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Found 129 with Last Name = 'coates' and Initial = 'ja'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM591((2R,4S)-2-[(R)-(benzylcarbamoyl)(1-phenylacetamido...)
Affinity DataIC50:  0.900nMAssay Description:Inhibitory activity towards HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321697(1-allyl-1-(1-(((3S,4R)-1-(cyclopentanecarbonyl)-4-...)
Affinity DataIC50:  1.10nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321683(4-chlorobenzyl allyl(1-(((3S,4R)-1-(cyclopentaneca...)
Affinity DataIC50:  1.10nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50325319(1-allyl-1-(1-(((3S,4R)-1-(cyclopentanecarbonyl)-4-...)
Affinity DataIC50:  1.38nMAssay Description:Inhibition of human CCR5 expressed in CHO cells assessed as inhibition of RANTES-stimulated [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321712(CHEMBL1172625 | N-allyl-N-(1-(((3S,4R)-1-(cyclopen...)
Affinity DataIC50:  1.5nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321699(1-allyl-1-(1-(((3S,4R)-1-(cyclopentanecarbonyl)-4-...)
Affinity DataIC50:  1.60nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321700(1-allyl-1-(1-(((3S,4R)-1-(cyclopentanecarbonyl)-4-...)
Affinity DataIC50:  1.70nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321694(1-allyl-1-(1-(((3S,4R)-1-(cyclopentanecarbonyl)-4-...)
Affinity DataIC50:  1.70nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321711(CHEMBL1172624 | N-allyl-N-(1-(((3S,4R)-1-(cyclopen...)
Affinity DataIC50:  2.10nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321695(1-allyl-3-(4-chlorobenzyl)-1-(1-(((3S,4R)-1-(cyclo...)
Affinity DataIC50:  2.70nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321682(CHEMBL1172035 | nifeviroc)
Affinity DataIC50:  2.90nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321701(4-((3-allyl-3-(1-(((3S,4R)-1-(cyclopentanecarbonyl...)
Affinity DataIC50:  2.90nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321682(CHEMBL1172035 | nifeviroc)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of human CCR5 expressed in CHO cells assessed as inhibition of RANTES-stimulated [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50325321(CHEMBL1222771 | N-allyl-N-(1-(((3S,4R)-1-(cyclopen...)
Affinity DataIC50:  2.98nMAssay Description:Inhibition of human CCR5 expressed in CHO cells assessed as inhibition of RANTES-stimulated [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM589((2R,4S)-2-[(R)-carbamoyl(1-phenylacetamido)methyl]...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity towards HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321696(1-allyl-1-(1-(((3S,4R)-1-(cyclopentanecarbonyl)-4-...)
Affinity DataIC50:  3.20nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321713(CHEMBL1172626 | N-allyl-N-(1-(((3S,4R)-1-(cyclopen...)
Affinity DataIC50:  3.30nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321682(CHEMBL1172035 | nifeviroc)
Affinity DataIC50:  3.5nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced calcium elevationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321703(CHEMBL1172157 | N-allyl-N-(1-(((3S,4R)-1-(cyclopen...)
Affinity DataIC50:  3.5nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321707(CHEMBL1171030 | N-allyl-2-(4-chlorophenyl)-N-(1-((...)
Affinity DataIC50:  3.60nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50325325(4-((3-allyl-3-((1R,3S,5S)-8-(((3S,4R)-1-(cyclopent...)
Affinity DataIC50:  3.98nMAssay Description:Inhibition of human CCR5 expressed in CHO cells assessed as inhibition of RANTES-stimulated [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321710(CHEMBL1172623 | N-allyl-N-(1-(((3S,4R)-1-(cyclopen...)
Affinity DataIC50:  4nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM590((2R,4S)-2-[(R)-(ethylcarbamoyl)(1-phenylacetamido)...)
Affinity DataIC50:  4.80nMAssay Description:Inhibitory activity towards HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321702(4-((3-allyl-3-(1-(((3S,4R)-1-(cyclopentanecarbonyl...)
Affinity DataIC50:  5nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321705(CHEMBL1172439 | N-allyl-N-(1-(((3S,4R)-1-(cyclopen...)
Affinity DataIC50:  5.30nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321691(4-methoxybenzyl allyl(1-(((3S,4R)-1-(cyclopentanec...)
Affinity DataIC50:  6.20nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321698(1-allyl-1-(1-(((3S,4R)-1-(cyclopentanecarbonyl)-4-...)
Affinity DataIC50:  6.20nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321685(4-(trifluoromethoxy)benzyl allyl(1-(((3S,4R)-1-(cy...)
Affinity DataIC50:  6.20nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50325322(1-allyl-1-((1R,3S,5S)-8-(((3S,4R)-1-(cyclopentanec...)
Affinity DataIC50:  6.77nMAssay Description:Inhibition of human CCR5 expressed in CHO cells assessed as inhibition of RANTES-stimulated [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321692(CHEMBL1171965 | benzyl allyl(1-(((3S,4R)-1-(cyclop...)
Affinity DataIC50:  8.80nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50325317(4-nitrobenzyl allyl(1-(((3S,4R)-1-(cyclopentanecar...)
Affinity DataIC50:  8.85nMAssay Description:Inhibition of human CCR5 expressed in CHO cells assessed as inhibition of RANTES-stimulated [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321706(CHEMBL1171029 | N-allyl-N-(1-(((3S,4R)-1-(cyclopen...)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50325320(CHEMBL1222770 | N-allyl-N-(1-(((3S,4R)-1-(cyclopen...)
Affinity DataIC50:  11.2nMAssay Description:Inhibition of human CCR5 expressed in CHO cells assessed as inhibition of RANTES-stimulated [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50325323(4-((3-allyl-3-((1R,3S,5S)-8-(((3S,4R)-1-(cyclopent...)
Affinity DataIC50:  11.4nMAssay Description:Inhibition of human CCR5 expressed in CHO cells assessed as inhibition of RANTES-stimulated [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50325326(1-allyl-1-((1R,3R,5S)-8-(((3S,4R)-1-(cyclopentanec...)
Affinity DataIC50:  14.3nMAssay Description:Inhibition of human CCR5 expressed in CHO cells assessed as inhibition of RANTES-stimulated [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321704(CHEMBL1172438 | N-allyl-N-(1-(((3S,4R)-1-(cyclopen...)
Affinity DataIC50:  15nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321708(CHEMBL1169819 | N-allyl-2-(4-bromophenyl)-N-(1-(((...)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321688(4-bromobenzyl allyl(1-(((3S,4R)-1-(cyclopentanecar...)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Avexa

Curated by ChEMBL
LigandPNGBDBM50482807(CHEMBL1222998)
Affinity DataIC50:  20nMAssay Description:Inhibition of HIV-1 integrase-mediated 3'-processing and strand transfer activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Avexa

Curated by ChEMBL
LigandPNGBDBM50479890(CHEMBL522653)
Affinity DataIC50:  25nMAssay Description:Inhibition of HIV1 integrase 3'-strand transferMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50325327(4-((3-allyl-3-((1R,3R,5S)-8-(((3S,4R)-1-(cyclopent...)
Affinity DataIC50:  27.1nMAssay Description:Inhibition of human CCR5 expressed in CHO cells assessed as inhibition of RANTES-stimulated [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321689(4-(trifluoromethyl)benzyl allyl(1-(((3S,4R)-1-(cyc...)
Affinity DataIC50: >30nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50325324(1-allyl-1-((1R,3S,5S)-8-(((3S,4R)-1-(cyclopentanec...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human CCR5 expressed in CHO cells assessed as inhibition of RANTES-stimulated [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50325316(4-nitrobenzyl allyl(1-(((3S,4R)-1-(cyclopentanecar...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human CCR5 expressed in CHO cells assessed as inhibition of RANTES-stimulated [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Avexa

Curated by ChEMBL
LigandPNGBDBM50482815(CHEMBL1258726)
Affinity DataIC50:  35nMAssay Description:Inhibition of HIV-1 integrase-mediated 3'-processing and strand transfer activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Avexa

Curated by ChEMBL
LigandPNGBDBM50482808(CHEMBL1222997)
Affinity DataIC50:  36nMAssay Description:Inhibition of HIV-1 integrase-mediated 3'-processing and strand transfer activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321686(4-(methylsulfonyl)benzyl allyl(1-(((3S,4R)-1-(cycl...)
Affinity DataIC50:  37nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50321693(1-allyl-3-benzyl-1-(1-(((3S,4R)-1-(cyclopentanecar...)
Affinity DataIC50:  38nMAssay Description:Antagonist activity at CCR5 expressed in CHO cells assessed as inhibition of RANTES-induced [35S]GTPgamma binding by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50325318(1-allyl-1-(1-(((3S,4R)-1-(cyclopentanecarbonyl)-4-...)
Affinity DataIC50:  38.3nMAssay Description:Inhibition of human CCR5 expressed in CHO cells assessed as inhibition of RANTES-stimulated [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Avexa

Curated by ChEMBL
LigandPNGBDBM50482809(CHEMBL1222999)
Affinity DataIC50:  42nMAssay Description:Inhibition of HIV-1 integrase-mediated 3'-processing and strand transfer activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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