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Found 722 with Last Name = 'gao' and Initial = 'b'

Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

Ki: 0.300nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532486(CHEMBL4564992)

Ki: 0.300nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532506(CHEMBL4536431)

Ki: 0.5nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532508(CHEMBL4471576)

Ki: 0.5nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532506(CHEMBL4536431)

Ki: 0.5nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532518(CHEMBL4440420)

Ki: 0.5nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532508(CHEMBL4471576)

Ki: 0.5nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532518(CHEMBL4440420)

Ki: 0.5nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532502(CHEMBL4538923)

Ki: 0.700nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532502(CHEMBL4538923)

Ki: 0.700nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532512(CHEMBL4539105)

Ki: 0.800nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532512(CHEMBL4539105)

Ki: 0.800nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532507(CHEMBL4593797)

Ki: 0.900nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)

Ki: 0.900nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor (unknown origin) expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair

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3D Structure (crystal)

Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532507(CHEMBL4593797)

Ki: 0.900nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532489(CHEMBL4434692)

Ki: 1.10nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532489(CHEMBL4434692)

Ki: 1.10nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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D(3) dopamine receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50338642((+)-R-11-(3-(4-((4-(2-Methoxyphenyl)piperazin-1-yl...)

Ki: 1.14nMAssay Description:Displacement of [3H]spiperone from dopamine D3 receptor expressed in human HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair

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D(1A) dopamine receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)

Ki: 1.20nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in human HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair

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D(2) dopamine receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)

Ki: 1.20nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor (unknown origin) expressed in human HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532503(CHEMBL4458060)

Ki: 1.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532521(CHEMBL4524740)

Ki: 1.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532521(CHEMBL4524740)

Ki: 1.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532503(CHEMBL4458060)

Ki: 1.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532505(CHEMBL4535404)

Ki: 1.80nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532505(CHEMBL4535404)

Ki: 1.80nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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D(3) dopamine receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50338650((-)-S-11-(3-(4-((4-(2-Methoxyphenyl)piperazin-1-yl...)

Ki: 1.82nMAssay Description:Displacement of [3H]spiperone from dopamine D3 receptor expressed in human HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair

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D(1A) dopamine receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50387561(CHEMBL2057455 | US9359372, DC037079)

Ki: 2.5nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in human HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair

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Sodium-dependent noradrenaline transporter(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL

BDBM35229(3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-met...)

Ki: 2.5nMAssay Description:Displacement of [3H]nisoxetine from human NET expressed in HEK293 cells measured after 30 minsMore data for this Ligand-Target Pair

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Sodium-dependent noradrenaline transporter(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL

BDBM35229(3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-met...)

Ki: 2.5nMAssay Description:Displacement of [3H]nisoxetine from human NET expressed in HEK293 cells measured after 30 minsMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532516(CHEMBL4460187)

Ki: 2.60nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532516(CHEMBL4460187)

Ki: 2.60nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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D(3) dopamine receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50338640((+)-R-11-((1-(3-(4-(2-Methoxyphenyl)piperazin-1-yl...)

Ki: 2.67nMAssay Description:Displacement of [3H]spiperone from dopamine D3 receptor expressed in human HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532493(CHEMBL4533250)

Ki: 2.70nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532493(CHEMBL4533250)

Ki: 2.70nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)

Ki: 2.90nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A receptor (unknown origin) expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532515(CHEMBL4470605)

Ki: 3.20nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532515(CHEMBL4470605)

Ki: 3.20nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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D(1A) dopamine receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50378584(STEPHOLIDINE)

Ki: 3.40nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in human HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532513(CHEMBL4579980)

Ki: 3.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532513(CHEMBL4579980)

Ki: 3.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532501(CHEMBL4452090)

Ki: 3.70nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532501(CHEMBL4452090)

Ki: 3.70nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532497(CHEMBL4447015)

Ki: 4nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532497(CHEMBL4447015)

Ki: 4nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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D(1A) dopamine receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50429044(CHEMBL2334893 | US9359372, DC037029)

Ki: 4.20nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in human HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532517(CHEMBL4454404)

Ki: 4.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532517(CHEMBL4454404)

Ki: 4.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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D(1A) dopamine receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50429057(CHEMBL2334891)

Ki: 4.5nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in human HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532509(CHEMBL4549596)

Ki: 5.30nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Displayed 1 to 50 (of 722 total ) | Next | Last >>

Filter my 722 hits

Targets 85▿
- Sigma intracellular receptor 2 94
- Sigma non-opioid intracellular receptor 1 94
- Epidermal growth factor receptor 50
- D(2) dopamine receptor 44
- D(1A) dopamine receptor 42
- 5-hydroxytryptamine receptor 1A 38
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform 35
- Poly [ADP-ribose] polymerase 2 28
- Poly [ADP-ribose] polymerase 1 28
- Phosphoglycerate mutase 1 24
- D(3) dopamine receptor 20
- Serine/threonine-protein kinase mTOR 20
- Lysine--tRNA ligase 13
- Sodium-dependent serotonin transporter 12
- Tyrosine-protein kinase JAK3 12
- Sodium-dependent noradrenaline transporter 12
- Sodium-dependent dopamine transporter 12
- 5-hydroxytryptamine receptor 2A 8
- Somatostatin receptor type 3 7
- Substance-K receptor 7
- Oxytocin receptor 7
- Atypical chemokine receptor 3 7
- C-C chemokine receptor type 10 7
- Potassium voltage-gated channel subfamily KQT member 2 6
- Potassium voltage-gated channel subfamily B member 2 6
- Potassium voltage-gated channel subfamily KQT member 4 5
- Potassium voltage-gated channel subfamily KQT member 5 4
- Potassium voltage-gated channel subfamily H member 2 4
- Phosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform 3
- Phosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit beta isoform 3
- Protein ENL 3
- Kallikrein-7 3
- Caspase-14 3
- Chymase 3
- Cytochrome P450 1A2 2
- Serine/threonine-protein kinase pim-1 2
- Serine/threonine-protein kinase B-raf 2
- Cytochrome P450 2C8 2
- Focal adhesion kinase 1 2
- Cytochrome P450 2B6 2
- Cytochrome P450 3A4 2
- 3-phosphoinositide-dependent protein kinase 1 1
- Ephrin type-A receptor 1 1
- Tyrosine-protein kinase Fer 1
- Mitogen-activated protein kinase 3 1
- Tyrosine-protein kinase BTK 1
- Proto-oncogene tyrosine-protein kinase ROS 1
- Protein kinase C delta type 1
- Solute carrier organic anion transporter family member 1A4 1
- Tyrosine-protein kinase receptor UFO 1
- Beta-2 adrenergic receptor 1
- Mitogen-activated protein kinase 8 1
- Mast/stem cell growth factor receptor Kit 1
- Ribosomal protein S6 kinase alpha-1 1
- Cyclin-T1/Cyclin-dependent kinase 9 1
- Protein-tyrosine kinase 6 1
- ALK tyrosine kinase receptor 1
- Hepatocyte growth factor receptor 1
- Potassium voltage-gated channel subfamily KQT member 3 1
- Cytochrome P450 2C9 1
- Mitogen-activated protein kinase 14 1
- Aurora kinase A 1
- Potassium voltage-gated channel subfamily KQT member 2/member 3 1
- Glycogen synthase kinase-3 beta 1
- RAC-gamma serine/threonine-protein kinase 1
- Alpha-1A adrenergic receptor 1
- Alpha-1D adrenergic receptor 1
- RAF proto-oncogene serine/threonine-protein kinase 1
- Platelet-derived growth factor receptor alpha 1
- RAC-alpha serine/threonine-protein kinase 1
- Cytochrome P450 4B1 1
- Tyrosine-protein kinase JAK2 1
- Alpha-1B adrenergic receptor 1
- Serine/threonine-protein kinase Chk1 1
- Ephrin type-B receptor 2 1
- Proto-oncogene tyrosine-protein kinase receptor Ret 1
- Polycystin-1 1
- Tyrosine-protein kinase ZAP-70 1
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform 1
- Rho-associated protein kinase 1 1
- Platelet-derived growth factor receptor beta 1
- Proto-oncogene tyrosine-protein kinase Src 1
- Cyclin-dependent kinase 6/G1/S-specific cyclin-D3 1
- Cytochrome P450 2C19 1
- Cytochrome P450 2D6 1
- ...
Publications 16▿
- J Med Chem 59: 6329-43 (2016) 224
- Bioorg Med Chem 70: (2022) 78
- Bioorg Med Chem 21: 856-68 (2013) 69
- Bioorg Med Chem Lett 31: (2021) 59
- Bioorg Med Chem 19: 1999-2008 (2011) 46
- J Med Chem 61: 6364-6378 (2018) 44
- J Med Chem 54: 4324-38 (2011) 41
- ACS Med Chem Lett 9: 256-261 (2018) 41
- J Nat Prod 81: 998-1006 (2018) 35
- Bioorg Med Chem Lett 36: (2021) 24
- Eur J Med Chem 209: (2021) 23
- J Med Chem 64: 5816-5837 (2021) 15
- ACS Med Chem Lett 10: 27-33 (2019) 13
- J Med Chem 50: 83-93 (2007) 6
- J Nat Prod 85: 317-326 (2022) 3
- Invest Ophthalmol Vis Sci 43: 510-4 (2002) 1
Institutions 11▿
- East China Normal University 224
- Chinese Academy Of Sciences 157
- Southeast University 78
- Central South University 59
- University Of Florida 44
- Wuxi Apptec (Shanghai) Co. 41
- Soochow University College Of Pharmaceutical Sciences 41
- Yunnan University 38
- China Pharmaceutical University 24
- Shanghai Institute Of Materia Medica 15
- University Hospital 1
Affinity: 0.050 to 5.2E+5 nM▿
- Ki 363
- IC50 326
- Kd 1
- EC50 32
- Affinity ≤ nM
Xtal structures: 11
Docked structures: 1
Catalog Cmpds: 48