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Found 67 with Last Name = 'emonds-alt' and Initial = 'x'
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  0.00430nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  0.00610nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.0420nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.0440nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(mouse)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM85083(NKB [MePhe7])
Affinity DataKi:  0.0530nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.0540nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.0590nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051290(CHEMBL299377 | N-(1-{3-[1-Benzoyl-3-(3,4-dichloro-...)
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Gerbil)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM85083(NKB [MePhe7])
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051290(CHEMBL299377 | N-(1-{3-[1-Benzoyl-3-(3,4-dichloro-...)
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051290(CHEMBL299377 | N-(1-{3-[1-Benzoyl-3-(3,4-dichloro-...)
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281769(Acetic acid 1-[4-(benzoyl-methyl-amino)-3-(3,4-dic...)
Affinity DataKi:  0.300nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281767(Acetic acid 1-{3-(3,4-dichloro-phenyl)-4-[ethyl-(t...)
Affinity DataKi:  0.300nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.330nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM85083(NKB [MePhe7])
Affinity DataKi:  0.340nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Gerbil)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051290(CHEMBL299377 | N-(1-{3-[1-Benzoyl-3-(3,4-dichloro-...)
Affinity DataKi:  0.420nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM85083(NKB [MePhe7])
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81942(CAS_55582 | NKA | NSC_55582 | Neurokinin alpha | S...)
Affinity DataKi:  0.480nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50071484(CHEMBL308148 | N-[(R)-4-(4-Acetylamino-4-phenyl-pi...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50335566(CHEMBL1651026 | Substance P [Sar9,Met(O2)11])
Affinity DataKi:  0.650nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM81942(CAS_55582 | NKA | NSC_55582 | Neurokinin alpha | S...)
Affinity DataKi:  0.760nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281771(CHEMBL173841 | N-[2-(3,4-Dichloro-phenyl)-4-(4-eth...)
Affinity DataKi:  0.900nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281768(CHEMBL176588 | Thiophene-3-carboxylic acid [2-(3,4...)
Affinity DataKi:  1nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50129513(CHEMBL71397 | N-[2-(3,4-Dichloro-phenyl)-4-(4-hydr...)
Affinity DataKi:  1nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Rattus norvegicus (rat))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  1.07nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  1.15nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(HAMSTER)
TBA

Curated by ChEMBL
LigandPNGBDBM50071484(CHEMBL308148 | N-[(R)-4-(4-Acetylamino-4-phenyl-pi...)
Affinity DataKi:  1.20nMAssay Description:The compound was evaluated for the inhibition of [125I]-NKA binding to neurokinin NK2 receptor from hamster urinary bladder membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281766(CHEMBL173008 | Thiophene-2-carboxylic acid [2-(3,4...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281773(CHEMBL176853 | Naphthalene-1-carboxylic acid [2-(3...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81942(CAS_55582 | NKA | NSC_55582 | Neurokinin alpha | S...)
Affinity DataKi:  2.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(mouse)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051290(CHEMBL299377 | N-(1-{3-[1-Benzoyl-3-(3,4-dichloro-...)
Affinity DataKi:  15nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50050650((S)-N-{(S)-1-[(S)-1-({[(S)-1-((S)-1-Carbamoyl-3-me...)
Affinity DataKi:  17.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281770(CHEMBL367542 | N-[4-[4-(Acetylamino-methyl)-4-phen...)
Affinity DataKi:  23nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  24nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051290(CHEMBL299377 | N-(1-{3-[1-Benzoyl-3-(3,4-dichloro-...)
Affinity DataKi:  26nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Gerbil)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051290(CHEMBL299377 | N-(1-{3-[1-Benzoyl-3-(3,4-dichloro-...)
Affinity DataKi:  30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051290(CHEMBL299377 | N-(1-{3-[1-Benzoyl-3-(3,4-dichloro-...)
Affinity DataKi:  32nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051290(CHEMBL299377 | N-(1-{3-[1-Benzoyl-3-(3,4-dichloro-...)
Affinity DataKi:  32nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  34nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281772(CHEMBL368372 | N-[2-(3,4-Dichloro-phenyl)-4-(4-hyd...)
Affinity DataKi:  50nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051290(CHEMBL299377 | N-(1-{3-[1-Benzoyl-3-(3,4-dichloro-...)
Affinity DataKi:  60nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  71nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051290(CHEMBL299377 | N-(1-{3-[1-Benzoyl-3-(3,4-dichloro-...)
Affinity DataKi:  73nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50129520(CHEMBL69335 | N-[2-(3,4-Dichloro-phenyl)-4-(4-phen...)
Affinity DataKi: >100nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281774(CHEMBL366382 | N-[4-(4-Acetylamino-4-phenyl-piperi...)
Affinity DataKi: >100nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50051290(CHEMBL299377 | N-(1-{3-[1-Benzoyl-3-(3,4-dichloro-...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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