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Found 176 with Last Name = 'dwivedi' and Initial = 'a'
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524365(CHEMBL4579211)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant human H3 receptor expressed in HEK293T cells measured after 90 mins by liquid scintillat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524374(CHEMBL4453810)
Affinity DataKi:  6.10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant human H3 receptor expressed in HEK293T cells measured after 90 mins by liquid scintillat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50035670(CHEMBL3338456)
Affinity DataKi:  3.53E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50035656(CHEMBL1986389)
Affinity DataKi:  3.86E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50035662(CHEMBL3338464)
Affinity DataKi:  5.25E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50035666(CHEMBL3338460)
Affinity DataKi:  6.38E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50035663(CHEMBL3338463)
Affinity DataKi:  7.01E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50035657(CHEMBL3338469)
Affinity DataKi:  7.32E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50035658(CHEMBL3338468)
Affinity DataKi:  7.59E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50035665(CHEMBL3338461)
Affinity DataKi:  7.68E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50035659(CHEMBL3338467)
Affinity DataKi:  9.04E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50035664(CHEMBL3338462)
Affinity DataKi:  9.21E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50035667(CHEMBL3338459)
Affinity DataKi:  1.08E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50035668(CHEMBL3338458)
Affinity DataKi:  1.25E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50035661(CHEMBL3338465)
Affinity DataKi:  1.31E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50035655(CHEMBL3338470)
Affinity DataKi:  1.85E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50035669(CHEMBL3338457)
Affinity DataKi:  2.29E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50035660(CHEMBL3338466)
Affinity DataKi:  2.65E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PknBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50595061(CHEMBL5209357)
Affinity DataIC50:  0.25nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as substrate preincubated for 20 mins followed by substrate addition by DTNB reagent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of human recombinant microsomal MAO-A expressed in baculovirus infected BTI-TN-5B1-4 cells assessed as reduction in production of H202 usi...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50595058(CHEMBL5199704)
Affinity DataIC50:  9.5nMAssay Description:Inhibition of recombinant human AChE using Amplex red, acetylthiocholine as substrate preincubated for 15 mins followed by substrate addition and mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50595064(CHEMBL582490 | GNF-Pf-3382)
Affinity DataIC50:  14nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50150726(3-(4-Methanesulfonyl-phenyl)-6-(4-methoxy-phenyl)-...)
Affinity DataIC50:  20nMAssay Description:Inhibition of COX2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50553263(CHEMBL4790416)
Affinity DataIC50:  30nMAssay Description:Inhibition of recombinant human AChE using Amplex red, acetylthiocholine as substrate preincubated for 15 mins followed by substrate addition and mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  30nMAssay Description:Inhibition of electric eel AChE assessed as reduction in production of H202 using acetylcholine as substrate incubated for 15 mins followed by substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50595063(DIHYDROACTINIDIOLIDE)
Affinity DataIC50:  30nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 45 mins followed by substrate addition by DTNB reage...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50595055(CHEMBL5200462)
Affinity DataIC50:  35nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524380(CHEMBL4451233)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524380(CHEMBL4451233)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524379(CHEMBL4540275)
Affinity DataIC50: <50nMAssay Description:Displacement of [I125]bolton hunter-CCK-8S from recombinant human CCK1 receptor expressed in stable CHO cells measured after 1 to 2 hrs by microscint...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524368(CHEMBL4452406)
Affinity DataIC50:  66nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524368(CHEMBL4452406)
Affinity DataIC50:  70nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524367(CHEMBL4580450)
Affinity DataIC50:  85nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524367(CHEMBL4580450)
Affinity DataIC50:  90nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50539579(CHEMBL4644113)
Affinity DataIC50:  120nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50595062(CHEMBL5196827)
Affinity DataIC50:  129nMAssay Description:Inhibition of human BACE-1 using Rh-EVNLDAEFK-quencher as peptide substrate incubated for 1 hr in dark by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50595052(CHEMBL5177450)
Affinity DataIC50:  150nMAssay Description:Inhibition of Electrophorus electricus AchE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition by El...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50172756(Benzyl-methyl-prop-2-ynyl-amine | CHEMBL673 | Euto...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human recombinant microsomal MAO-B expressed in baculovirus infected BTI-TN-5B1-4 cells assessed as reduction in production of H202 usi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50595064(CHEMBL582490 | GNF-Pf-3382)
Affinity DataIC50:  182nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlutamate receptor ionotropic, NMDA 2A(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50595057(CHEMBL5202551)
Affinity DataIC50:  240nMAssay Description:Inhibition of NMDA receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524363(CHEMBL4585616)
Affinity DataIC50:  240nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524363(CHEMBL4585616)
Affinity DataIC50:  245nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50117930((4-{1-[2-(6-Methyl-pyridin-2-yl)-ethyl]-piperidine...)
Affinity DataIC50: <300nMAssay Description:Inhibition of tracer Red binding to human ERG expressed in membranes after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50595067(CHEMBL5208806)
Affinity DataIC50:  390nMAssay Description:Inhibition of Electrophorus electricus AchE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50504429(CHEMBL4455506)
Affinity DataIC50:  440nMAssay Description:Inhibition of Electrophorus electricus AchE using acetylthiocholine iodide as substrate incubated for 15 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM24724((adamantan-1-ylmethyl)({3-[(7-chloroquinolin-4-yl)...)
Affinity DataIC50:  500nMAssay Description:Inhibition of recombinant human AChE using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524371(CHEMBL4456972)
Affinity DataIC50:  550nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524371(CHEMBL4456972)
Affinity DataIC50:  560nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50595056(CHEMBL5197661)
Affinity DataIC50:  615nMAssay Description:Inhibition of horse serum BuChE using butyrylthiocholine chloride as substrate by spectrophotometric based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50553263(CHEMBL4790416)
Affinity DataIC50:  660nMAssay Description:Inhibition of human BuChE using butyrylthiocholine iodide as substrate preincubated for 30 mins followed by substrate addition and measured after 20 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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