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Found 100 with Last Name = 'chabrier' and Initial = 'pe'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM21283(3-[(2-iodo-5-nitrophenyl)carbonyl]-1-[(1-methylpip...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089965(CHEMBL3581222)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089958(CHEMBL3581226)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089956(CHEMBL3581228)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089959(CHEMBL3581225)
Affinity DataKi:  77nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089968(CHEMBL3581220)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089970(CHEMBL3581229)
Affinity DataKi:  127nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089963(CHEMBL3581224)
Affinity DataKi:  144nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089957(CHEMBL3581227)
Affinity DataKi:  177nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089956(CHEMBL3581228)
Affinity DataKi:  817nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089965(CHEMBL3581222)
Affinity DataKi:  857nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM21283(3-[(2-iodo-5-nitrophenyl)carbonyl]-1-[(1-methylpip...)
Affinity DataKi:  2.08E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089958(CHEMBL3581226)
Affinity DataKi:  2.17E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089963(CHEMBL3581224)
Affinity DataKi:  2.27E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089968(CHEMBL3581220)
Affinity DataKi:  2.34E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089964(CHEMBL3581223)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089959(CHEMBL3581225)
Affinity DataKi:  3.30E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089970(CHEMBL3581229)
Affinity DataKi:  4.71E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089966(CHEMBL3581221)
Affinity DataKi:  6.24E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089964(CHEMBL3581223)
Affinity DataKi:  6.96E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50179750((S)-2-((S)-2-(benzyloxycarbonyl)-4-methylpentanami...)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50179749((S)-2-(2-(2-(10H-phenothiazin-2-yloxy)acetamido)ac...)
Affinity DataIC50:  8nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50223720(CHEMBL332257)
Affinity DataIC50:  8nMAssay Description:Concentration required to inhibit [3H]BTX binding to Sodium channel of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50223731(CHEMBL118603)
Affinity DataIC50:  16nMAssay Description:Concentration required to inhibit [3H]BTX binding to Sodium channel of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50223721(CHEMBL331513)
Affinity DataIC50:  19nMAssay Description:Concentration required to inhibit [3H]BTX binding to Sodium channel of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50149195(1-Benzyl-2,3-dihydro-1H-indole-5-carboxylic acid [...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against on human calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50223715(CHEMBL3706732)
Affinity DataIC50:  23nMAssay Description:Inhibitory activity against on human calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50223726(CHEMBL117331)
Affinity DataIC50:  25nMAssay Description:Concentration required to inhibit [3H]BTX binding to Sodium channel of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50179745((S)-2-((S)-2-(2-(10H-phenothiazin-2-yloxy)acetamid...)
Affinity DataIC50:  25nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50223735(CHEMBL119139)
Affinity DataIC50:  26nMAssay Description:Concentration required to inhibit [3H]BTX binding to Sodium channel of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50223734(CHEMBL331942)
Affinity DataIC50:  28nMAssay Description:Concentration required to inhibit [3H]BTX binding to Sodium channel of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50223733(CHEMBL120306)
Affinity DataIC50:  30nMAssay Description:Concentration required to inhibit [3H]BTX binding to Sodium channel of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50179747((S)-2-((2S,3S)-2-(2-(10H-phenothiazin-2-yloxy)acet...)
Affinity DataIC50:  38nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50179743((S)-2-((S)-2-(2-(10H-phenothiazin-2-yloxy)acetamid...)
Affinity DataIC50:  48.7nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50065843(CHEMBL553081 | CHEMBL555715 | N-(3-Aminomethyl-phe...)
Affinity DataIC50:  50nMAssay Description:Inhibitory concentration tested against neuronal nitric oxide synthase (nNOS ) from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50179744((S)-4-Methyl-2-[(S)-4-methyl-2-(2-10H-phenothiazin...)
Affinity DataIC50:  55.4nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50223722(CHEMBL334104)
Affinity DataIC50:  70nMAssay Description:Concentration required to inhibit [3H]BTX binding to Sodium channel of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50179741((S)-2-((S)-2-(2-(10H-phenothiazin-2-yloxy)acetamid...)
Affinity DataIC50:  75.9nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50122299(CHEMBL538500 | N-[4-(2-Amino-ethyl)-phenyl]-thioph...)
Affinity DataIC50:  80nMAssay Description:Inhibitory concentration tested against neuronal nitric oxide synthase (nNOS ) from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50223717(CHEMBL3706727)
Affinity DataIC50:  82nMAssay Description:Inhibitory activity against on calpain in C6 glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50179738(CHEMBL203244 | N-((S)-1-((S)-1-((3S)-2-hydroxy-tet...)
Affinity DataIC50:  85.5nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50223723(CHEMBL119494)
Affinity DataIC50:  86nMAssay Description:Concentration required to inhibit [3H]BTX binding to Sodium channel of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50179746((S)-2-((S)-2-(2-(10H-phenothiazin-2-yloxy)acetamid...)
Affinity DataIC50:  88.6nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50223725(CHEMBL118682)
Affinity DataIC50:  100nMAssay Description:Concentration required to inhibit [3H]BTX binding to Sodium channel of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50179739((S)-4-Methyl-2-{(S)-4-methyl-2-[2-(10H-phenothiazi...)
Affinity DataIC50:  105nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50122300(CHEMBL541300 | N-(3-{[3-(4-Hydroxy-3,5-diisopropyl...)
Affinity DataIC50:  120nMAssay Description:Inhibitory concentration tested against neuronal nitric oxide synthase (nNOS ) from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM196649(US9212144, 4)
Affinity DataIC50:  120nMAssay Description:Inhibitory concentration tested against neuronal nitric oxide synthase (nNOS ) from rat cerebellumMore data for this Ligand-Target Pair
TargetCalpain small subunit 1/1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50179754((S)-2-(2-(2-(10H-phenothiazin-2-yloxy)acetamido)-2...)
Affinity DataIC50:  138nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50223729(CHEMBL418863)
Affinity DataIC50:  146nMAssay Description:Concentration required to inhibit [3H]BTX binding to Sodium channel of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50149199(6-Hydroxy-2,5,7,8-tetramethyl-chroman-2-carboxylic...)
Affinity DataIC50:  147nMAssay Description:Inhibitory activity against on human calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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