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Found 30 with Last Name = 'connell' and Initial = 'mj'
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50119774(1,1'-(dodecane-1,12-diyl)bis(3-methylpyridinium)br...)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at nAChRalpha6beta2 in Sprague-Dawley rat striatal slices assessed as inhibition of nicotine-evoked [3H]dopamine uptake by liquid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50470256(CHEMBL86200)
Affinity DataIC50:  22nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230226(CHEMBL144015)
Affinity DataIC50:  40nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230281(CHEMBL144682)
Affinity DataIC50:  48nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50470255(CHEMBL87298)
Affinity DataIC50:  62nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50470254(CHEMBL313940)
Affinity DataIC50:  67nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50470258(CHEMBL87448)
Affinity DataIC50:  83nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230227(CHEMBL356549)
Affinity DataIC50:  140nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230235(CHEMBL144395)
Affinity DataIC50:  140nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230228(CHEMBL144154)
Affinity DataIC50:  160nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230229(CHEMBL144190)
Affinity DataIC50:  170nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230225(CHEMBL144713)
Affinity DataIC50:  230nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50470257(CHEMBL87191)
Affinity DataIC50:  240nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230231(CHEMBL556516)
Affinity DataIC50:  300nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50470259(CHEMBL313681)
Affinity DataIC50:  330nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM15296(6-methyl-2-oxo-5-(pyridin-4-yl)-1,2-dihydropyridin...)
Affinity DataIC50:  360nMAssay Description:Inhibition of cAMP Phosphodiesterase 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50470253(CHEMBL83014)
Affinity DataIC50:  430nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230222(Medorinone | WIN-49016)
Affinity DataIC50:  550nMAssay Description:Inhibition of cAMP PDE 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230237(CHEMBL357234)
Affinity DataIC50:  570nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230238(CHEMBL356805)
Affinity DataIC50:  600nMAssay Description:Inhibition of cAMP Phosphodiesterase 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230223(CHEMBL144453)
Affinity DataIC50:  940nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230279(CHEMBL144706)
Affinity DataIC50:  960nMAssay Description:Inhibition of cAMP Phosphodiesterase 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230239(CHEMBL343895)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230232(CHEMBL145429)
Affinity DataIC50:  1.42E+3nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230224(CHEMBL147736)
Affinity DataIC50:  2.20E+3nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230280(CHEMBL142834)
Affinity DataIC50:  2.80E+3nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230236(CHEMBL2112000)
Affinity DataIC50:  3.10E+3nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230234(CHEMBL356143)
Affinity DataIC50:  3.20E+3nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230233(CHEMBL145024)
Affinity DataIC50:  3.70E+3nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50230230(CHEMBL422303)
Affinity DataIC50:  1.88E+4nMAssay Description:In vitro inhibitory activity against cAMP PDE III.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed