Compile Data Set for Download or QSAR
maximum 50k data
Found 28 with Last Name = 'doukas' and Initial = 'p'
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [3H]QNB (quinuclidinyl benzylate) from muscarinic M2 receptor of rat heart homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]pirenzepine from muscarinic M1 receptor of rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]pirenzepine from muscarinic M1 receptor of rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291598(2-(4-Diethylamino-but-2-ynyl)-isoindole-1,3-dione ...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]pirenzepine from muscarinic M1 receptor of rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291598(2-(4-Diethylamino-but-2-ynyl)-isoindole-1,3-dione ...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]QNB (quinuclidinyl benzylate) from muscarinic M2 receptor of rat heart homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291596(1-(4-Diethylamino-but-2-ynyl)-3,3-diphenyl-pyrroli...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]pirenzepine from muscarinic M1 receptor of rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  267nMAssay Description:Displacement of [3H]QNB (quinuclidinyl benzylate) from muscarinic M2 receptor of rat heart homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291592(3-(4-Diethylamino-but-2-ynyl)-5,5-diphenyl-imidazo...)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]pirenzepine from muscarinic M1 receptor of rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291596(1-(4-Diethylamino-but-2-ynyl)-3,3-diphenyl-pyrroli...)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]QNB (quinuclidinyl benzylate) from muscarinic M2 receptor of rat heart homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291601(1-(4-Diisopropylamino-but-2-ynyl)-3,3-diphenyl-pyr...)
Affinity DataKi:  440nMAssay Description:Displacement of [3H]QNB (quinuclidinyl benzylate) from muscarinic M2 receptor of rat heart homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291591(1'-(4-diethylamino-2-butynyl)spiro[10,11-dihydro-5...)
Affinity DataKi:  460nMAssay Description:Displacement of [3H]pirenzepine from muscarinic M1 receptor of rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291601(1-(4-Diisopropylamino-but-2-ynyl)-3,3-diphenyl-pyr...)
Affinity DataKi:  530nMAssay Description:Displacement of [3H]pirenzepine from muscarinic M1 receptor of rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291600(5,5-Diphenyl-3-(4-pyrrolidin-1-yl-but-2-ynyl)-imid...)
Affinity DataKi:  640nMAssay Description:Displacement of [3H]pirenzepine from muscarinic M1 receptor of rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291602(1'-(4-diethylamino-2-butynyl)spiro[2,3-dihydro-1H-...)
Affinity DataKi:  680nMAssay Description:Displacement of [3H]pirenzepine from muscarinic M1 receptor of rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291592(3-(4-Diethylamino-but-2-ynyl)-5,5-diphenyl-imidazo...)
Affinity DataKi:  950nMAssay Description:Displacement of [3H]QNB (quinuclidinyl benzylate) from muscarinic M2 receptor of rat heart homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291597(1-(4-diethylamino-2-butynyl)spiro[tetrahydro-1H-im...)
Affinity DataKi:  1.05E+3nMAssay Description:Displacement of [3H]pirenzepine from muscarinic M1 receptor of rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291593(1'-(4-tetrahydro-1H-1-pyrrolyl-2-butynyl)spiro[2,3...)
Affinity DataKi:  1.59E+3nMAssay Description:Displacement of [3H]pirenzepine from muscarinic M1 receptor of rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291595(1'-(4-diisopropylamino-2-butynyl)spiro[9H-fluorene...)
Affinity DataKi:  1.62E+3nMAssay Description:Displacement of [3H]pirenzepine from muscarinic M1 receptor of rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291599(1'-(4-diethylamino-2-butynyl)spiro[9H-fluorene-9,3...)
Affinity DataKi:  1.63E+3nMAssay Description:Displacement of [3H]pirenzepine from muscarinic M1 receptor of rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291591(1'-(4-diethylamino-2-butynyl)spiro[10,11-dihydro-5...)
Affinity DataKi:  2.09E+3nMAssay Description:Displacement of [3H]QNB (quinuclidinyl benzylate) from muscarinic M2 receptor of rat heart homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291594(1-(4-Diethylamino-but-2-ynyl)-3-phenyl-pyrrolidine...)
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of [3H]pirenzepine from muscarinic M1 receptor of rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291602(1'-(4-diethylamino-2-butynyl)spiro[2,3-dihydro-1H-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]QNB (quinuclidinyl benzylate) from muscarinic M2 receptor of rat heart homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291600(5,5-Diphenyl-3-(4-pyrrolidin-1-yl-but-2-ynyl)-imid...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]QNB (quinuclidinyl benzylate) from muscarinic M2 receptor of rat heart homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291599(1'-(4-diethylamino-2-butynyl)spiro[9H-fluorene-9,3...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]QNB (quinuclidinyl benzylate) from muscarinic M2 receptor of rat heart homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291595(1'-(4-diisopropylamino-2-butynyl)spiro[9H-fluorene...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]QNB (quinuclidinyl benzylate) from muscarinic M2 receptor of rat heart homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291593(1'-(4-tetrahydro-1H-1-pyrrolyl-2-butynyl)spiro[2,3...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]QNB (quinuclidinyl benzylate) from muscarinic M2 receptor of rat heart homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291594(1-(4-Diethylamino-but-2-ynyl)-3-phenyl-pyrrolidine...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]QNB (quinuclidinyl benzylate) from muscarinic M2 receptor of rat heart homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291597(1-(4-diethylamino-2-butynyl)spiro[tetrahydro-1H-im...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]QNB (quinuclidinyl benzylate) from muscarinic M2 receptor of rat heart homogenates.More data for this Ligand-Target Pair
In DepthDetails Article