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Found 112 with Last Name = 'campo' and Initial = 'b'
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009661(CHEMBL3235218)
Affinity DataKi:  588nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009659(CHEMBL3235216)
Affinity DataKi:  1.49E+3nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009660(CHEMBL3235217)
Affinity DataKi:  3.08E+3nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009658(CHEMBL3235215)
Affinity DataKi:  6.22E+3nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009664(CHEMBL3235221)
Affinity DataKi:  3.12E+4nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009670(CHEMBL3235227)
Affinity DataKi:  5.52E+4nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009694(CHEMBL3235232)
Affinity DataKi:  1.37E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009663(CHEMBL3235220)
Affinity DataKi:  1.44E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009667(CHEMBL3235224)
Affinity DataKi:  1.59E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009662(CHEMBL3235219 | US9162983, C)
Affinity DataKi:  1.80E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009715(CHEMBL3235235)
Affinity DataKi:  1.99E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009665(CHEMBL3235222)
Affinity DataKi:  1.99E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009675(CHEMBL3235230)
Affinity DataKi:  2.33E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009650(CHEMBL3235207)
Affinity DataKi:  2.34E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009713(CHEMBL3235234)
Affinity DataKi:  2.66E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009671(CHEMBL3235228)
Affinity DataKi:  2.86E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009669(CHEMBL3235226)
Affinity DataKi:  2.98E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009673(CHEMBL3235229)
Affinity DataKi:  3.45E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009692(CHEMBL3235231)
Affinity DataKi:  5.51E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009655(CHEMBL3235212)
Affinity DataKi:  5.95E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009652(CHEMBL3235209)
Affinity DataKi:  7.33E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009668(CHEMBL3235225)
Affinity DataKi:  1.61E+6nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009654(CHEMBL3235211)
Affinity DataKi:  1.63E+6nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009656(CHEMBL3235213)
Affinity DataKi:  1.93E+6nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009666(CHEMBL3235223)
Affinity DataKi:  1.93E+6nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009651(CHEMBL3235208 | US9162983, E)
Affinity DataKi:  2.30E+6nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009648(CHEMBL3235205)
Affinity DataKi:  2.43E+6nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009711(CHEMBL3235233)
Affinity DataKi:  2.52E+6nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009657(CHEMBL3235214)
Affinity DataKi:  2.67E+6nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009649(CHEMBL3235206)
Affinity DataKi:  3.18E+6nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Southwest Research Institute

Curated by ChEMBL
LigandPNGBDBM50009653(CHEMBL3235210)
Affinity DataKi:  9.50E+7nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate after 4 hrs by robotic spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50603975(CHEMBL5201780)
Affinity DataIC50:  3nMAssay Description:Inhibition of human Haspin kinase domain using histone H3 biotin peptide as substrate preincubated with enzyme for 30 mins followed by substrate and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50603974(CHEMBL5201904)
Affinity DataIC50:  5nMAssay Description:Inhibition of human Haspin kinase domain using histone H3 biotin peptide as substrate preincubated with enzyme for 30 mins followed by substrate and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50603992(CHEMBL5179988)
Affinity DataIC50:  11nMAssay Description:Inhibition of human Haspin kinase domain using histone H3 biotin peptide as substrate preincubated with enzyme for 30 mins followed by substrate and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of Liverpool

Curated by ChEMBL
LigandPNGBDBM151585(US11739089, Compound Ketoconazole | US8987315, Ket...)
Affinity DataIC50:  13nMAssay Description:Inhibition of CYP3A4 in human liver microsomes assessed as testosterone 6beta-hydroxylation after 4 to 40 mins in presence of NADPH by LCMS analysisMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of Liverpool

Curated by ChEMBL
LigandPNGBDBM151585(US11739089, Compound Ketoconazole | US8987315, Ket...)
Affinity DataIC50:  22nMAssay Description:Inhibition of CYP3A4 in human liver microsomes assessed as midazolam 1'-hydroxylation after 4 to 40 mins in presence of NADPH by LCMS analysisMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
University Of Liverpool

Curated by ChEMBL
LigandPNGBDBM50121975((6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2...)
Affinity DataIC50:  25nMAssay Description:Inhibition of CYP2D6 in human liver microsomes assessed as dextromethorphan O-demethylation after 4 to 40 mins in presence of NADPH by LCMS analysisMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50603978(CHEMBL5187817)
Affinity DataIC50:  32nMAssay Description:Inhibition of human Haspin kinase domain using histone H3 biotin peptide as substrate preincubated with enzyme for 30 mins followed by substrate and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50603989(CHEMBL5192443)
Affinity DataIC50:  45nMAssay Description:Inhibition of human Haspin kinase domain using histone H3 biotin peptide as substrate preincubated with enzyme for 30 mins followed by substrate and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50603986(CHEMBL5187610)
Affinity DataIC50:  78nMAssay Description:Inhibition of human Haspin kinase domain using histone H3 biotin peptide as substrate preincubated with enzyme for 30 mins followed by substrate and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50603988(CHEMBL5170360)
Affinity DataIC50:  140nMAssay Description:Inhibition of human Haspin kinase domain using histone H3 biotin peptide as substrate preincubated with enzyme for 30 mins followed by substrate and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50603984(CHEMBL5195201)
Affinity DataIC50:  200nMAssay Description:Inhibition of human Haspin kinase domain using histone H3 biotin peptide as substrate preincubated with enzyme for 30 mins followed by substrate and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
University Of Liverpool

Curated by ChEMBL
LigandPNGBDBM50273689(CHEMBL4128999)
Affinity DataIC50:  480nMAssay Description:Inhibition of CYP2C19 in human liver microsomes assessed as (S)-mephenytoin 4'-hydroxylation after 4 to 40 mins in presence of NADPH by LCMS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50603985(CHEMBL5207627)
Affinity DataIC50:  690nMAssay Description:Inhibition of human Haspin kinase domain using histone H3 biotin peptide as substrate preincubated with enzyme for 30 mins followed by substrate and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
University Of Liverpool

Curated by ChEMBL
LigandPNGBDBM50090677(4-Amino-N-(2-phenyl-2H-pyrazol-3-yl)-benzenesulfon...)
Affinity DataIC50:  720nMAssay Description:Inhibition of CYP2C9 in human liver microsomes assessed as tolbutamide methylhydroxylation after 4 to 40 mins in presence of NADPH by LCMS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50603979(CHEMBL5204715)
Affinity DataIC50:  770nMAssay Description:Inhibition of human Haspin kinase domain using histone H3 biotin peptide as substrate preincubated with enzyme for 30 mins followed by substrate and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50603976(CHEMBL5200247)
Affinity DataIC50:  1.28E+3nMAssay Description:Inhibition of human Haspin kinase domain using histone H3 biotin peptide as substrate preincubated with enzyme for 30 mins followed by substrate and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50603983(CHEMBL5181699)
Affinity DataIC50:  1.33E+3nMAssay Description:Inhibition of human Haspin kinase domain using histone H3 biotin peptide as substrate preincubated with enzyme for 30 mins followed by substrate and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50603977(CHEMBL5189523)
Affinity DataIC50:  1.74E+3nMAssay Description:Inhibition of human Haspin kinase domain using histone H3 biotin peptide as substrate preincubated with enzyme for 30 mins followed by substrate and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50603977(CHEMBL5189523)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of hERG by Qpatch-clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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