Affinity DataKi: 0.0501nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in human U20S cells assessed as effect on substance P-induced intracellular calcium l...More data for this Ligand-Target Pair
Affinity DataKi: 0.0631nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in human U20S cells assessed as effect on substance P-induced intracellular calcium l...More data for this Ligand-Target Pair
Affinity DataKi: 0.0794nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in human U20S cells assessed as effect on substance P-induced intracellular calcium l...More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in human U20S cells assessed as effect on substance P-induced intracellular calcium l...More data for this Ligand-Target Pair
Affinity DataKi: 0.158nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in human U20S cells assessed as effect on substance P-induced intracellular calcium l...More data for this Ligand-Target Pair
Affinity DataKi: 0.251nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in human U20S cells assessed as effect on substance P-induced intracellular calcium l...More data for this Ligand-Target Pair
Affinity DataKi: 0.251nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in human U20S cells assessed as effect on substance P-induced intracellular calcium l...More data for this Ligand-Target Pair
Affinity DataKi: 0.251nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in human U20S cells assessed as effect on substance P-induced intracellular calcium l...More data for this Ligand-Target Pair
Affinity DataKi: 0.251nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in human U20S cells assessed as effect on substance P-induced intracellular calcium l...More data for this Ligand-Target Pair
Affinity DataKi: 0.316nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in human U20S cells assessed as effect on substance P-induced intracellular calcium l...More data for this Ligand-Target Pair
Affinity DataKi: 0.501nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in human U20S cells assessed as effect on substance P-induced intracellular calcium l...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in human U20S cells assessed as effect on NKB-induced intracellular calcium level by ...More data for this Ligand-Target Pair
Affinity DataKi: 1.58nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in human U20S cells assessed as effect on NKB-induced intracellular calcium level by ...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in human U20S cells assessed as effect on NKB-induced intracellular calcium level by ...More data for this Ligand-Target Pair
Affinity DataKi: 5.01nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in human U20S cells assessed as effect on NKB-induced intracellular calcium level by ...More data for this Ligand-Target Pair
Affinity DataKi: 5.01nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in human U20S cells assessed as effect on NKB-induced intracellular calcium level by ...More data for this Ligand-Target Pair
Affinity DataKi: 6.31nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in human U20S cells assessed as effect on NKB-induced intracellular calcium level by ...More data for this Ligand-Target Pair
Affinity DataKi: 7.94nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in human U20S cells assessed as effect on NKB-induced intracellular calcium level by ...More data for this Ligand-Target Pair
Affinity DataKi: 19.9nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in human U20S cells assessed as effect on NKB-induced intracellular calcium level by ...More data for this Ligand-Target Pair
Affinity DataKi: 25.1nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in human U20S cells assessed as effect on NKB-induced intracellular calcium level by ...More data for this Ligand-Target Pair
Affinity DataKi: 31.6nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in human U20S cells assessed as effect on NKB-induced intracellular calcium level by ...More data for this Ligand-Target Pair
Affinity DataKi: 31.6nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in human U20S cells assessed as effect on NKB-induced intracellular calcium level by ...More data for this Ligand-Target Pair
Affinity DataKi: 39.8nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in human U20S cells assessed as effect on NKB-induced intracellular calcium level by ...More data for this Ligand-Target Pair
Affinity DataKi: 79.4nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in human U20S cells assessed as effect on NKB-induced intracellular calcium level by ...More data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in human U20S cells assessed as effect on NKB-induced intracellular calcium level by ...More data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in human U20S cells assessed as effect on NKB-induced intracellular calcium level by ...More data for this Ligand-Target Pair
Affinity DataKi: 794nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in human U20S cells assessed as effect on NKB-induced intracellular calcium level by ...More data for this Ligand-Target Pair
Affinity DataIC50: 0.410nMAssay Description:Inhibition of Matrix metalloprotease-2 in MMPi assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.70nMAssay Description:Inhibition of Matrix metalloprotease-14 in MMPi assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30nMAssay Description:Inhibition of Matrix metalloprotease-9 in MMPi assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.80nMAssay Description:Inhibition of Matrix metalloprotease-2 in MMPi assayMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of Matrix metalloprotease-9 in MMPi assayMore data for this Ligand-Target Pair
Affinity DataIC50: 197nMAssay Description:Inhibition of Matrix metalloprotease-2 in MMPi assayMore data for this Ligand-Target Pair
Affinity DataIC50: 397nMAssay Description:Inhibition of Matrix metalloprotease-1 in MMPi assayMore data for this Ligand-Target Pair
Affinity DataIC50: 983nMAssay Description:Inhibition of Matrix metalloprotease-9 in MMPi assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.49E+3nMAssay Description:Inhibition of Matrix metalloprotease-14 in MMPi assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Matrix metalloprotease-2 in MMPi assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Matrix metalloprotease-1 in MMPi assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Matrix metalloprotease-9 in MMPi assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Matrix metalloprotease-1 in MMPi assayMore data for this Ligand-Target Pair