Compile Data Set for Download or QSAR
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Found 187 with Last Name = 'damonte' and Initial = 'g'
TargetLanC-like protein 2(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50041087(CHEMBL3355910)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of ABA binding to LANCL2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50451276(CHEMBL4217987)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human recombinant SIRT6 assessed as reduction in NAD+-dependent deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50451275(CHEMBL4205716)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of human recombinant SIRT6 assessed as reduction in NAD+-dependent deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50451274(CHEMBL4206619)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of human recombinant SIRT6 assessed as reduction in NAD+-dependent deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50017342(CHEMBL1588664)
Affinity DataIC50:  8.90E+4nMAssay Description:Inhibition of human recombinant SIRT6 assessed as reduction in NAD+-dependent deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50451276(CHEMBL4217987)
Affinity DataIC50:  3.33E+5nMAssay Description:Inhibition of human recombinant SIRT2 assessed as reduction in NAD+-dependent deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50451276(CHEMBL4217987)
Affinity DataIC50:  4.24E+5nMAssay Description:Inhibition of human recombinant SIRT1 assessed as reduction in NAD+-dependent deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50451274(CHEMBL4206619)
Affinity DataIC50:  4.53E+5nMAssay Description:Inhibition of human recombinant SIRT2 assessed as reduction in NAD+-dependent deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50451275(CHEMBL4205716)
Affinity DataIC50:  4.82E+5nMAssay Description:Inhibition of human recombinant SIRT2 assessed as reduction in NAD+-dependent deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50451275(CHEMBL4205716)
Affinity DataIC50:  5.99E+5nMAssay Description:Inhibition of human recombinant SIRT1 assessed as reduction in NAD+-dependent deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50017342(CHEMBL1588664)
Affinity DataIC50:  7.51E+5nMAssay Description:Inhibition of human recombinant SIRT2 assessed as reduction in NAD+-dependent deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50451274(CHEMBL4206619)
Affinity DataIC50:  7.83E+5nMAssay Description:Inhibition of human recombinant SIRT1 assessed as reduction in NAD+-dependent deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50017342(CHEMBL1588664)
Affinity DataIC50:  1.58E+6nMAssay Description:Inhibition of human recombinant SIRT1 assessed as reduction in NAD+-dependent deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108517(CHEMBL3597843)
Affinity DataEC50:  2.70E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50105910(CHEMBL3597907)
Affinity DataEC50:  3.20E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108492(CHEMBL3597874)
Affinity DataEC50:  6.40E+3nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50105911(CHEMBL3597886)
Affinity DataEC50:  5.80E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108496(CHEMBL3597875)
Affinity DataEC50:  7.10E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108513(CHEMBL3597853)
Affinity DataEC50:  5.30E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108350(CHEMBL3597884)
Affinity DataEC50:  9.50E+3nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108483(CHEMBL3597841)
Affinity DataEC50:  3.40E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50105909(CHEMBL3597937)
Affinity DataEC50:  1.50E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108523(CHEMBL3597889)
Affinity DataEC50:  5.70E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as iodide influx after 24 hrs by HS-YFP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108302(CHEMBL3597927)
Affinity DataEC50:  1.40E+4nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as iodide influx after 24 hrs by HS-YFP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108301(CHEMBL3597882)
Affinity DataEC50:  8.50E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as iodide influx after 24 hrs by HS-YFP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108513(CHEMBL3597853)
Affinity DataEC50:  5.30E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as iodide influx after 24 hrs by HS-YFP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289534(CHEMBL2018574)
Affinity DataEC50:  5.90E+3nMAssay Description:Potentiator activity at CFTR F508-del mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289535(CHEMBL4176184)
Affinity DataEC50:  1.60E+4nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289702(CHEMBL3746059)
Affinity DataEC50:  1.40E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289534(CHEMBL2018574)
Affinity DataEC50:  1.50E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289703(Lumacaftor | VRT 826809 | VRT-826809 | VX 809 | VX...)
Affinity DataEC50:  2.60E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin)More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289704(CHEMBL260775)
Affinity DataEC50: <3.00E+3nMAssay Description:Corrector activity at human CFTR F508-del mutant expressed in rat FTR cells harboring YFP-H148Q/I152L preincubated for 18 to 24 hrs followed by forsk...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289705(CHEMBL3745884)
Affinity DataEC50:  2.82E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289706(CHEMBL1257047)
Affinity DataEC50:  2.19E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289704(CHEMBL260775)
Affinity DataEC50:  1.10E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289703(Lumacaftor | VRT 826809 | VRT-826809 | VX 809 | VX...)
Affinity DataEC50:  2.57E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289707(CHEMBL4170223)
Affinity DataEC50:  2.20E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289708(CHEMBL4174717)
Affinity DataEC50:  8.00E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289709(CHEMBL4166815)
Affinity DataEC50:  4.00E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289710(CHEMBL4171265)
Affinity DataEC50:  1.70E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289711(CHEMBL4163361)
Affinity DataEC50:  1.30E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289712(CHEMBL4167920)
Affinity DataEC50:  5.40E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289755(CHEMBL4160001)
Affinity DataEC50:  3.80E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289764(CHEMBL4162319)
Affinity DataEC50:  2.90E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289771(CHEMBL4167675)
Affinity DataEC50: >5.00E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289773(CHEMBL4169748)
Affinity DataEC50:  900nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289774(CHEMBL4161828)
Affinity DataEC50:  1.60E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289779(CHEMBL4166332)
Affinity DataEC50:  2.30E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289853(CHEMBL4176955)
Affinity DataEC50:  1.90E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50289854(CHEMBL4162876)
Affinity DataEC50:  2.90E+3nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin) expressed in human CFBE41o cells harboring HS-YFP preincubated for 24 hrs followed by for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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