Affinity DataKi: 1.10nMAssay Description:Compound was evaluated for affinity towards human tachykinin NK-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Compound was evaluated for affinity towards human tachykinin NK-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Compound was evaluated for affinity towards human tachykinin NK-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Compound was evaluated for affinity towards human tachykinin NK-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Compound was evaluated for affinity towards human tachykinin NK-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Compound was evaluated for affinity towards human tachykinin NK-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 630nMAssay Description:Compound was evaluated for affinity towards human tachykinin NK-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-SP to Neurokinin-1 (NK-1) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.640nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-SP to Neurokinin-1 (NK-1) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-SP to Neurokinin-1 (NK-1) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-SP to Neurokinin-1 (NK-1) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-SP to Neurokinin-1 (NK-1) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-SP to Neurokinin-1 (NK-1) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-SP to Neurokinin-1 (NK-1) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Displacement of Eu-DTPA-CCK8 from CCK2 receptor in HEK293 cells after 2 hrs by TRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Displacement of Eu-DTPA-CCK8 from CCK2 receptor in HEK293 cells after 2 hrs by TRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.80nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-SP to Neurokinin-1 (NK-1) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 8.5nMAssay Description:Displacement of Eu-DTPA-CCK8 from CCK2 receptor in HEK293 cells after 2 hrs by TRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Concentration required to inhibit the specific binding of [125I]NKA to Neurokinin-2 (NK-2) receptor in rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of Eu-DTPA-CCK8 from CCK2 receptor in HEK293 cells after 2 hrs by TRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Binding affinity to MC4R in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Displacement of Eu-NDP-alpha-MSH from human MC4R expressed in HEK293 cells by time resolved fluorescence binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Displacement of Eu-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 2 hrs by time resolved fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Displacement of Eu-DTPA-CCK8 from CCK2 receptor in HEK293 cells after 2 hrs by TRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-SP to Neurokinin-1 (NK-1) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-SP to Neurokinin-1 (NK-1) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Concentration required to inhibit the specific binding of [125I]NKA to Neurokinin-2 (NK-2) receptor in rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Binding affinity to MC4R in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Concentration required to inhibit the specific binding of [125I]NKA to Neurokinin-2 (NK-2) receptor in rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Displacement of Eu-NDP-alpha-MSH from human MC4R expressed in HEK293 cells by time resolved fluorescence binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-SP to Neurokinin-1 (NK-1) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 57nMAssay Description:Concentration required to inhibit the specific binding of [125I]NKA to Neurokinin-2 (NK-2) receptor in rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 62nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-SP to Neurokinin-1 (NK-1) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-SP to Neurokinin-1 (NK-1) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 68nMAssay Description:Concentration required to inhibit the specific binding of [125I]NKA to Neurokinin-2 (NK-2) receptor in rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 71nMAssay Description:Displacement of Eu-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 2 hrs by time resolved fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 73nMAssay Description:Displacement of Eu-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 2 hrs by time resolved fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-SP to Neurokinin-1 (NK-1) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 88nMAssay Description:Displacement of Eu-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 2 hrs by time resolved fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 91nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-SP to Neurokinin-1 (NK-1) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Concentration required to inhibit the specific binding of [125I]NKA to Neurokinin-2 (NK-2) receptor in rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-SP to Neurokinin-1 (NK-1) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Displacement of Eu-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 2 hrs by time resolved fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Concentration required to inhibit the specific binding of [125I]NKA to Neurokinin-2 (NK-2) receptor in rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair