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Found 167 with Last Name = 'diamantidis' and Initial = 'g'
LigandPNGBDBM94503(2-hydroxypropane-1,2,3-tricarboxylic acid;N-[4-(me...)
Affinity DataKi:  0.0200nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50008984(4-(4-Chloro-benzyl)-2-(1-methyl-azepan-4-yl)-2H-ph...)
Affinity DataKi:  2.20nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
LigandPNGBDBM50228269(CHEMBL178035)
Affinity DataKi:  3.5nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has Muscarinic acetylcholine receptor M2 sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228255(CHEMBL362439)
Affinity DataKi:  7.70nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM83450(ALFENTANIL | Alfentanil hydrochloride | MLS0023206...)
Affinity DataKi:  8.20nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has Muscarinic acetylcholine receptor M2 sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228260(CHEMBL367286)
Affinity DataKi:  8.20nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228221(CHEMBL366899)
Affinity DataKi:  9.10nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228224(CHEMBL367667)
Affinity DataKi:  10nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228217(CHEMBL174694)
Affinity DataKi:  10nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228259(CHEMBL426034)
Affinity DataKi:  12nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228219(CHEMBL178847)
Affinity DataKi:  14nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228251(CHEMBL176438)
Affinity DataKi:  14nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228218(CHEMBL368487)
Affinity DataKi:  24nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has M2 muscarinic receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228231(CHEMBL174828)
Affinity DataKi:  26nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228225(CHEMBL174758)
Affinity DataKi:  27nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228230(CHEMBL174947)
Affinity DataKi:  30nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228264(CHEMBL367661)
Affinity DataKi:  30nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has M2 muscarinic receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228253(CHEMBL367968)
Affinity DataKi:  41nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228256(CHEMBL369412)
Affinity DataKi:  49nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228226(CHEMBL172032)
Affinity DataKi:  56nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228263(CHEMBL175126)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228257(CHEMBL172703)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228258(CHEMBL172717)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228223(CHEMBL369448)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228222(CHEMBL175148)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228250(CHEMBL369455)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228254(CHEMBL172910)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228262(CHEMBL172531)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228252(CHEMBL435340)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228268(CHEMBL173971)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228228(CHEMBL366436)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228270(CHEMBL178434)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228227(CHEMBL174962)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228265(CHEMBL263783)
Affinity DataKi: >100nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228267(CHEMBL177046)
Affinity DataKi: >100nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has M2 muscarinic receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228229(CHEMBL174834)
Affinity DataKi: >100nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has M2 muscarinic receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228266(CHEMBL369871)
Affinity DataKi: >100nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has M2 muscarinic receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228220(CHEMBL174926)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228261(CHEMBL176618)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50303103(1-(3-(3-(4-chloro-3-hydroxyphenyl)-2-(pyridin-4-yl...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of B-RafMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50303123(CHEMBL570681 | ethyl 3-(3-(7-fluoro-1H-indazol-4-y...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of B-RafMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50303098(5-(7-(8-azabicyclo[3.2.1]octan-3-yl)-2-(pyridin-4-...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of B-RafMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50303121(CHEMBL585144 | ethyl 3-(3-(7-chloro-1H-indazol-4-y...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of B-RafMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50303100(2-chloro-5-(7-(8-ethyl-8-azabicyclo[3.2.1]octan-3-...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of B-RafMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50303131(2-chloro-5-[13-(hydroxymethyl)-15-methyl-5-(pyridi...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of B-RafMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50303127(CHEMBL583133 | ethyl 3-(3-(7-methyl-1H-indazol-4-y...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of B-RafMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50303132(2-chloro-5-[13-(hydroxymethyl)-15-methyl-5-(pyridi...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of B-RafMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50303094(CHEMBL571129 | ethyl 3-(3-(3-hydroxyphenyl)-2-(pyr...)
Affinity DataIC50:  1nMAssay Description:Inhibition of B-RafMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50303130(CHEMBL585148 | Methyl 6-(4-chloro-3-hydroxyphenyl)...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of B-RafMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50303110(CHEMBL585334 | ethyl 3-(3-(1H-indazol-4-yl)-2-(pyr...)
Affinity DataIC50:  2nMAssay Description:Inhibition of B-RafMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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