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Found 115 with Last Name = 'gacel' and Initial = 'g'
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018723(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50019055(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of [3H]-DTLET binding torat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50019046(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of [3H]-DTLET binding torat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018707(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  2.20nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  2.20nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018713(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  2.70nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50019051(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  3.10nMAssay Description:Inhibition of [3H]-DTLET binding torat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018715(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  4.20nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50019054(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  4.70nMAssay Description:Inhibition of [3H]-DTLET binding torat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018708(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  4.80nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018708(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  4.80nMAssay Description:Inhibition of [3H]-DTLET binding torat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018717(2-{1-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  5.60nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50019053(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  6.10nMAssay Description:Inhibition of [3H]-DTLET binding torat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50019049(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  6.40nMAssay Description:Inhibition of [3H]-DTLET binding torat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50019056((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataKi:  7.30nMAssay Description:Inhibition of [3H]-DTLET binding torat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018724(2-[2-{2-[2-(2-Amino-3-phenyl-propionylamino)-acety...)
Affinity DataKi:  7.30nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018720(1-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  7.60nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM21025((2R)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydro...)
Affinity DataKi:  7.70nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM21025((2R)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydro...)
Affinity DataKi:  8.40nMAssay Description:Ability to inhibit the binding of [3H]-DAGO to Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018711(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  9.10nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018717(2-{1-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  9.20nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018719(2-Amino-3-(4-hydroxy-phenyl)-N-(1-{[(3-methyl-buty...)
Affinity DataKi:  10nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi:  11nMAssay Description:Inhibition of [3H]-DTLET binding torat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi:  11nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018709(2-Amino-N-(2-tert-butoxy-1-{[(1,3-dimethyl-butylca...)
Affinity DataKi:  14nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018725(2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-N-...)
Affinity DataKi:  15nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018707(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  16nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018721(2-Amino-N-(1-{[(1,3-dimethyl-butylcarbamoyl)-methy...)
Affinity DataKi:  17nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50019050(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi:  19nMAssay Description:Inhibition of [3H]-DTLET binding torat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50019055(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  23nMAssay Description:Inhibition of [3H]-DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018723(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  25nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50019056((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataKi:  28nMAssay Description:Inhibition of [3H]-DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018724(2-[2-{2-[2-(2-Amino-3-phenyl-propionylamino)-acety...)
Affinity DataKi:  28nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018727(2-{2-[2-({2-[2-Amino-3-(4-hydroxy-phenyl)-propiony...)
Affinity DataKi:  30nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018726(2-(2-{[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propi...)
Affinity DataKi:  31nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018708(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  31nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018708(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  31nMAssay Description:Inhibition of [3H]-DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018716(2-Amino-N-[1-({[(1,3-dimethyl-butyl)-ethyl-carbamo...)
Affinity DataKi:  36nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018713(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  38nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018709(2-Amino-N-(2-tert-butoxy-1-{[(1,3-dimethyl-butylca...)
Affinity DataKi:  39nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018715(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  42nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50019046(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  42nMAssay Description:Inhibition of [3H]-DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018722(2-Amino-N-(1-{[(1,3-dimethyl-butylcarbamoyl)-methy...)
Affinity DataKi:  43nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018722(2-Amino-N-(1-{[(1,3-dimethyl-butylcarbamoyl)-methy...)
Affinity DataKi:  43nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018720(1-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  44nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018727(2-{2-[2-({2-[2-Amino-3-(4-hydroxy-phenyl)-propiony...)
Affinity DataKi:  61nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50019051(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  65nMAssay Description:Inhibition of [3H]-DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018714(2-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  116nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018726(2-(2-{[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propi...)
Affinity DataKi:  157nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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