TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Binding affinity to Plasmodium falciparum TrxR in presence of thioredoxinMore data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Binding affinity to Plasmodium falciparum TrxR in presence of NADPHMore data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataKi: 650nMAssay Description:Binding affinity to Plasmodium falciparum TrxR in presence of thioredoxinMore data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Binding affinity to Plasmodium falciparum TrxR in presence of NADPHMore data for this Ligand-Target Pair
Affinity DataKi: 3.60E+3nMAssay Description:Inhibitory concentration against Plasmodium falciparum glutathione reductaseMore data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:Inhibitory concentration against human glutathione reductaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.21E+4nMAssay Description:Inhibitory concentration against human glutathione reductase (In presence of glutathione disulfide)More data for this Ligand-Target Pair
Affinity DataKi: 1.61E+4nMAssay Description:Inhibitory concentration against human glutathione reductase (In presence of NADPH)More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory concentration against human glutathione reductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Inhibitory concentration against human glutathione reductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Concentration required for inhibition of Trypanothione reductase (TcTR) from Trypanosoma cruzi in the presence of 50 uM TS2 as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione disulfide reductase, assay in presence of 57 microM T(S)2.More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:In vitro inhibition of Plasmodium falciparum Glutathione ReductaseMore data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of Plasmodium falciparum TrxRMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Concentration required for inhibition of Trypanothione reductase (TcTR) from Trypanosoma cruzi in the presence of 50 uM TS2 as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 550nMAssay Description:Inhibition of trypanothione reductase from T. cruzi, in the presence 57 microM of trypanothione T(SH)2More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Concentration required for inhibition of Trypanothione reductase (TcTR) from Trypanosoma cruzi in the presence of 50 uM TS2 as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 750nMAssay Description:In vitro inhibition of human Glutathione ReductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione disulfide reductase, assay in presence of 57 microM T(S)2.More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibition of human Glutathione ReductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Concentration required for inhibition of Trypanothione reductase (TcTR) from Trypanosoma cruzi in the presence of 50 uM TS2 as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione disulfide reductase, assay in presence of 57 microM T(S)2.More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:In vitro inhibition of Plasmodium falciparum Glutathione ReductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione disulfide reductase, assay in presence of 57 microM T(S)2.More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione disulfide reductase, assay in presence of 57 microM T(S)2.More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione disulfide reductase, assay in presence of 57 microM T(S)2.More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione disulfide reductase, assay in presence of 57 microM T(S)2.More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione disulfide reductase, assay in presence of 57 microM T(S)2.More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of trypanothione reductase from T. cruzi, in the presence 57 microM of trypanothione T(SH)2More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione disulfide reductase, assay in presence of 57 microM T(S)2.More data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Plasmodium falciparum TrxRMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione disulfide reductase, assay in presence of 57 microM T(S)2.More data for this Ligand-Target Pair
TargetThioredoxin reductase 1, cytoplasmic/2, mitochondrial/3(Homo sapiens (Human))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human TrxRMore data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Plasmodium falciparum TrxRMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione disulfide reductase, assay in presence of 57 microM T(S)2.More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi trypanothione reductase after 5 mins preincubation with NADPH in presence of 100 uM TS2 substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione disulfide reductase, assay in presence of 57 microM T(S)2.More data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione disulfide reductase, assay in presence of 57 microM T(S)2.More data for this Ligand-Target Pair