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Found 170 with Last Name = 'froissant' and Initial = 'j'
TargetRelaxin receptor 1(Homo sapiens (Human))
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563230(CHEMBL4754949)
Affinity DataKi:  1.10nMAssay Description:Displacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRelaxin receptor 1(Homo sapiens (Human))
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563231(CHEMBL4780098)
Affinity DataKi:  2.88E+3nMAssay Description:Displacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207024(US9233965, 2)
Affinity DataIC50: <1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206926(US9233965, 87)
Affinity DataIC50: <1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207003(US9233965, 86)
Affinity DataIC50: <1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207001(US9233965, 84)
Affinity DataIC50:  1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207020(US9233965, 107)
Affinity DataIC50: <1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207015(US9233965, 100)
Affinity DataIC50: >1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207023(US9233965, 110)
Affinity DataIC50: <1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206925(US9233965, 105)
Affinity DataIC50: <1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206924(US9233965, 104)
Affinity DataIC50: <1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206971(US9233965, 48)
Affinity DataIC50:  1.5nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207005(US9233965, 89)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207002(US9233965, 85)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206915(US9233965, 79)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206920(US9233965, 64)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206981(US9233965, 62)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206928(US9233965, 4)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207019(US9233965, 106)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206998(US9233965, 78)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206984(US9233965, 67)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206939(US9233965, 15)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206923(US9233965, 83)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207021(US9233965, 108)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206935(US9233965, 11)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206951(US9233965, 28)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206955(US9233965, 32)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206986(US9233965, 55)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206980(US9233965, 61)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206983(US9233965, 66)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206990(US9233965, 70)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206991(US9233965, 71)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206995(US9233965, 75)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207000(US9233965, 82)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207004(US9233965, 88)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207007(US9233965, 91)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207014(US9233965, 99)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206996(US9233965, 77)
Affinity DataIC50:  5nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206989(US9233965, 69)
Affinity DataIC50:  5nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206987(US9233965, 54)
Affinity DataIC50:  6nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206994(US9233965, 74)
Affinity DataIC50:  6nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207006(US9233965, 90)
Affinity DataIC50:  6nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206993(US9233965, 73)
Affinity DataIC50:  6nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206916(US9233965, 95)
Affinity DataIC50:  6nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206917(US9233965, 60)
Affinity DataIC50:  7nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206985(US9233965, 53)
Affinity DataIC50:  7nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM206969(US9233965, 46)
Affinity DataIC50:  8nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207017(US9233965, 102)
Affinity DataIC50:  8nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207013(US9233965, 98)
Affinity DataIC50:  9nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM207022(US9233965, 109)
Affinity DataIC50:  9nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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