TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5086 Cnrs/Universit£
Curated by ChEMBL
Umr 5086 Cnrs/Universit£
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of BCRP expressed in human HEK293 cells assessed as maximal mitoxantrone accumulationMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5086 Cnrs/Universit£
Curated by ChEMBL
Umr 5086 Cnrs/Universit£
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of BCRP expressed in human HEK293 cells assessed as maximal mitoxantrone accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+8nMAssay Description:Inhibition of beta-hematin formation by BHIA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90E+8nMAssay Description:Inhibition of beta-hematin formation by BHIA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.10E+8nMAssay Description:Inhibition of beta-hematin formation by BHIA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.69E+9nMAssay Description:Inhibition of beta-hematin formationMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+9nMAssay Description:Inhibition of beta-hematin formationMore data for this Ligand-Target Pair
Affinity DataIC50: 2.53E+9nMAssay Description:Inhibition of beta-hematin formationMore data for this Ligand-Target Pair