Compile Data Set for Download or QSAR
maximum 50k data
Found 222 with Last Name = 'corso' and Initial = 'g'
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50265993(CHEMBL451230 | phenyl 4-(4,5-dihydro-1H-imidazol-2...)
Affinity DataKi:  1.38E+3nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240366(2-(naphthalen-2-yl)-4,5-dihydro-1H-imidazole | 2-N...)
Affinity DataKi:  1.49E+3nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50086502(2-BFi | 2-Benzofuran-2-yl-4,5-dihydro-1H-imidazole...)
Affinity DataKi:  3.63E+3nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266030(2-(2,4-dichlorophenyl)-4,5-dihydro-1H-imidazole | ...)
Affinity DataKi:  3.98E+3nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240365(2-(4,5-Dihydro-1H-imidazol-2-yl)-quinoline | 2-(4,...)
Affinity DataKi:  4.86E+3nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240365(2-(4,5-Dihydro-1H-imidazol-2-yl)-quinoline | 2-(4,...)
Affinity DataKi:  5.32E+3nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266028(2-(4-chlorophenyl)-4,5-dihydro-1H-imidazole | CHEM...)
Affinity DataKi:  5.35E+3nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50265993(CHEMBL451230 | phenyl 4-(4,5-dihydro-1H-imidazol-2...)
Affinity DataKi:  1.28E+4nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240362(2-p-tolyl-4,5-dihydro-1H-imidazole | CHEMBL269197)
Affinity DataKi:  1.31E+4nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50265991(2-(3,4-dimethoxyphenyl)-4,5-dihydro-1H-imidazole |...)
Affinity DataKi:  1.36E+4nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240366(2-(naphthalen-2-yl)-4,5-dihydro-1H-imidazole | 2-N...)
Affinity DataKi:  1.39E+4nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240364(2-(4-Methoxy-phenyl)-4,5-dihydro-1H-imidazole | 2-...)
Affinity DataKi:  1.58E+4nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266032(2-(3-nitrophenyl)-4,5-dihydro-1H-imidazole | CHEMB...)
Affinity DataKi:  1.93E+4nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240363(2-Phenyl-4,5-dihydro-1H-imidazole | CHEMBL274548)
Affinity DataKi:  2.13E+4nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266029(2-(2-chlorophenyl)-4,5-dihydro-1H-imidazole | CHEM...)
Affinity DataKi:  2.46E+4nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50086502(2-BFi | 2-Benzofuran-2-yl-4,5-dihydro-1H-imidazole...)
Affinity DataKi:  2.49E+4nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240368(2-(4,5-Dihydro-1H-imidazol-2-yl)-pyridine | 2-(4,5...)
Affinity DataKi:  2.53E+4nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50086502(2-BFi | 2-Benzofuran-2-yl-4,5-dihydro-1H-imidazole...)
Affinity DataKi:  2.60E+4nMAssay Description:Binding affinity to human MAOB imidazoline binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266030(2-(2,4-dichlorophenyl)-4,5-dihydro-1H-imidazole | ...)
Affinity DataKi:  2.88E+4nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240363(2-Phenyl-4,5-dihydro-1H-imidazole | CHEMBL274548)
Affinity DataKi:  2.88E+4nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240364(2-(4-Methoxy-phenyl)-4,5-dihydro-1H-imidazole | 2-...)
Affinity DataKi:  3.27E+4nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240362(2-p-tolyl-4,5-dihydro-1H-imidazole | CHEMBL269197)
Affinity DataKi:  1.02E+5nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50265992(2-(3,4,5-trimethoxyphenyl)-4,5-dihydro-1H-imidazol...)
Affinity DataKi:  1.14E+5nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266028(2-(4-chlorophenyl)-4,5-dihydro-1H-imidazole | CHEM...)
Affinity DataKi:  1.66E+5nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266031(2-(4-nitrophenyl)-4,5-dihydro-1H-imidazole | CHEMB...)
Affinity DataKi:  1.81E+5nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50138501(2-(furan-2-yl)-4,5-dihydro-1H-imidazole | 2-Furan-...)
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266031(2-(4-nitrophenyl)-4,5-dihydro-1H-imidazole | CHEMB...)
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50265991(2-(3,4-dimethoxyphenyl)-4,5-dihydro-1H-imidazole |...)
Affinity DataKi:  1.00E+6nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50240368(2-(4,5-Dihydro-1H-imidazol-2-yl)-pyridine | 2-(4,5...)
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50265992(2-(3,4,5-trimethoxyphenyl)-4,5-dihydro-1H-imidazol...)
Affinity DataKi:  1.00E+6nMAssay Description:Binding affinity to MAOB imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266029(2-(2-chlorophenyl)-4,5-dihydro-1H-imidazole | CHEM...)
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50266032(2-(3-nitrophenyl)-4,5-dihydro-1H-imidazole | CHEMB...)
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade Federal De Santa Maria

Curated by ChEMBL
LigandPNGBDBM50138501(2-(furan-2-yl)-4,5-dihydro-1H-imidazole | 2-Furan-...)
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity to MAOA imidazoline binding site in rat brain mitochondrial homogenate assessed as 4-hydroxyquinoline production by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Angelini

Curated by ChEMBL
LigandPNGBDBM50518949(CHEMBL4448131)
Affinity DataIC50:  8nMAssay Description:Inhibition of Staphylococcus aureus DNA gyraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Angelini

Curated by ChEMBL
LigandPNGBDBM50359538(CHEMBL1235773)
Affinity DataIC50:  14nMAssay Description:Inhibition of Staphylococcus aureus DNA gyraseMore data for this Ligand-Target Pair
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Angelini

Curated by ChEMBL
LigandPNGBDBM50518919(CHEMBL4575906)
Affinity DataIC50:  20nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as reduction in enzyme-mediated supercoiling of relaxed plasmid by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A(Staphylococcus aureus)
Angelini

Curated by ChEMBL
LigandPNGBDBM50518915(CHEMBL4583368)
Affinity DataIC50:  20nMAssay Description:Inhibition of Staphylococcus aureus ATCC 29213 DNA gyrase A assessed as reduction in enzyme-mediated supercoiling of relaxed pBR322 DNA by ethidium b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A(Staphylococcus aureus)
Angelini

Curated by ChEMBL
LigandPNGBDBM50518940(CHEMBL4541988)
Affinity DataIC50:  20nMAssay Description:Inhibition of Staphylococcus aureus ATCC 29213 DNA gyrase A assessed as reduction in enzyme-mediated supercoiling of relaxed pBR322 DNA by ethidium b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 4 subunit A(Staphylococcus aureus)
Angelini

Curated by ChEMBL
LigandPNGBDBM50518915(CHEMBL4583368)
Affinity DataIC50:  40nMAssay Description:Inhibition of Staphylococcus aureus ATCC 29213 DNA topoisomerase 4 subunit ParC assessed as reduction in decatenation of kinetoplast DNA incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Angelini

Curated by ChEMBL
LigandPNGBDBM50518948(CHEMBL4574863)
Affinity DataIC50:  40nMAssay Description:Inhibition of Escherichia coli ATCC 25922 DNA gyrase A assessed as reduction in enzyme-mediated supercoiling of relaxed pBR322 DNA by ethidium bromid...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Angelini

Curated by ChEMBL
LigandPNGBDBM50050549(GSK2140944 | Gepotidacin)
Affinity DataIC50:  47nMAssay Description:Inhibition of Staphylococcus aureus DNA gyraseMore data for this Ligand-Target Pair
TargetDNA topoisomerase 4 subunit A(Staphylococcus aureus)
Angelini

Curated by ChEMBL
LigandPNGBDBM50518940(CHEMBL4541988)
Affinity DataIC50:  50nMAssay Description:Inhibition of Staphylococcus aureus ATCC 29213 DNA topoisomerase 4 subunit ParC assessed as reduction in decatenation of kinetoplast DNA incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Angelini

Curated by ChEMBL
LigandPNGBDBM50518915(CHEMBL4583368)
Affinity DataIC50:  100nMAssay Description:Inhibition of Escherichia coli ATCC 25922 DNA gyrase A assessed as reduction in enzyme-mediated supercoiling of relaxed pBR322 DNA by ethidium bromid...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A(Staphylococcus aureus)
Angelini

Curated by ChEMBL
LigandPNGBDBM50518948(CHEMBL4574863)
Affinity DataIC50: <100nMAssay Description:Inhibition of Staphylococcus aureus ATCC 29213 DNA gyrase A assessed as reduction in enzyme-mediated supercoiling of relaxed pBR322 DNA by ethidium b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Angelini

Curated by ChEMBL
LigandPNGBDBM50359538(CHEMBL1235773)
Affinity DataIC50:  100nMAssay Description:Inhibition of Escherichia coli DNA gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 4 subunit A(Escherichia coli (strain K12))
Angelini

Curated by ChEMBL
LigandPNGBDBM50518915(CHEMBL4583368)
Affinity DataIC50:  100nMAssay Description:Inhibition of Escherichia coli ATCC 25922 DNA topoisomerase 4 subunit ParC assessed as reduction in decatenation of kinetoplast DNA incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 4 subunit A(Escherichia coli (strain K12))
Angelini

Curated by ChEMBL
LigandPNGBDBM50518948(CHEMBL4574863)
Affinity DataIC50:  100nMAssay Description:Inhibition of Escherichia coli ATCC 25922 DNA topoisomerase 4 subunit ParC assessed as reduction in decatenation of kinetoplast DNA incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 4 subunit A(Escherichia coli (strain K12))
Angelini

Curated by ChEMBL
LigandPNGBDBM50518940(CHEMBL4541988)
Affinity DataIC50:  100nMAssay Description:Inhibition of Escherichia coli ATCC 25922 DNA topoisomerase 4 subunit ParC assessed as reduction in decatenation of kinetoplast DNA incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 4 subunit A(Staphylococcus aureus)
Angelini

Curated by ChEMBL
LigandPNGBDBM50518948(CHEMBL4574863)
Affinity DataIC50: <100nMAssay Description:Inhibition of Staphylococcus aureus ATCC 29213 DNA topoisomerase 4 subunit ParC assessed as reduction in decatenation of kinetoplast DNA incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Angelini

Curated by ChEMBL
LigandPNGBDBM50518949(CHEMBL4448131)
Affinity DataIC50:  125nMAssay Description:Inhibition of Escherichia coli DNA gyraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 222 total ) | Next | Last >>
Jump to: