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Found 192 with Last Name = 'estrella' and Initial = 'm'
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087536(3-(3-Carbamimidoyl-phenyl)-isoxazole-4-carboxylic ...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087533(3-(3-Carbamimidoyl-phenyl)-isoxazole-4-carboxylic ...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Oryctolagus cuniculus)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087533(3-(3-Carbamimidoyl-phenyl)-isoxazole-4-carboxylic ...)
Affinity DataKi:  0.400nMAssay Description:Inhibitory activity of the compound was tested against rabbit Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087540(3-(3-Carbamimidoyl-phenyl)-5-hydroxymethyl-isoxazo...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087538((4S,5S)-3-(3-Carbamimidoyl-phenyl)-5-methoxymethyl...)
Affinity DataKi:  0.550nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087532(3-(3-Carbamimidoyl-phenyl)-5-methoxymethyl-isoxazo...)
Affinity DataKi:  0.630nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Oryctolagus cuniculus)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087538((4S,5S)-3-(3-Carbamimidoyl-phenyl)-5-methoxymethyl...)
Affinity DataKi:  0.640nMAssay Description:Inhibitory activity of the compound was tested against rabbit Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087535(3-(3-Carbamimidoyl-phenyl)-5-methoxymethyl-isoxazo...)
Affinity DataKi:  0.75nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Oryctolagus cuniculus)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079252(3-(3-Carbamimidoyl-phenyl)-5-methoxymethyl-4,5-dih...)
Affinity DataKi:  0.800nMAssay Description:Inhibitory activity of the compound was tested against rabbit Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079236(3-(3-Carbamimidoyl-phenyl)-5-tetrazol-1-ylmethyl-4...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087539((4S,5R)-3-(3-Carbamimidoyl-phenyl)-5-methyl-4,5-di...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087537((4S,5S)-3-(3-Carbamimidoyl-phenyl)-5-tetrazol-1-yl...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087528(5-Amino-3-(3-carbamimidoyl-phenyl)-isoxazole-4-car...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079252(3-(3-Carbamimidoyl-phenyl)-5-methoxymethyl-4,5-dih...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087534(3-(3-Carbamimidoyl-phenyl)-5-trifluoromethyl-isoxa...)
Affinity DataKi:  9.5nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079247(3-(3-Carbamimidoyl-phenyl)-5-methyl-4,5-dihydro-is...)
Affinity DataKi:  11nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087533(3-(3-Carbamimidoyl-phenyl)-isoxazole-4-carboxylic ...)
Affinity DataKi:  21nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087536(3-(3-Carbamimidoyl-phenyl)-isoxazole-4-carboxylic ...)
Affinity DataKi:  25nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087540(3-(3-Carbamimidoyl-phenyl)-5-hydroxymethyl-isoxazo...)
Affinity DataKi:  50nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079252(3-(3-Carbamimidoyl-phenyl)-5-methoxymethyl-4,5-dih...)
Affinity DataKi:  70nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087532(3-(3-Carbamimidoyl-phenyl)-5-methoxymethyl-isoxazo...)
Affinity DataKi:  76nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079236(3-(3-Carbamimidoyl-phenyl)-5-tetrazol-1-ylmethyl-4...)
Affinity DataKi:  91nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087539((4S,5R)-3-(3-Carbamimidoyl-phenyl)-5-methyl-4,5-di...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087528(5-Amino-3-(3-carbamimidoyl-phenyl)-isoxazole-4-car...)
Affinity DataKi:  117nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079247(3-(3-Carbamimidoyl-phenyl)-5-methyl-4,5-dihydro-is...)
Affinity DataKi:  120nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50115021(1-(3-Cyano-phenyl)-3-{3-[4-(4-fluoro-benzyl)-piper...)
Affinity DataKi:  167nMAssay Description:Inhibition of [125I]-eotaxin binding to serotonin 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50142464(1-(3-Cyano-phenyl)-3-{3-[3-(4-fluoro-benzyl)-pyrro...)
Affinity DataKi:  178nMAssay Description:Inhibition of [125I]-eotaxin binding to serotonin 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087537((4S,5S)-3-(3-Carbamimidoyl-phenyl)-5-tetrazol-1-yl...)
Affinity DataKi:  180nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087538((4S,5S)-3-(3-Carbamimidoyl-phenyl)-5-methoxymethyl...)
Affinity DataKi:  190nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50115023(1-(3-Acetyl-phenyl)-3-{3-[4-(4-fluoro-benzyl)-pipe...)
Affinity DataKi:  193nMAssay Description:Inhibition of [125I]-eotaxin binding to serotonin 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087535(3-(3-Carbamimidoyl-phenyl)-5-methoxymethyl-isoxazo...)
Affinity DataKi:  200nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50115071(1-{3-[4-(4-Fluoro-benzyl)-piperidin-1-yl]-propyl}-...)
Affinity DataKi:  224nMAssay Description:Inhibition of [125I]-eotaxin binding to serotonin 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087534(3-(3-Carbamimidoyl-phenyl)-5-trifluoromethyl-isoxa...)
Affinity DataKi:  400nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087536(3-(3-Carbamimidoyl-phenyl)-isoxazole-4-carboxylic ...)
Affinity DataKi:  540nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50115090(1-[3-(4-Benzyl-piperidin-1-yl)-propyl]-3-(3-methox...)
Affinity DataKi:  613nMAssay Description:Inhibition of [125I]-eotaxin binding to serotonin 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50115010(1-[3-(4-Benzyl-piperidin-1-yl)-propyl]-3-(3-cyano-...)
Affinity DataKi:  770nMAssay Description:Inhibition of [125I]-eotaxin binding to serotonin 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079236(3-(3-Carbamimidoyl-phenyl)-5-tetrazol-1-ylmethyl-4...)
Affinity DataKi:  900nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50142459(1-[3-(3-Benzyl-piperidin-1-yl)-propyl]-3-(3-methox...)
Affinity DataKi:  913nMAssay Description:Inhibition of [125I]-eotaxin binding to serotonin 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50142448((S)-1-(3-(3-(4-fluorobenzyl)piperidin-1-yl)propyl)...)
Affinity DataKi:  1.35E+3nMAssay Description:Inhibition of [125I]-eotaxin binding to serotonin 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087540(3-(3-Carbamimidoyl-phenyl)-5-hydroxymethyl-isoxazo...)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087533(3-(3-Carbamimidoyl-phenyl)-isoxazole-4-carboxylic ...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50142465(1-(3-Cyano-phenyl)-3-{3-[3-(2-fluoro-benzyl)-piper...)
Affinity DataKi:  2.24E+3nMAssay Description:Inhibition of [125I]-eotaxin binding to serotonin 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50142466(1-(3-Cyano-phenyl)-3-{3-[3-(4-fluoro-benzyl)-piper...)
Affinity DataKi:  2.31E+3nMAssay Description:Inhibition of [125I]-eotaxin binding to serotonin 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50142455(1-(3-Cyano-phenyl)-3-{3-[3-(2,4-difluoro-benzyl)-p...)
Affinity DataKi:  2.36E+3nMAssay Description:Inhibition of [125I]-eotaxin binding to serotonin 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079252(3-(3-Carbamimidoyl-phenyl)-5-methoxymethyl-4,5-dih...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50142463(1-[3-(3-Benzyl-piperidin-1-yl)-propyl]-3-(3-cyano-...)
Affinity DataKi:  2.94E+3nMAssay Description:Inhibition of [125I]-eotaxin binding to serotonin 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087532(3-(3-Carbamimidoyl-phenyl)-5-methoxymethyl-isoxazo...)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087528(5-Amino-3-(3-carbamimidoyl-phenyl)-isoxazole-4-car...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087539((4S,5R)-3-(3-Carbamimidoyl-phenyl)-5-methyl-4,5-di...)
Affinity DataKi:  4.50E+3nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087538((4S,5S)-3-(3-Carbamimidoyl-phenyl)-5-methoxymethyl...)
Affinity DataKi:  4.60E+3nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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