Compile Data Set for Download or QSAR
maximum 50k data
Found 266 with Last Name = 'cichy-knight' and Initial = 'm'
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064027(5-{(2S,3S,4R,5R,6S)-3,4-Bis-benzyloxy-5-(1H-imidaz...)
Affinity DataKi:  100nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064027(5-{(2S,3S,4R,5R,6S)-3,4-Bis-benzyloxy-5-(1H-imidaz...)
Affinity DataKi:  300nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064025(CHEMBL282129 | N*1*-{(2R,3R,4S,5R,6R)-3,4,5-Tris-b...)
Affinity DataKi:  500nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064025(CHEMBL282129 | N*1*-{(2R,3R,4S,5R,6R)-3,4,5-Tris-b...)
Affinity DataKi:  600nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064025(CHEMBL282129 | N*1*-{(2R,3R,4S,5R,6R)-3,4,5-Tris-b...)
Affinity DataKi:  600nMAssay Description:Binding affinity for human receptor subtype hSSTR3.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064027(5-{(2S,3S,4R,5R,6S)-3,4-Bis-benzyloxy-5-(1H-imidaz...)
Affinity DataKi:  800nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064027(5-{(2S,3S,4R,5R,6S)-3,4-Bis-benzyloxy-5-(1H-imidaz...)
Affinity DataKi:  900nMAssay Description:Binding affinity for human receptor subtype hSSTR3.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50051567(5-{(2R,3R,4S,5R,6R)-3,4,5-Tris-benzyloxy-6-[2-(1H-...)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064025(CHEMBL282129 | N*1*-{(2R,3R,4S,5R,6R)-3,4,5-Tris-b...)
Affinity DataKi:  1.30E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR5.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50051578(5-{(2R,3S,5R,6R)-3,5-Bis-benzyloxy-6-[2-(1H-indol-...)
Affinity DataKi:  1.70E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50051567(5-{(2R,3R,4S,5R,6R)-3,4,5-Tris-benzyloxy-6-[2-(1H-...)
Affinity DataKi:  1.80E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064024(5-{(2S,3S,4R,5R,6S)-3,4,5-Tris-benzyloxy-6-[2-(1H-...)
Affinity DataKi:  1.90E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064030(5-((2R,3R,4S,5R,6R)-3,4,5-Tris-benzyloxy-6-methoxy...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064026(5-{(2S,3S,4R,5S,6S)-3,4,5-Tris-benzyloxy-6-[2-(1H-...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064025(CHEMBL282129 | N*1*-{(2R,3R,4S,5R,6R)-3,4,5-Tris-b...)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064030(5-((2R,3R,4S,5R,6R)-3,4,5-Tris-benzyloxy-6-methoxy...)
Affinity DataKi:  2.40E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064024(5-{(2S,3S,4R,5R,6S)-3,4,5-Tris-benzyloxy-6-[2-(1H-...)
Affinity DataKi:  2.60E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064026(5-{(2S,3S,4R,5S,6S)-3,4,5-Tris-benzyloxy-6-[2-(1H-...)
Affinity DataKi:  2.70E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50051567(5-{(2R,3R,4S,5R,6R)-3,4,5-Tris-benzyloxy-6-[2-(1H-...)
Affinity DataKi:  2.80E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR3.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064030(5-((2R,3R,4S,5R,6R)-3,4,5-Tris-benzyloxy-6-methoxy...)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR5.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064029(5-{(2R,3S,5R,6R)-3-Benzyloxy-5-(1H-imidazol-4-ylme...)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064030(5-((2R,3R,4S,5R,6R)-3,4,5-Tris-benzyloxy-6-methoxy...)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR3.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50051578(5-{(2R,3S,5R,6R)-3,5-Bis-benzyloxy-6-[2-(1H-indol-...)
Affinity DataKi:  3.10E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064024(5-{(2S,3S,4R,5R,6S)-3,4,5-Tris-benzyloxy-6-[2-(1H-...)
Affinity DataKi:  3.30E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR3.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50051578(5-{(2R,3S,5R,6R)-3,5-Bis-benzyloxy-6-[2-(1H-indol-...)
Affinity DataKi:  3.30E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR3.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064026(5-{(2S,3S,4R,5S,6S)-3,4,5-Tris-benzyloxy-6-[2-(1H-...)
Affinity DataKi:  3.40E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR5.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50051567(5-{(2R,3R,4S,5R,6R)-3,4,5-Tris-benzyloxy-6-[2-(1H-...)
Affinity DataKi:  3.70E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR5.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064024(5-{(2S,3S,4R,5R,6S)-3,4,5-Tris-benzyloxy-6-[2-(1H-...)
Affinity DataKi:  3.90E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR5.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064024(5-{(2S,3S,4R,5R,6S)-3,4,5-Tris-benzyloxy-6-[2-(1H-...)
Affinity DataKi:  4.00E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50051567(5-{(2R,3R,4S,5R,6R)-3,4,5-Tris-benzyloxy-6-[2-(1H-...)
Affinity DataKi:  4.00E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064029(5-{(2R,3S,5R,6R)-3-Benzyloxy-5-(1H-imidazol-4-ylme...)
Affinity DataKi:  4.00E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR5.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50051578(5-{(2R,3S,5R,6R)-3,5-Bis-benzyloxy-6-[2-(1H-indol-...)
Affinity DataKi:  4.10E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064026(5-{(2S,3S,4R,5S,6S)-3,4,5-Tris-benzyloxy-6-[2-(1H-...)
Affinity DataKi:  4.40E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064029(5-{(2R,3S,5R,6R)-3-Benzyloxy-5-(1H-imidazol-4-ylme...)
Affinity DataKi:  4.60E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064030(5-((2R,3R,4S,5R,6R)-3,4,5-Tris-benzyloxy-6-methoxy...)
Affinity DataKi:  4.60E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50051578(5-{(2R,3S,5R,6R)-3,5-Bis-benzyloxy-6-[2-(1H-indol-...)
Affinity DataKi:  5.10E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR5.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064029(5-{(2R,3S,5R,6R)-3-Benzyloxy-5-(1H-imidazol-4-ylme...)
Affinity DataKi:  6.20E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR3.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064026(5-{(2S,3S,4R,5S,6S)-3,4,5-Tris-benzyloxy-6-[2-(1H-...)
Affinity DataKi:  6.40E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR3.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064029(5-{(2R,3S,5R,6R)-3-Benzyloxy-5-(1H-imidazol-4-ylme...)
Affinity DataKi:  6.80E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064035((5S,8R,11S,14R,17S,19aS)-5-Benzyl-11-(4-fluoro-ben...)
Affinity DataIC50:  2nMAssay Description:Binding affinity was measured for Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50407836(CHEMBL2112240)
Affinity DataIC50:  2nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50407838(CHEMBL2112243)
Affinity DataIC50:  15nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50064032(CHEMBL29161 | N-(5-{(2R,3R,4S,5R,6R)-4,5-Bis-benzy...)
Affinity DataIC50:  27nMAssay Description:Binding affinity was measured for Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50407835(CHEMBL2112242)
Affinity DataIC50:  28nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50407839(CHEMBL2112244)
Affinity DataIC50:  35nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLipoprotein lipase(Rattus norvegicus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50254432(1-(2-methyl-5-(morpholinosulfonyl)furan-3-yl)-3-ph...)
Affinity DataIC50:  40nMAssay Description:Inhibition of Lipoprotein lipase from adipose tissue of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLipoprotein lipase(Rattus norvegicus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50254434(5-Methyl-4-(3-phenyl-ureido)-furan-2-sulfonic acid...)
Affinity DataIC50:  50nMAssay Description:Inhibition of Lipoprotein lipase from adipose tissue of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50407840(CHEMBL2112241)
Affinity DataIC50:  59nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50254343((S)-1-(2-methyl-5-(piperidin-1-ylsulfonyl)furan-3-...)
Affinity DataIC50:  60nMAssay Description:Inhibition of endothelial lipase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50051573(CHEMBL420221 | N-(5-{(2R,3R,4S,5R,6R)-3,4,5-Tris-b...)
Affinity DataIC50:  60nMAssay Description:Binding affinity towards Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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