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Found 57 with Last Name = 'dubreuil' and Initial = 'p'
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50024328(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  90nMAssay Description:In vitro inhibitory activity for binding of [125I]-(Nle11)-HG-13 to gastrin receptor on isolated rabbit gastric mucosal cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataIC50:  100nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50341636((3Z)-N-(3-CHLOROPHENYL)-3-({3,5-DIMETHYL-4-[(4-MET...)
Affinity DataIC50:  152nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359981(CHEMBL1927770)
Affinity DataIC50:  171nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359982(CHEMBL1927771)
Affinity DataIC50:  206nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50341636((3Z)-N-(3-CHLOROPHENYL)-3-({3,5-DIMETHYL-4-[(4-MET...)
Affinity DataIC50:  228nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human GTL16 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50024330(3-(3-Benzyl-ureido)-3-{2-[2-tert-butoxycarbonylami...)
Affinity DataIC50:  300nMAssay Description:In vitro inhibitory activity for binding of [125I]-(Nle11)-HG-13 to gastrin receptor on isolated rabbit gastric mucosal cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174413(2-(2-Diethylamino-ethyl)-9-hydroxy-5,11-dimethyl-6...)
Affinity DataIC50:  300nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359981(CHEMBL1927770)
Affinity DataIC50:  321nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human HepG2 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004227(5,11-Dimethyl-6H-pyrido[4,3-b]carbazol-9-ol | 5,11...)
Affinity DataIC50:  400nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004227(5,11-Dimethyl-6H-pyrido[4,3-b]carbazol-9-ol | 5,11...)
Affinity DataIC50:  400nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004235((NMHE)9-Hydroxy-2,5,11-trimethyl-6H-pyrido[4,3-b]c...)
Affinity DataIC50:  400nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004227(5,11-Dimethyl-6H-pyrido[4,3-b]carbazol-9-ol | 5,11...)
Affinity DataIC50:  400nMAssay Description:Inhibitory activity against Fibroblast growth factor receptor 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004235((NMHE)9-Hydroxy-2,5,11-trimethyl-6H-pyrido[4,3-b]c...)
Affinity DataIC50:  400nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174413(2-(2-Diethylamino-ethyl)-9-hydroxy-5,11-dimethyl-6...)
Affinity DataIC50:  450nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004235((NMHE)9-Hydroxy-2,5,11-trimethyl-6H-pyrido[4,3-b]c...)
Affinity DataIC50:  500nMAssay Description:Inhibitory activity against Fibroblast growth factor receptor 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359983(CHEMBL1927769)
Affinity DataIC50:  559nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004227(5,11-Dimethyl-6H-pyrido[4,3-b]carbazol-9-ol | 5,11...)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity against Platelet-derived growth factor receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174412(9-Methoxy-5,11-dimethyl-6H-pyrido[4,3-b]carbazole ...)
Affinity DataIC50:  600nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359984(CHEMBL1927768)
Affinity DataIC50:  607nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359982(CHEMBL1927771)
Affinity DataIC50:  620nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human HepG2 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004235((NMHE)9-Hydroxy-2,5,11-trimethyl-6H-pyrido[4,3-b]c...)
Affinity DataIC50:  700nMAssay Description:Inhibitory activity against Platelet-derived growth factor receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359985(CHEMBL1927772)
Affinity DataIC50:  760nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359986(CHEMBL1927625)
Affinity DataIC50:  793nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174412(9-Methoxy-5,11-dimethyl-6H-pyrido[4,3-b]carbazole ...)
Affinity DataIC50:  800nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359981(CHEMBL1927770)
Affinity DataIC50:  811nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human GTL16 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359982(CHEMBL1927771)
Affinity DataIC50:  1.19E+3nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human GTL16 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174410(1-(3-Diethylamino-propylamino)-5,11-dimethyl-6H-py...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50024327(CHEMBL349888 | N-{1-[2-tert-Butoxycarbonylamino-3-...)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro inhibitory activity for binding of [125I]-(Nle11)-HG-13 to gastrin receptor on isolated rabbit gastric mucosal cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174410(1-(3-Diethylamino-propylamino)-5,11-dimethyl-6H-py...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174408(1-(3-Diethylamino-propylamino)-5,6,11-trimethyl-6H...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity against Fibroblast growth factor receptor 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50341636((3Z)-N-(3-CHLOROPHENYL)-3-({3,5-DIMETHYL-4-[(4-MET...)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human HepG2 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359984(CHEMBL1927768)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human HepG2 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174411(CHEMBL197610 | N,N-Diethyl-N'-(10-methyl-11H-pyrid...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174408(1-(3-Diethylamino-propylamino)-5,6,11-trimethyl-6H...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity against Platelet-derived growth factor receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174407(CHEMBL279472 | N,N-Diethyl-N'-(9-methoxy-5-methyl-...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174411(CHEMBL197610 | N,N-Diethyl-N'-(10-methyl-11H-pyrid...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174408(1-(3-Diethylamino-propylamino)-5,6,11-trimethyl-6H...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174407(CHEMBL279472 | N,N-Diethyl-N'-(9-methoxy-5-methyl-...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174408(1-(3-Diethylamino-propylamino)-5,6,11-trimethyl-6H...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359981(CHEMBL1927770)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of TPR-fused MET-mediated mouse BA/F3 cell proliferation after 48 hrs by cell titre blue based spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359985(CHEMBL1927772)
Affinity DataIC50:  5.65E+3nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human GTL16 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50024332(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  6.00E+3nMAssay Description:In vitro inhibitory activity for binding of [125I]-(Nle11)-HG-13 to gastrin receptor on isolated rabbit gastric mucosal cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359987(CHEMBL1927778)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359984(CHEMBL1927768)
Affinity DataIC50:  7.73E+3nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human GTL16 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174409(9-Bromo-5,11-dimethyl-6H-pyrido[4,3-b]carbazole | ...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174409(9-Bromo-5,11-dimethyl-6H-pyrido[4,3-b]carbazole | ...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004233(5,11-dimethyl-2H-pyrido[4,3-b]carbazole | CHEMBL12...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004233(5,11-dimethyl-2H-pyrido[4,3-b]carbazole | CHEMBL12...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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