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Found 35 with Last Name = 'choi' and Initial = 'yk'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50254065(CHEMBL513174 | MCL-515 | R(-)-2-methoxy-11-acetylo...)
Affinity DataKi:  18.9nMAssay Description:Displacement of [3H]nemonapride from dopamine D2 receptor in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM84636(CHEMBL27559 | NPA-11-OH-R,(+))
Affinity DataKi:  28.5nMAssay Description:Displacement of [3H]nemonapride from dopamine D2 receptor in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50202291(Acetic acid (R)-6-propyl-5,6,6a,7-tetrahydro-4H-di...)
Affinity DataKi:  72.3nMAssay Description:Displacement of [3H]nemonapride from dopamine D2 receptor in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50254090(CHEMBL468056 | Pentanoic acid (R)-2-methoxy-6-prop...)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]nemonapride from dopamine D2 receptor in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50254064(Acetic acid (R)-2-methoxy-6-methyl-5,6,6a,7-tetrah...)
Affinity DataKi:  165nMAssay Description:Displacement of [3H]nemonapride from dopamine D2 receptor in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50252323((R)-2-Methoxyaporphin-11-yl pentanoate | CHEMBL482...)
Affinity DataKi:  192nMAssay Description:Displacement of [3H]nemonapride from dopamine D2 receptor in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50202292(11-valeryloxynoraporphine | CHEMBL403550 | Pentano...)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]nemonapride from dopamine D2 receptor in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50254064(Acetic acid (R)-2-methoxy-6-methyl-5,6,6a,7-tetrah...)
Affinity DataKi:  526nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM84636(CHEMBL27559 | NPA-11-OH-R,(+))
Affinity DataKi:  699nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50252323((R)-2-Methoxyaporphin-11-yl pentanoate | CHEMBL482...)
Affinity DataKi:  1.48E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50254090(CHEMBL468056 | Pentanoic acid (R)-2-methoxy-6-prop...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50202291(Acetic acid (R)-6-propyl-5,6,6a,7-tetrahydro-4H-di...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50254065(CHEMBL513174 | MCL-515 | R(-)-2-methoxy-11-acetylo...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50202292(11-valeryloxynoraporphine | CHEMBL403550 | Pentano...)
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50147178((Z)-Octadec-9-enoic acid phenylamide | CHEMBL15611...)
Affinity DataIC50:  140nMAssay Description:Concentration of the compound required to inhibit Acyl coenzyme A:cholesterol acyltransferase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50147178((Z)-Octadec-9-enoic acid phenylamide | CHEMBL15611...)
Affinity DataIC50:  170nMAssay Description:Concentration of the compound required to inhibit Acyl coenzyme A:cholesterol acyltransferase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50150482(Acetic acid 3-acetoxy-4-acetoxymethyl-12-hydroxy-4...)
Affinity DataIC50:  640nMAssay Description:In vitro inhibitory concentration against human Acyl coenzyme A:cholesterol acyltransferase 2 expressed in Hi5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50147176(1-(3,4-Dimethoxy-phenyl)-2-[4-((2S,3R,4R,5S)-5-{4-...)
Affinity DataIC50:  8.00E+3nMAssay Description:Concentration of the compound required to inhibit Acyl coenzyme A:cholesterol acyltransferase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50147176(1-(3,4-Dimethoxy-phenyl)-2-[4-((2S,3R,4R,5S)-5-{4-...)
Affinity DataIC50:  8.00E+3nMAssay Description:In vitro inhibitory concentration against human Acyl coenzyme A:cholesterol acyltransferase 2 expressed in Hi5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50348088(CHEMBL78920)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of GST-tagged PHD2 assessed as inhibition of hydroxylation of fluorescein-labeled HIF1alpha CODD peptide after 1 hr by fluorescent polariz...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50158058(5-(2-{4-[(2S,3R,4S,5R)-5-(3,4-Dimethoxy-phenyl)-3,...)
Affinity DataIC50:  1.40E+4nMAssay Description:In vitro inhibitory concentration against human Acyl coenzyme A:cholesterol acyltransferase 1 expressed in Hi5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50158062(5-(1-Butoxy-2-{4-[(2S,3R,4S,5R)-5-(3,4-dimethoxy-p...)
Affinity DataIC50:  1.70E+4nMAssay Description:In vitro inhibitory concentration against human Acyl coenzyme A:cholesterol acyltransferase 1 expressed in Hi5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50158061(5-(2-{4-[(2S,3R,4S,5R)-5-(3,4-Dimethoxy-phenyl)-3,...)
Affinity DataIC50:  2.00E+4nMAssay Description:In vitro inhibitory concentration against human Acyl coenzyme A:cholesterol acyltransferase 1 expressed in Hi5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50158057(5-(2-{4-[(2S,3R,4S,5R)-5-(3,4-Dimethoxy-phenyl)-3,...)
Affinity DataIC50:  3.10E+4nMAssay Description:In vitro inhibitory concentration against human Acyl coenzyme A:cholesterol acyltransferase 1 expressed in Hi5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50158060(5-(2-{4-[(2S,3R,4S,5R)-5-(3,4-Dimethoxy-phenyl)-3,...)
Affinity DataIC50:  3.40E+4nMAssay Description:In vitro inhibitory concentration against human Acyl coenzyme A:cholesterol acyltransferase 1 expressed in Hi5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50158063(5-(2-{4-[(2S,3R,4S,5R)-5-(3,4-Dimethoxy-phenyl)-3,...)
Affinity DataIC50:  3.50E+4nMAssay Description:In vitro inhibitory concentration against human Acyl coenzyme A:cholesterol acyltransferase 1 expressed in Hi5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50147176(1-(3,4-Dimethoxy-phenyl)-2-[4-((2S,3R,4R,5S)-5-{4-...)
Affinity DataIC50:  3.90E+4nMAssay Description:Concentration of the compound required to inhibit Acyl coenzyme A:cholesterol acyltransferase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50147176(1-(3,4-Dimethoxy-phenyl)-2-[4-((2S,3R,4R,5S)-5-{4-...)
Affinity DataIC50:  3.90E+4nMAssay Description:In vitro inhibitory concentration against human Acyl coenzyme A:cholesterol acyltransferase 1 expressed in Hi5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50158059(1-Benzo[1,3]dioxol-5-yl-2-{4-[(2S,3R,4S,5R)-5-(3,4...)
Affinity DataIC50:  4.30E+4nMAssay Description:In vitro inhibitory concentration against human Acyl coenzyme A:cholesterol acyltransferase 1 expressed in Hi5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50147179(5-((R)-2-{4-[(2S,3R,4S,5R)-5-(3,4-Dimethoxy-phenyl...)
Affinity DataIC50:  4.30E+4nMAssay Description:Concentration of the compound required to inhibit Acyl coenzyme A:cholesterol acyltransferase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50158056(5-(2-{4-[(2S,3R,4S,5R)-5-(3,4-Dimethoxy-phenyl)-3,...)
Affinity DataIC50:  5.00E+4nMAssay Description:In vitro inhibitory concentration against human Acyl coenzyme A:cholesterol acyltransferase 1 expressed in Hi5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50348089(CHEMBL1800368)
Affinity DataIC50:  6.97E+4nMAssay Description:Inhibition of GST-tagged PHD2 assessed as inhibition of hydroxylation of fluorescein-labeled HIF1alpha CODD peptide after 1 hr by fluorescent polariz...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50147177(2-(4-{(2S,3R,4R,5S)-5-[4-(2-Benzo[1,3]dioxol-5-yl-...)
Affinity DataIC50:  8.20E+4nMAssay Description:Concentration of the compound required to inhibit Acyl coenzyme A:cholesterol acyltransferase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50147177(2-(4-{(2S,3R,4R,5S)-5-[4-(2-Benzo[1,3]dioxol-5-yl-...)
Affinity DataIC50:  8.20E+4nMAssay Description:In vitro inhibitory concentration against human Acyl coenzyme A:cholesterol acyltransferase 1 expressed in Hi5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50147179(5-((R)-2-{4-[(2S,3R,4S,5R)-5-(3,4-Dimethoxy-phenyl...)
Affinity DataIC50:  1.24E+5nMAssay Description:Concentration of the compound required to inhibit Acyl coenzyme A:cholesterol acyltransferase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed