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Found 268 with Last Name = 'darcq' and Initial = 'e'
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50064751(CHEMBL3403780)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]RTI-33 from GPR88 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50554975(CHEMBL4595209)
Affinity DataKi:  224nMAssay Description:Displacement of [3H]RTI-33 from GPR88 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50065915(CHEMBL3401461)
Affinity DataKi:  277nMAssay Description:Displacement of [3H]RTI-33 from GPR88 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50610306(CHEMBL5285428)
Affinity DataKi:  487nMAssay Description:Displacement of [3H]RTI-33 from GPR88 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50064645(CHEMBL3403768)
Affinity DataKi:  612nMAssay Description:Displacement of [3H]RTI-33 from GPR88 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50506615(CHEMBL4452474)
Affinity DataKi:  750nMAssay Description:Displacement of [3H]-Paroxetine from recombinant human full length SERT after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50506615(CHEMBL4452474)
Affinity DataKi:  2.29E+3nMAssay Description:Binding affinity to human full length KOR after 60 mins by radioligand-based scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50506615(CHEMBL4452474)
Affinity DataIC50:  2.51E+4nMAssay Description:Inhibition of human SERT expressed in HEK293 cells assessed as reduction in SERT-mediated substrate uptake after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506609(CHEMBL4583504)
Affinity DataEC50:  63nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Mus musculus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50065915(CHEMBL3401461)
Affinity DataEC50:  1.14E+3nMAssay Description:Agonist activity at GPR88 in wild type mouse striatal membranes assessed as increase in [35S]-GTPgammaS binding after 1 hr by liquid scintillation co...More data for this Ligand-Target Pair
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506610(CHEMBL4550415)
Affinity DataEC50:  126nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50065915(CHEMBL3401461)
Affinity DataEC50:  126nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506611(CHEMBL4464331)
Affinity DataEC50:  501nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506612(CHEMBL4454531)
Affinity DataEC50:  398nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506613(CHEMBL4453972)
Affinity DataEC50:  316nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506614(CHEMBL4454851)
Affinity DataEC50:  126nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506610(CHEMBL4550415)
Affinity DataEC50:  126nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506615(CHEMBL4452474)
Affinity DataEC50:  100nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Mus musculus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50506615(CHEMBL4452474)
Affinity DataEC50:  535nMAssay Description:Agonist activity at GPR88 in wild type mouse striatal membranes assessed as increase in [35S]-GTPgammaS binding after 1 hr by liquid scintillation co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506613(CHEMBL4453972)
Affinity DataEC50:  316nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506616(CHEMBL4443664)
Affinity DataEC50:  158nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506614(CHEMBL4454851)
Affinity DataEC50:  126nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506615(CHEMBL4452474)
Affinity DataEC50:  100nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506615(CHEMBL4452474)
Affinity DataEC50:  100nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506617(CHEMBL4513479)
Affinity DataEC50:  501nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506609(CHEMBL4583504)
Affinity DataEC50:  63nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506617(CHEMBL4513479)
Affinity DataEC50:  501nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506618(CHEMBL4587388)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506612(CHEMBL4454531)
Affinity DataEC50:  398nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50065915(CHEMBL3401461)
Affinity DataEC50:  56nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506616(CHEMBL4443664)
Affinity DataEC50:  158nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506615(CHEMBL4452474)
Affinity DataEC50:  100nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50065915(CHEMBL3401461)
Affinity DataEC50:  126nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506618(CHEMBL4587388)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506619(CHEMBL4456708)
Affinity DataEC50:  96nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50506611(CHEMBL4464331)
Affinity DataEC50:  501nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50064645(CHEMBL3403768)
Affinity DataEC50:  195nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50554976(CHEMBL4759345)
Affinity DataEC50:  380nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50554977(CHEMBL4764409)
Affinity DataEC50:  282nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50554978(CHEMBL4789594)
Affinity DataEC50:  295nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50554979(CHEMBL4757666)
Affinity DataEC50:  251nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50064644(CHEMBL3403767)
Affinity DataEC50:  174nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50554980(CHEMBL4741911)
Affinity DataEC50:  257nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50554981(CHEMBL4776381)
Affinity DataEC50:  380nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50554982(CHEMBL4763920)
Affinity DataEC50:  234nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50554983(CHEMBL4749174)
Affinity DataEC50:  562nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50554984(CHEMBL4752713)
Affinity DataEC50:  631nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50554985(CHEMBL4782249)
Affinity DataEC50:  4.68E+3nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50554986(CHEMBL4787574)
Affinity DataEC50:  5.89E+3nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50554987(CHEMBL4754796)
Affinity DataEC50: <1.00E+4nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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