Affinity DataKi: 1nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 106nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 167nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 658nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 706nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 2.09E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 3.36E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 4.11E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 7.84E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 9.66E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Amgen
Curated by ChEMBL
Amgen
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-terminal His-tagged PERK expressed in Escherichia coli using AviTag C-terminal, N-terminal His-tagged eIF2alpha (3 to 315) as s...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Amgen
Curated by ChEMBL
Amgen
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-terminal His-tagged PERK expressed in Escherichia coli using AviTag C-terminal, N-terminal His-tagged eIF2alpha (3 to 315) as s...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Amgen
Curated by ChEMBL
Amgen
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of human N-terminal His-tagged PERK expressed in Escherichia coli using AviTag C-terminal, N-terminal His-tagged eIF2alpha (3 to 315) as s...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of PHD2 (unknown origin) by fluorescence energy transfer analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of human PHD2 assesssed as hydroxylation of Pro564 in human HIF-1alpha by TR-FRET assayMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Amgen
Curated by ChEMBL
Amgen
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of human N-terminal His-tagged PERK expressed in Escherichia coli using AviTag C-terminal, N-terminal His-tagged eIF2alpha (3 to 315) as s...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Amgen
Curated by ChEMBL
Amgen
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of human N-terminal His-tagged PERK expressed in Escherichia coli using AviTag C-terminal, N-terminal His-tagged eIF2alpha (3 to 315) as s...More data for this Ligand-Target Pair
TargetCell division cycle 7-related protein kinase/Protein DBF4 homolog A(Homo sapiens (Human))
Amgen
Curated by ChEMBL
Amgen
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Amgen
Curated by ChEMBL
Amgen
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of human N-terminal His-tagged PERK expressed in Escherichia coli using AviTag C-terminal, N-terminal His-tagged eIF2alpha (3 to 315) as s...More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Amgen
Curated by ChEMBL
Amgen
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of human N-terminal His-tagged PERK expressed in Escherichia coli using AviTag C-terminal, N-terminal His-tagged eIF2alpha (3 to 315) as s...More data for this Ligand-Target Pair