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Found 97 with Last Name = 'deshmukh' and Initial = 'gd'
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM84796(PF-00215924)
Affinity DataIC50:  1.80nMpH: 7.5 T: 2°CAssay Description:Inhibition of active p38a MAP kinase by inhibitors was determinedusing a p38a cascade activity assay. A 30-lL reaction mixture wasprepared containing...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323438(4-(3-(3-tert-butyl-5-(3-naphthalen-1-ylureido)-1H-...)
Affinity DataIC50:  5nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM84788((9a) BIRB796)
Affinity DataIC50:  6nMpH: 7.5 T: 2°CAssay Description:Binding of inhibitors to unactivated p38a that leads to decreasedphosphorylation of p38alpha by MKK6 was determined by measuringthe activated p38alph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323438(4-(3-(3-tert-butyl-5-(3-naphthalen-1-ylureido)-1H-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323416(2-acetamido-N-(3-(3-tert-butyl-5-(3-phenylureido)-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM84786((10a) BIRB796)
Affinity DataIC50:  7nMpH: 7.5 T: 2°CAssay Description:Binding of inhibitors to unactivated p38a that leads to decreasedphosphorylation of p38alpha by MKK6 was determined by measuringthe activated p38alph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM84782((5a) BIRB796)
Affinity DataIC50:  8nMpH: 7.5 T: 2°CAssay Description:Binding of inhibitors to unactivated p38a that leads to decreasedphosphorylation of p38alpha by MKK6 was determined by measuringthe activated p38alph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM84791((11a) BIRB796)
Affinity DataIC50:  11nMpH: 7.5 T: 2°CAssay Description:Binding of inhibitors to unactivated p38a that leads to decreasedphosphorylation of p38alpha by MKK6 was determined by measuringthe activated p38alph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM84785((7a) BIRB796)
Affinity DataIC50:  11nMpH: 7.5 T: 2°CAssay Description:Binding of inhibitors to unactivated p38a that leads to decreasedphosphorylation of p38alpha by MKK6 was determined by measuringthe activated p38alph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM84784((6a) BIRB796 | (8a) BIRB796)
Affinity DataIC50:  11nMpH: 7.5 T: 2°CAssay Description:Binding of inhibitors to unactivated p38a that leads to decreasedphosphorylation of p38alpha by MKK6 was determined by measuringthe activated p38alph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323437((1R)-6-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyra...)
Affinity DataIC50:  14nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323427(CHEMBL1209482 | N-(3-(3-tert-butyl-5-(3-phenylurei...)
Affinity DataIC50:  16nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323420(CHEMBL1209343 | N-(2-(3-(3-tert-butyl-5-(3-phenylu...)
Affinity DataIC50:  18nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM84789((9b) BIRB796)
Affinity DataIC50:  22nMpH: 7.5 T: 2°CAssay Description:Binding of inhibitors to unactivated p38a that leads to decreasedphosphorylation of p38alpha by MKK6 was determined by measuringthe activated p38alph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM84784((6a) BIRB796 | (8a) BIRB796)
Affinity DataIC50:  25nMpH: 7.5 T: 2°CAssay Description:Binding of inhibitors to unactivated p38a that leads to decreasedphosphorylation of p38alpha by MKK6 was determined by measuringthe activated p38alph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM84783((5b) BIRB796)
Affinity DataIC50:  26nMpH: 7.5 T: 2°CAssay Description:Binding of inhibitors to unactivated p38a that leads to decreasedphosphorylation of p38alpha by MKK6 was determined by measuringthe activated p38alph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323431(CHEMBL1209564 | N-(3-(3-tert-butyl-5-(3-phenylurei...)
Affinity DataIC50:  27.9nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323435((1R)-2-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyra...)
Affinity DataIC50:  30nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323416(2-acetamido-N-(3-(3-tert-butyl-5-(3-phenylureido)-...)
Affinity DataIC50:  34nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM84792((11b) BIRB796)
Affinity DataIC50:  35nMpH: 7.5 T: 2°CAssay Description:Binding of inhibitors to unactivated p38a that leads to decreasedphosphorylation of p38alpha by MKK6 was determined by measuringthe activated p38alph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM84790((7b) BIRB796)
Affinity DataIC50:  36nMpH: 7.5 T: 2°CAssay Description:Binding of inhibitors to unactivated p38a that leads to decreasedphosphorylation of p38alpha by MKK6 was determined by measuringthe activated p38alph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323433(4-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50:  37nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323419(CHEMBL1209342 | N-(2-(3-(3-tert-butyl-5-(3-phenylu...)
Affinity DataIC50:  38nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323434(4-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50:  39nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323430(CHEMBL1209563 | N-(3-(3-tert-butyl-5-(3-phenylurei...)
Affinity DataIC50:  48.8nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323418(CHEMBL1209276 | N-(2-(3-(3-tert-butyl-5-(3-phenylu...)
Affinity DataIC50:  51nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM84794((12a) BIRB796)
Affinity DataIC50:  53nMpH: 7.5 T: 2°CAssay Description:Binding of inhibitors to unactivated p38a that leads to decreasedphosphorylation of p38alpha by MKK6 was determined by measuringthe activated p38alph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323436((1R)-2-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyra...)
Affinity DataIC50:  57nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM84793((12b) BIRB796)
Affinity DataIC50:  62nMpH: 7.5 T: 2°CAssay Description:Binding of inhibitors to unactivated p38a that leads to decreasedphosphorylation of p38alpha by MKK6 was determined by measuringthe activated p38alph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323427(CHEMBL1209482 | N-(3-(3-tert-butyl-5-(3-phenylurei...)
Affinity DataIC50:  63nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323425(CHEMBL1209407 | N-(3-(3-tert-butyl-5-(3-phenylurei...)
Affinity DataIC50:  68nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323415(CHEMBL1209273 | N-(3-(3-tert-butyl-5-(3-phenylurei...)
Affinity DataIC50:  68nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323432(CHEMBL1209565 | N-(3-(3-tert-butyl-5-(3-phenylurei...)
Affinity DataIC50:  78.2nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323420(CHEMBL1209343 | N-(2-(3-(3-tert-butyl-5-(3-phenylu...)
Affinity DataIC50:  88nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323423(CHEMBL1209405 | N-(3-(3-tert-butyl-5-(3-phenylurei...)
Affinity DataIC50:  108nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM84796(PF-00215924)
Affinity DataIC50:  110nMpH: 7.5 T: 2°CAssay Description:Binding of inhibitors to unactivated p38a that leads to decreasedphosphorylation of p38alpha by MKK6 was determined by measuringthe activated p38alph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323429(CHEMBL1209484 | N-(3-(3-tert-butyl-5-(3-phenylurei...)
Affinity DataIC50:  132nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323430(CHEMBL1209563 | N-(3-(3-tert-butyl-5-(3-phenylurei...)
Affinity DataIC50:  135nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323421(2-acetamido-N-(3-(3-tert-butyl-5-(3-phenylureido)-...)
Affinity DataIC50:  168nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323417(CHEMBL1209275 | N-(2-(3-(3-tert-butyl-5-(3-phenylu...)
Affinity DataIC50:  169nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323413(2-amino-N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-p...)
Affinity DataIC50:  176nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323414(CHEMBL1209214 | methyl 2-(3-(3-tert-butyl-5-(3-phe...)
Affinity DataIC50:  176nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323426(CHEMBL1209481 | N-(3-(3-tert-butyl-5-(3-phenylurei...)
Affinity DataIC50:  185nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323431(CHEMBL1209564 | N-(3-(3-tert-butyl-5-(3-phenylurei...)
Affinity DataIC50:  201nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323418(CHEMBL1209276 | N-(2-(3-(3-tert-butyl-5-(3-phenylu...)
Affinity DataIC50:  205nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323424(2-acetamido-N-(3-(3-tert-butyl-5-(3-phenylureido)-...)
Affinity DataIC50:  211nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM84797(PF-00215937 | PF-00215955)
Affinity DataIC50:  220nMpH: 7.5 T: 2°CAssay Description:Binding of inhibitors to unactivated p38a that leads to decreasedphosphorylation of p38alpha by MKK6 was determined by measuringthe activated p38alph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323428(CHEMBL1209483 | N-(3-(3-tert-butyl-5-(3-phenylurei...)
Affinity DataIC50:  231nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM50323419(CHEMBL1209342 | N-(2-(3-(3-tert-butyl-5-(3-phenylu...)
Affinity DataIC50:  243nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pfizer

LigandPNGBDBM84786((10a) BIRB796)
Affinity DataIC50:  261nMpH: 7.5 T: 2°CAssay Description:Inhibition of active p38a MAP kinase by inhibitors was determinedusing a p38a cascade activity assay. A 30-lL reaction mixture wasprepared containing...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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