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Found 373 with Last Name = 'dao' and Initial = 'j'
TargetProcathepsin L(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137388(((R)-2-Methyl-1-{3-phenyl-1-[(4-piperidin-1-yl-phe...)
Affinity DataKi:  1nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137398(((R)-2-(4-Hydroxy-phenyl)-1-{3-phenyl-1-[(4-piperi...)
Affinity DataKi:  1nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137394(((R)-2-(3H-Indol-3-yl)-1-{3-phenyl-1-[(4-piperidin...)
Affinity DataKi:  1nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137400(((R)-2-Phenyl-1-{3-phenyl-1-[(4-piperidin-1-yl-phe...)
Affinity DataKi:  1nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137392(CHEMBL99195 | [(S)-1-((S)-1-Formyl-3-methylsulfany...)
Affinity DataKi:  1.30nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137393(CHEMBL353725 | {(S)-1-[(S)-1-Benzyl-2-(4-piperidin...)
Affinity DataKi:  2nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137389(((R)-3-Methyl-1-{3-phenyl-1-[(4-piperidin-1-yl-phe...)
Affinity DataKi:  2nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137395(CHEMBL170242 | {(S)-1-[(S)-1-Benzyl-2-(4-morpholin...)
Affinity DataKi:  2nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137400(((R)-2-Phenyl-1-{3-phenyl-1-[(4-piperidin-1-yl-phe...)
Affinity DataKi:  3nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137390(((R)-3-Methylsulfanyl-1-{3-phenyl-1-[(4-piperidin-...)
Affinity DataKi:  3nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137388(((R)-2-Methyl-1-{3-phenyl-1-[(4-piperidin-1-yl-phe...)
Affinity DataKi:  4nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137389(((R)-3-Methyl-1-{3-phenyl-1-[(4-piperidin-1-yl-phe...)
Affinity DataKi:  5nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137388(((R)-2-Methyl-1-{3-phenyl-1-[(4-piperidin-1-yl-phe...)
Affinity DataKi:  7nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137398(((R)-2-(4-Hydroxy-phenyl)-1-{3-phenyl-1-[(4-piperi...)
Affinity DataKi:  8nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137387(((R)-3-Phenyl-1-{3-phenyl-1-[(4-piperidin-1-yl-phe...)
Affinity DataKi:  9nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137391(((R)-1-{3-Phenyl-1-[(4-piperidin-1-yl-phenylamino)...)
Affinity DataKi:  9nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137393(CHEMBL353725 | {(S)-1-[(S)-1-Benzyl-2-(4-piperidin...)
Affinity DataKi:  10nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137386(2-{(S)-3-Phenyl-1-[(4-piperidin-1-yl-phenylamino)-...)
Affinity DataKi:  12nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137390(((R)-3-Methylsulfanyl-1-{3-phenyl-1-[(4-piperidin-...)
Affinity DataKi:  12nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137387(((R)-3-Phenyl-1-{3-phenyl-1-[(4-piperidin-1-yl-phe...)
Affinity DataKi:  14nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137395(CHEMBL170242 | {(S)-1-[(S)-1-Benzyl-2-(4-morpholin...)
Affinity DataKi:  15nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137397(CHEMBL341014 | [(S)-1-((S)-1-Benzyl-2-oxo-ethylcar...)
Affinity DataKi:  20nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137401(CHEMBL171998 | {(S)-1-[(S)-1-Benzyl-2-(biphenyl-4-...)
Affinity DataKi:  32nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137390(((R)-3-Methylsulfanyl-1-{3-phenyl-1-[(4-piperidin-...)
Affinity DataKi:  36nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137394(((R)-2-(3H-Indol-3-yl)-1-{3-phenyl-1-[(4-piperidin...)
Affinity DataKi:  48nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137398(((R)-2-(4-Hydroxy-phenyl)-1-{3-phenyl-1-[(4-piperi...)
Affinity DataKi:  106nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137400(((R)-2-Phenyl-1-{3-phenyl-1-[(4-piperidin-1-yl-phe...)
Affinity DataKi:  167nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137396(CHEMBL423447 | [(S)-1-((S)-1-Benzyl-2-phenylamino-...)
Affinity DataKi:  230nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137389(((R)-3-Methyl-1-{3-phenyl-1-[(4-piperidin-1-yl-phe...)
Affinity DataKi:  658nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137401(CHEMBL171998 | {(S)-1-[(S)-1-Benzyl-2-(biphenyl-4-...)
Affinity DataKi:  706nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137396(CHEMBL423447 | [(S)-1-((S)-1-Benzyl-2-phenylamino-...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137391(((R)-1-{3-Phenyl-1-[(4-piperidin-1-yl-phenylamino)...)
Affinity DataKi:  2.09E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137394(((R)-2-(3H-Indol-3-yl)-1-{3-phenyl-1-[(4-piperidin...)
Affinity DataKi:  3.36E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137391(((R)-1-{3-Phenyl-1-[(4-piperidin-1-yl-phenylamino)...)
Affinity DataKi:  4.11E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137386(2-{(S)-3-Phenyl-1-[(4-piperidin-1-yl-phenylamino)-...)
Affinity DataKi:  7.84E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137387(((R)-3-Phenyl-1-{3-phenyl-1-[(4-piperidin-1-yl-phe...)
Affinity DataKi:  9.66E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137386(2-{(S)-3-Phenyl-1-[(4-piperidin-1-yl-phenylamino)-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137399(({3-Phenyl-1-[(4-piperidin-1-yl-phenylamino)-methy...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137399(({3-Phenyl-1-[(4-piperidin-1-yl-phenylamino)-methy...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50137399(({3-Phenyl-1-[(4-piperidin-1-yl-phenylamino)-methy...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50072072(CHEMBL3407849)
Affinity DataIC50:  1nMAssay Description:Inhibition of human N-terminal His-tagged PERK expressed in Escherichia coli using AviTag C-terminal, N-terminal His-tagged eIF2alpha (3 to 315) as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50072075(CHEMBL3407846)
Affinity DataIC50:  1nMAssay Description:Inhibition of human N-terminal His-tagged PERK expressed in Escherichia coli using AviTag C-terminal, N-terminal His-tagged eIF2alpha (3 to 315) as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50072038(CHEMBL3407863)
Affinity DataIC50:  2nMAssay Description:Inhibition of human N-terminal His-tagged PERK expressed in Escherichia coli using AviTag C-terminal, N-terminal His-tagged eIF2alpha (3 to 315) as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50264220(2-(1,6-diphenyl-1H-imidazo[4,5-c]pyridine-4-carbox...)
Affinity DataIC50:  3nMAssay Description:Inhibition of PHD2 (unknown origin) by fluorescence energy transfer analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50251959(2-(2-(2-(4-tert-butylbenzylsulfonyl)acetamido)-3-h...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human PHD2 assesssed as hydroxylation of Pro564 in human HIF-1alpha by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50072070(CHEMBL3407504)
Affinity DataIC50:  3nMAssay Description:Inhibition of human N-terminal His-tagged PERK expressed in Escherichia coli using AviTag C-terminal, N-terminal His-tagged eIF2alpha (3 to 315) as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50071957(CHEMBL3407850)
Affinity DataIC50:  3nMAssay Description:Inhibition of human N-terminal His-tagged PERK expressed in Escherichia coli using AviTag C-terminal, N-terminal His-tagged eIF2alpha (3 to 315) as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50016163(CHEMBL3261514)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50072073(CHEMBL3407848)
Affinity DataIC50:  4nMAssay Description:Inhibition of human N-terminal His-tagged PERK expressed in Escherichia coli using AviTag C-terminal, N-terminal His-tagged eIF2alpha (3 to 315) as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50072030(CHEMBL3407856)
Affinity DataIC50:  4nMAssay Description:Inhibition of human N-terminal His-tagged PERK expressed in Escherichia coli using AviTag C-terminal, N-terminal His-tagged eIF2alpha (3 to 315) as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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