyridin-3-yl)-4,5'-bipyri...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211688(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}-1-m...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211684(4'-(2-furyl)-N-(2-methoxypyrimidin-5-yl)-4,5'-bipy...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211686(4'-(2-furyl)-N-pyrazin-2-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211680(4'-(2-furyl)-N-pyrimidin-5-yl-4,5'-bipyrimidin-2'-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211679(4'-(2-furyl)-N-(1-oxidopyridin-3-yl)-4,5'-bipyrimi...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211685(4'-(2-furyl)-N-pyridin-3-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211681(4'-(2-furyl)-N-(6-methoxypyridin-3-yl)-4,5'-bipyri...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211685(4'-(2-furyl)-N-pyridin-3-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211687(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}nico...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211682(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}pyri...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211680(4'-(2-furyl)-N-pyrimidin-5-yl-4,5'-bipyrimidin-2'-...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211683(1-(cyclopropylmethyl)-5-{[4'-(2-furyl)-4,5'-bipyri...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211684(4'-(2-furyl)-N-(2-methoxypyrimidin-5-yl)-4,5'-bipy...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211679(4'-(2-furyl)-N-(1-oxidopyridin-3-yl)-4,5'-bipyrimi...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211688(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}-1-m...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211686(4'-(2-furyl)-N-pyrazin-2-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211681(4'-(2-furyl)-N-(6-methoxypyridin-3-yl)-4,5'-bipyri...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211682(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}pyri...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211679(4'-(2-furyl)-N-(1-oxidopyridin-3-yl)-4,5'-bipyrimi...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211687(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}nico...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211688(5-{[4'-(2-furyl)-4,5'-bipyrimidin-2'-yl]amino}-1-m...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211683(1-(cyclopropylmethyl)-5-{[4'-(2-furyl)-4,5'-bipyri...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211686(4'-(2-furyl)-N-pyrazin-2-yl-4,5'-bipyrimidin-2'-am...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211680(4'-(2-furyl)-N-pyrimidin-5-yl-4,5'-bipyrimidin-2'-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211680(4'-(2-furyl)-N-pyrimidin-5-yl-4,5'-bipyrimidin-2'-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Almirall

Curated by ChEMBL
LigandPNGBDBM50211684(4'-(2-furyl)-N-(2-methoxypyrimidin-5-yl)-4,5'-bipy...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50450675(CHEMBL4166977)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant human N-terminal His-tagged full length p110delta/recombinant human full length p85alpha using PIP2 as substrate preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
LigandPNGBDBM236931(US9388189, 27)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant human N-terminal His-tagged full length p110delta/recombinant human full length p85alpha using PIP2 as substrate preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50450680(CHEMBL4168702)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant human N-terminal His-tagged full length p110delta/recombinant human full length p85alpha using PIP2 as substrate preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM236932(US9388189, 28)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant human N-terminal His-tagged full length p110delta/recombinant human full length p85alpha using PIP2 as substrate preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50450688(CHEMBL4168086)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant human N-terminal His-tagged full length p110delta/recombinant human full length p85alpha using PIP2 as substrate preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM236935(US9388189, 36)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant human N-terminal His-tagged full length p110delta/recombinant human full length p85alpha using PIP2 as substrate preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50450693(CHEMBL4164842)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant human N-terminal His-tagged full length p110delta/recombinant human full length p85alpha using PIP2 as substrate preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50450687(CHEMBL4164818)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant human N-terminal His-tagged full length p110delta/recombinant human full length p85alpha using PIP2 as substrate preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50450679(CHEMBL4164652)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant human N-terminal His-tagged full length p110delta/recombinant human full length p85alpha using PIP2 as substrate preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 752 total ) | Next | Last >>
Jump to: