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Found 186 with Last Name = 'fujisawa' and Initial = 'y'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221787(CHEMBL3216418)
Affinity DataKi:  0.0420nMAssay Description:Compound was tested for Opioid receptor mu 1 agonism in isolated tissues from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221778(CHEMBL3216392)
Affinity DataKi:  0.114nMAssay Description:Compound was tested for binding affinity towards Opioid receptor mu 1 by displacing [3H]DAGO radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221781(CHEMBL3215968)
Affinity DataKi:  0.115nMAssay Description:Compound was tested for Opioid receptor mu 1 agonism in isolated tissues from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221780(CHEMBL3217089)
Affinity DataKi:  1.20nMAssay Description:Compound was tested for binding affinity towards Opioid receptor mu 1 by displacing [3H]DAGO radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221781(CHEMBL3215968)
Affinity DataKi:  7.30nMAssay Description:Compound was tested for binding affinity towards opioid receptor delta 1 by displacing [3H]DPDPE radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221787(CHEMBL3216418)
Affinity DataKi:  13nMAssay Description:pA2 is the negative log of the molar concentration required to double the agonism of opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221780(CHEMBL3217089)
Affinity DataKi:  16nMAssay Description:Compound was tested for binding affinity towards opioid receptor delta 1 by displacing [3H]DPDPE radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221778(CHEMBL3216392)
Affinity DataKi:  23nMAssay Description:Compound was tested for Opioid receptor mu 1 agonism in isolated tissues from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221779(CHEMBL3215974)
Affinity DataKi:  26nMAssay Description:Compound was tested for binding affinity towards Opioid receptor mu 1 by displacing [3H]DAGO radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221782(CHEMBL3215530)
Affinity DataKi:  70nMAssay Description:Compound was tested for binding affinity towards Opioid receptor mu 1 by displacing [3H]DAGO radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50146023(2-Amino-N-[2-(5-{2-[2-amino-3-(4-hydroxy-phenyl)-p...)
Affinity DataKi:  309nMAssay Description:Compound was tested for binding affinity towards Opioid receptor mu 1 by displacing [3H]DAGO radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221779(CHEMBL3215974)
Affinity DataKi:  435nMAssay Description:Compound was tested for binding affinity towards opioid receptor delta 1 by displacing [3H]DPDPE radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50146020(2-Amino-N-(5-{[2-amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  460nMAssay Description:Compound was tested for binding affinity towards Opioid receptor mu 1 by displacing [3H]DAGO radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50146020(2-Amino-N-(5-{[2-amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  1.83E+3nMAssay Description:Compound was tested for binding affinity towards opioid receptor delta 1 by displacing [3H]DPDPE radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221782(CHEMBL3215530)
Affinity DataKi:  2.19E+3nMAssay Description:Compound was tested for binding affinity towards opioid receptor delta 1 by displacing [3H]DPDPE radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50146023(2-Amino-N-[2-(5-{2-[2-amino-3-(4-hydroxy-phenyl)-p...)
Affinity DataKi:  2.90E+3nMAssay Description:Compound was tested for binding affinity towards opioid receptor delta 1 by displacing [3H]DPDPE radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50062810(3-{(S)-1-[2-(4-Carbamimidoyl-benzoylamino)-acetyl]...)
Affinity DataIC50:  0.210nMAssay Description:Ability to inhibit binding of biotin-labeled human fibrinogen to immobilized fibrinogen receptor purified from human erythroleukemia(HEL) cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50062797(3-{(S)-1-[2-(4-Carbamimidoyl-benzoylamino)-acetyl]...)
Affinity DataIC50:  0.290nMAssay Description:Ability to inhibit binding of biotin-labeled human fibrinogen to immobilized fibrinogen receptor purified from human erythroleukemia(HEL) cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50062785(CHEMBL147976 | {4-[2-(4-Carbamimidoyl-benzoylamino...)
Affinity DataIC50:  0.420nMAssay Description:Ability to inhibit binding of biotin-labeled human fibrinogen to immobilized fibrinogen receptor purified from human erythroleukemia(HEL) cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50067612((S)-3-Methyl-2-(naphthalene-1-sulfonylamino)-penta...)
Affinity DataIC50:  0.740nMAssay Description:Inhibition of human cathepsin L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50062803(3-((S)-1-{2-[4-(2-Amino-ethyl)-benzoylamino]-acety...)
Affinity DataIC50:  0.890nMAssay Description:Ability to inhibit binding of biotin-labeled human fibrinogen to immobilized fibrinogen receptor purified from human erythroleukemia(HEL) cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50062789(((S)-4-{2-[4-(2-Amino-ethyl)-benzoylamino]-acetyl}...)
Affinity DataIC50:  0.910nMAssay Description:Ability to inhibit binding of biotin-labeled human fibrinogen to immobilized fibrinogen receptor purified from human erythroleukemia(HEL) cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50062798(CHEMBL148010 | {(S)-4-[2-(4-Carbamimidoyl-benzoyla...)
Affinity DataIC50:  0.920nMAssay Description:Ability to inhibit binding of biotin-labeled human fibrinogen to immobilized fibrinogen receptor purified from human erythroleukemia(HEL) cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50067608((S)-3-Methyl-2-(naphthalene-1-sulfonylamino)-penta...)
Affinity DataIC50:  0.950nMAssay Description:Inhibition of human cathepsin L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50067606((S)-3-Methyl-2-(naphthalene-1-sulfonylamino)-penta...)
Affinity DataIC50:  0.950nMAssay Description:Inhibition of human cathepsin L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50067604((S)-N-[(R)-1-Formyl-2-(1H-indol-3-yl)-ethyl]-3-met...)
Affinity DataIC50:  0.970nMAssay Description:Inhibition of human cathepsin L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50422277(CHEMBL118402)
Affinity DataIC50:  1nMAssay Description:Ability to inhibit binding of biotin-labeled human fibrinogen to immobilized fibrinogen receptor purified from human erythroleukemia(HEL) cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50062783(CHEMBL310081 | TAK-029 | {(S)-1-[2-(4-Carbamimidoy...)
Affinity DataIC50:  1nMAssay Description:Ability to inhibit binding of biotin-labeled human fibrinogen to immobilized fibrinogen receptor purified from human erythroleukemia(HEL) cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50062782(3-((S)-1-{2-[4-(2-Amino-ethyl)-benzoylamino]-acety...)
Affinity DataIC50:  1nMAssay Description:Ability to inhibit binding of biotin-labeled human fibrinogen to immobilized fibrinogen receptor purified from human erythroleukemia(HEL) cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221787(CHEMBL3216418)
Affinity DataIC50:  1.30nMAssay Description:Compound was tested for Opioid receptor mu 1 agonism in isolated tissues from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50067613((S)-3-Methyl-2-(naphthalene-1-sulfonylamino)-penta...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of human cathepsin L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50062787((4-{2-[4-(2-Amino-ethyl)-benzoylamino]-acetyl}-2-o...)
Affinity DataIC50:  1.60nMAssay Description:Ability to inhibit binding of biotin-labeled human fibrinogen to immobilized fibrinogen receptor purified from human erythroleukemia(HEL) cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50369397(CHEMBL1790993)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of human cathepsin L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221778(CHEMBL3216392)
Affinity DataIC50:  1.90nMAssay Description:Compound was tested for Opioid receptor mu 1 agonism in isolated tissues from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50369410(CHEMBL1790989)
Affinity DataIC50:  2nMAssay Description:Inhibition of human cathepsin L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50369405(CHEMBL1790991)
Affinity DataIC50:  2nMAssay Description:Inhibition of human cathepsin L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50369397(CHEMBL1790993)
Affinity DataIC50:  2nMAssay Description:Compound was measured for inhibition of collagenolytic of human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50062791(CHEMBL146393 | {(S)-3-Benzyl-4-[2-(4-carbamimidoyl...)
Affinity DataIC50:  2nMAssay Description:Ability to inhibit binding of biotin-labeled human fibrinogen to immobilized fibrinogen receptor purified from human erythroleukemia(HEL) cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50369402(CHEMBL1790996)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of human cathepsin L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50369400(CHEMBL1791000)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of human cathepsin L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50067597((S)-4-Methyl-2-(naphthalene-1-sulfonylamino)-penta...)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of human cathepsin L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50369403(CHEMBL1790995)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of human cathepsin L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50369398(CHEMBL1790999)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of human cathepsin L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50062781(((S)-1-{2-[4-(2-Amino-ethyl)-benzoylamino]-acetyl}...)
Affinity DataIC50:  2.5nMAssay Description:Ability to inhibit binding of biotin-labeled human fibrinogen to immobilized fibrinogen receptor purified from human erythroleukemia(HEL) cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50286441((S)-2-((S)-2-Acetylamino-4-(S)-methyl-pentanoylami...)
Affinity DataIC50:  2.5nMAssay Description:Compound was measured for inhibition of collagenolytic of human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50067594((S)-3-Methyl-2-(naphthalene-1-sulfonylamino)-penta...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of human cathepsin L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50369406(CHEMBL1791001)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of human cathepsin L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50369408(CHEMBL1790997)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of human cathepsin L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50369409(CHEMBL1791004)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of human cathepsin L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50067614((S)-N-[(R)-1-Formyl-2-(1H-indol-3-yl)-ethyl]-3-(na...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of human cathepsin L.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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