Affinity DataKi: 219nMAssay Description:Displacement of [3H]RTI-33 from GPR88 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 224nMAssay Description:Displacement of [3H]RTI-33 from GPR88 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 277nMAssay Description:Displacement of [3H]RTI-33 from GPR88 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 487nMAssay Description:Displacement of [3H]RTI-33 from GPR88 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 612nMAssay Description:Displacement of [3H]RTI-33 from GPR88 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 750nMAssay Description:Displacement of [3H]-Paroxetine from recombinant human full length SERT after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.29E+3nMAssay Description:Binding affinity to human full length KOR after 60 mins by radioligand-based scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of human SERT expressed in HEK293 cells assessed as reduction in SERT-mediated substrate uptake after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 63nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
TargetProbable G-protein coupled receptor 88(Mus musculus)
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataEC50: 1.14E+3nMAssay Description:Agonist activity at GPR88 in wild type mouse striatal membranes assessed as increase in [35S]-GTPgammaS binding after 1 hr by liquid scintillation co...More data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 501nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 398nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 316nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
TargetProbable G-protein coupled receptor 88(Mus musculus)
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataEC50: 535nMAssay Description:Agonist activity at GPR88 in wild type mouse striatal membranes assessed as increase in [35S]-GTPgammaS binding after 1 hr by liquid scintillation co...More data for this Ligand-Target Pair
Affinity DataEC50: 316nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 158nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 501nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 63nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 501nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+3nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 398nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 56nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 158nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+3nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 96nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 501nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in PPLS-HA-GPR88 CHO cells assessed as effect on forskolin-induced cAMP accumulation after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 195nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 380nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 282nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 295nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 251nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 174nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 257nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 380nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 234nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 562nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 631nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.68E+3nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.89E+3nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+4nMAssay Description:Agonist activity at GPR88 (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by TR-FRET assayMore data for this Ligand-Target Pair