Affinity DataKi: 111nMAssay Description:Invitro inhibition was measured against Human Thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 145nMAssay Description:Invitro inhibition was measured against Human Thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 751nMAssay Description:Invitro inhibition was measured against Human Thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 1.45E+3nMAssay Description:Invitro inhibition was measured against Human Thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 3.40E+3nMAssay Description:Invitro inhibition was measured against Human bovine pancreatic trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 3.58E+3nMAssay Description:Invitro inhibition was measured against Human bovine pancreatic trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 5.10E+3nMAssay Description:Invitro inhibition was measured against Human bovine pancreatic trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 5.10E+3nMAssay Description:Invitro inhibition was measured against Human Thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 5.30E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 5.36E+3nMAssay Description:Invitro inhibition was measured against Human bovine pancreatic trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 5.80E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 6.78E+3nMAssay Description:Invitro inhibition was measured against Human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 6.80E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 7.50E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 7.90E+3nMAssay Description:Invitro inhibition was measured against Human bovine pancreatic trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 9.40E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Westf£Lischen Wilhelms-Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Westf£Lischen Wilhelms-Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Displacement of [3H]-(+)-MK-801 from phencyclidine binding site of NMDA receptor in human frontal cortex after 22 hrs by scintillation counting analy...More data for this Ligand-Target Pair
Affinity DataKi: 1.03E+4nMAssay Description:Invitro inhibition was measured against Human Thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 1.16E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.33E+4nMAssay Description:Invitro inhibition was measured against Human bovine pancreatic trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 1.58E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.59E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.78E+4nMAssay Description:Invitro inhibition was measured against Human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.86E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.95E+4nMAssay Description:Invitro inhibition was measured against Human Thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 1.96E+4nMAssay Description:Invitro inhibition was measured against Bovine pancreatic trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 2.05E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 2.21E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 2.51E+4nMAssay Description:Invitro inhibition was measured against Human bovine pancreatic trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 2.60E+4nMAssay Description:Invitro inhibition was measured against Human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 2.86E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 3.30E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: >3.37E+4nMAssay Description:Invitro inhibition was measured against Human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: >3.37E+4nMAssay Description:Invitro inhibition was measured against Human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 4.07E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 4.13E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 4.37E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 4.74E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 5.10E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 6.14E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 6.24E+4nMAssay Description:Invitro inhibition was measured against Human Thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 1.09E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.13E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.15E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.38E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.93E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair