TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Compound was tested for the displacement of [125I]-PYY (SK-N-MC) from Neuropeptide Y receptor type 1 in the membranes prepared from cellsMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Compound was tested for the displacement of [125I]-PYY (SK-N-MC) from Neuropeptide Y receptor type 1 in the membranes prepared from cellsMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Compound was tested for the displacement of [125I]-PYY (SK-N-MC) from Neuropeptide Y receptor type 1 in the membranes prepared from cellsMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Compound was tested for the displacement of [125I]-PYY (SK-N-MC) from Neuropeptide Y receptor type 1 in the membranes prepared from cellsMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataKi: 93nMAssay Description:Compound was tested for the displacement of [125I]-PYY (SK-N-MC) from Neuropeptide Y receptor type 1 in the membranes prepared from cellsMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Compound was tested for the displacement of [125I]-PYY (SK-N-MC) from Neuropeptide Y receptor type 1 in the membranes prepared from cellsMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataKi: 143nMAssay Description:Compound was tested for the displacement of [125I]-PYY (SK-N-MC) from Neuropeptide Y receptor type 1 in the membranes prepared from cellsMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataKi: 621nMAssay Description:Compound was tested for the displacement of [125I]-PYY(3-36) (SK-N-BE2) from Neuropeptide Y receptor type 2 in the membranes prepared from cellsMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataKi: 704nMAssay Description:Compound was tested for the displacement of [125I]-PYY(3-36) (SK-N-BE2) from Neuropeptide Y receptor type 2 in the membranes prepared from cellsMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataKi: 988nMAssay Description:Compound was tested for the displacement of [125I]-PYY(3-36) (SK-N-BE2) from Neuropeptide Y receptor type 2 in the membranes prepared from cellsMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataKi: 2.09E+3nMAssay Description:Compound was tested for the displacement of [125I]-PYY(3-36) (SK-N-BE2) from Neuropeptide Y receptor type 2 in the membranes prepared from cellsMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataKi: 3.41E+3nMAssay Description:Compound was tested for the displacement of [125I]-PYY(3-36) (SK-N-BE2) from Neuropeptide Y receptor type 2 in the membranes prepared from cellsMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataKi: 3.98E+3nMAssay Description:Compound was tested for the displacement of [125I]-PYY(3-36) (SK-N-BE2) from Neuropeptide Y receptor type 2 in the membranes prepared from cellsMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Compound was tested for the displacement of [125I]-PYY(3-36) (SK-N-BE2) from Neuropeptide Y receptor type 2 in the membranes prepared from cellsMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataIC50: 0.0200nMAssay Description:Affinity against Neuropeptide Y receptor Y1 in SK-N-MC cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataIC50: 0.0700nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
Affinity DataIC50: 0.310nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataIC50: 0.320nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 0.360nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataIC50: 0.390nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 0.560nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
Affinity DataIC50: 0.590nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Tested for the affinity for intestinal PYY from rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
Affinity DataIC50: 0.630nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
Affinity DataIC50: 0.910nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataIC50: 0.980nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.05nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 1.07nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.09nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 1.12nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.16nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.32nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.39nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.75nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.83nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.08nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.09nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Tested for the affinity for intestinal PYY from rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
Affinity DataIC50: 2.42nMAssay Description:Tested for the affinity for intestinal PYY from rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.63nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.68nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati Medical Center
Curated by ChEMBL
University Of Cincinnati Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.69nMAssay Description:Affinity against Neuropeptide Y receptor Y1 in SK-N-MC cell lineMore data for this Ligand-Target Pair