Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute
Curated by ChEMBL
Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 0.589nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptor in the rabbit heartMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute
Curated by ChEMBL
Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 0.603nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor entirely in guinea pig ileumMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute
Curated by ChEMBL
Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptors in the rabbit heartMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute
Curated by ChEMBL
Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptor in the rabbit heartMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute
Curated by ChEMBL
Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor of neuronal in the afferent rabbit vagusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute
Curated by ChEMBL
Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor of neuronal in the afferent rabbit vagusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute
Curated by ChEMBL
Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 3.31nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptors in the rabbit heartMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute
Curated by ChEMBL
Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 9.10nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor of neuronal in the afferent rabbit vagusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute
Curated by ChEMBL
Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptors in the rabbit heartMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
Hoechst Marion Roussel
Curated by PDSP Ki Database
Hoechst Marion Roussel
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Hoechst Marion Roussel
Curated by PDSP Ki Database
Hoechst Marion Roussel
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Hoechst Marion Roussel
Curated by PDSP Ki Database
Hoechst Marion Roussel
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute
Curated by ChEMBL
Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor entirely in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Mixed non-competitive inhibition of Leishmania infantum TryR using TS2 as substrate assessed as inhibition constant of two-step induced-fit mechanism...More data for this Ligand-Target Pair
Ligand Info
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Merrell Dow Research Institute
Curated by ChEMBL
Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 229nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptor in the rabbit heartMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Mixed non-competitive inhibition of Leishmania infantum TryR using TS2 as substrate assessed as inhibition constant of first equilibrium by plot anal...More data for this Ligand-Target Pair
Ligand Info
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Hoechst Marion Roussel
Curated by PDSP Ki Database
Hoechst Marion Roussel
Curated by PDSP Ki Database
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Hoechst Marion Roussel
Curated by PDSP Ki Database
Hoechst Marion Roussel
Curated by PDSP Ki Database
Affinity DataKi: 7.30E+3nMAssay Description:Competitive inhibition of HIS-FLAG-tagged recombinant Leishmania infantum TryR expressed in Escherichia coli using TS2 substrate assessed as inhibiti...More data for this Ligand-Target Pair
Ligand Info
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Hoechst Marion Roussel
Curated by PDSP Ki Database
Hoechst Marion Roussel
Curated by PDSP Ki Database
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of HIS-tagged recombinant Leishmania infantum TryR oxidoreductase activity expressed in Escherichia coli in the presence of NADPH by spect...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of HIS-tagged recombinant Leishmania infantum TryR oxidoreductase activity expressed in Escherichia coli in the presence of NADPH by spect...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of HIS-tagged recombinant Leishmania infantum TryR oxidoreductase activity expressed in Escherichia coli in the presence of NADPH by spect...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of HIS-tagged recombinant Leishmania infantum TryR oxidoreductase activity expressed in Escherichia coli in the presence of NADPH by spect...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of HIS-tagged recombinant Trypanosoma congolense TryR oxidoreductase activity expressed in Escherichia coli in the presence of NADPH by sp...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of HIS-tagged recombinant Leishmania infantum TryR oxidoreductase activity expressed in Escherichia coli in the presence of NADPH by spect...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of HIS-tagged recombinant Leishmania infantum TryR oxidoreductase activity expressed in Escherichia coli in the presence of NADPH by spect...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of HIS-tagged recombinant Leishmania infantum TryR oxidoreductase activity expressed in Escherichia coli in the presence of NADPH by spect...More data for this Ligand-Target Pair
Ligand Info