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Found 260 with Last Name = 'endo' and Initial = 'y'
TargetEstrogen receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50076331(1-(hydroxymethyl)-12-(4-hydroxyphenyl)-1,12-dicarb...)
Affinity DataKi:  0.100nMAssay Description:In vitro inhibition of [6,7-3H]-17beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064089(4-hydroxymethyl-7,10-diisopropyl-8,10,13-trimethyl...)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50076330(1-(4-hydroxyphenyl)-1,12-dicarba-closo-dodecaboran...)
Affinity DataKi:  0.400nMAssay Description:In vitro inhibition of [6,7-3H]-17beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50076332(1-amino-12-(4-hydroxyphenyl)-1,12-dicarba-closo-do...)
Affinity DataKi:  0.650nMAssay Description:In vitro inhibition of [6,7-3H]-17beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
Ligand InfoCHEMBLPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50084059((2S,5S)-2-Dodecyl-5-hydroxymethyl-1-methyl-1,4,5,6...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity for human recombinant protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50084058((2S,5S)-2-Decyl-5-hydroxymethyl-1-methyl-1,4,5,6-t...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity for human recombinant protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50084061((2S,5S)-5-Hydroxymethyl-1-methyl-2-tetradecyl-1,4,...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity for human recombinant protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50081077(CHEMBL216658 | Dicarba-Closo-Dodecaborane analogue)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50081078(CHEMBL374446 | Dicarba-Closo-Dodecaborane analogue)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064091((2S,5S)-9-Decyl-5-hydroxymethyl-2-isopropyl-1-meth...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50081076(CHEMBL414278 | Dicarba-Closo-Dodecaborane analogue)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064090((S)-2-Decyl-5-hydroxymethyl-1-methyl-1,4,5,6-tetra...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064091((2S,5S)-9-Decyl-5-hydroxymethyl-2-isopropyl-1-meth...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073876((1S,4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-met...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064092(5'-hydroxymethyl-2'-isopropyl-1',4,4-trimethyl-(2'...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073875((1S,4S,5aS,9aS)-1,7,7-Tributyl-4-hydroxymethyl-5a-...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064094(5'-hydroxymethyl-2'-isopropyl-1'-methyl-(2'S,5'S)-...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073873((1S,4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-1,5a-d...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50057510((2S,5S)-8-Decyl-5-hydroxymethyl-2-isopropyl-1-meth...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073874((4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-methyl...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064093((7S,10S)-10-Hydroxymethyl-7-isopropyl-4,4,6-trimet...)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50290875((S)-13-Hydroxymethyl-10-((S)-isopropyl)-3,9,12-tri...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]-PDBu from Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073874((4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-methyl...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073878((4R,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-methyl...)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50290877((3S,6S)-6-Hydroxymethyl-3-isopropyl-4-tetradecyl-p...)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]-PDBu from Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073872((4S,5aS,5bS,7aS,10aS,10bS,12aS)-4-Hydroxymethyl-5a...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073870((4R,5aS,5bS,7aR,8R,10aS,10bR,12aS)-8-(1,5-Dimethyl...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073871((4R,5aS,5bS,7aS,10aS,10bS,12aS)-4-Hydroxymethyl-5a...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073877((4S,5aS,5bS,7aR,8R,10aS,10bR,12aS)-8-(1,5-Dimethyl...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50084060((2S,5S)-5-Hydroxymethyl-2-icosyl-1-methyl-1,4,5,6-...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for human recombinant protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064088((7S,10S)-10-Hydroxymethyl-7-isopropyl-1,1,6-trimet...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50057513((2S,5S)-5-Hydroxymethyl-2-isopropyl-1-methyl-1,4,5...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50290876((3S,6R)-6-Hydroxymethyl-3-isopropyl-4-tetradecyl-p...)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of [3H]-PDBu from Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064095((7S,10S)-10-Hydroxymethyl-7-isopropyl-1,1,4,4,6-pe...)
Affinity DataKi:  5.10E+3nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50290874((3R,6S)-6-Hydroxymethyl-3-isopropyl-4-tetradecyl-p...)
Affinity DataKi:  6.50E+3nMAssay Description:Displacement of [3H]-PDBu from Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50290873((3R,6R)-6-Hydroxymethyl-3-isopropyl-4-tetradecyl-p...)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [3H]-PDBu from Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetBDNF/NT-3 growth factors receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50512464(CHEMBL4555442)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of human GST-tagged TRKB (456 to 822) expressed in baculovirus expression system using TK-biotin peptide as substrate incubated for 45 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50512470(CHEMBL4462919)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of human GST-tagged TRKA (436 to 790) expressed in baculovirus expression system using TK-biotin peptide as substrate incubated for 45 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50512464(CHEMBL4555442)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of human GST-tagged TRKA (436 to 790) expressed in baculovirus expression system using TK-biotin peptide as substrate incubated for 45 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50512463(CHEMBL4528647)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of human GST-tagged TRKA (436 to 790) expressed in baculovirus expression system using TK-biotin peptide as substrate incubated for 45 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
Kyoto 607-8042

Curated by ChEMBL
LigandPNGBDBM50042053(CHEMBL3360172)
Affinity DataIC50:  0.320nMAssay Description:Inhibition of PDE7A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50135513(CHEMBL219004 | Carboron Cluster with phenol)
Affinity DataIC50:  0.590nMAssay Description:Binding affinity for estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
Kyoto 607-8042

Curated by ChEMBL
LigandPNGBDBM50042036(CHEMBL3360170)
Affinity DataIC50:  0.680nMAssay Description:Inhibition of PDE7A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50512462(CHEMBL4549659)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of human GST-tagged TRKA (436 to 790) expressed in baculovirus expression system using TK-biotin peptide as substrate incubated for 45 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
Kyoto 607-8042

Curated by ChEMBL
LigandPNGBDBM50032547(CHEMBL3354181)
Affinity DataIC50:  1nMAssay Description:Inhibition of human PDE7A1 expressed in insect cells assessed as inhibition of [3H]cAMP to [3H]AMP hydrolysis after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
Kyoto 607-8042

Curated by ChEMBL
LigandPNGBDBM50042037(CHEMBL3360169)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of PDE7A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
Kyoto 607-8042

Curated by ChEMBL
LigandPNGBDBM50042035(CHEMBL3360171)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of PDE7A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
Kyoto 607-8042

Curated by ChEMBL
LigandPNGBDBM50068286(CHEMBL3403373)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of human PDE7A expressed in insect cells assessed as inhibition of [3H]cAMP to [3H]AMP hydrolysis after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50512461(CHEMBL4457481)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of human GST-tagged TRKA (436 to 790) expressed in baculovirus expression system using TK-biotin peptide as substrate incubated for 45 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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