TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Northeastern University
Curated by ChEMBL
Northeastern University
Curated by ChEMBL
Affinity DataKi: 0.0340nMAssay Description:Compound was evaluated for its ability to inhibit Striatal Dopamine Receptor in rat brain through radioreceptor assay carried out with agonist ligand...More data for this Ligand-Target Pair
Affinity DataKi: 0.0530nMAssay Description:Binding affinity at rat striatal Dopamine receptor D2 using [3H]- piperone radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Binding affinity at rat striatal Dopamine receptor D2 using [3H]- piperone radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Dopamine receptor D2 affinity was tested in vitro against corpus striatum from rat brain membranesMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Northeastern University
Curated by ChEMBL
Northeastern University
Curated by ChEMBL
Affinity DataKi: 0.230nMAssay Description:Agonist activity was tested in vitro against Dopamine receptor from rat brain membranes with [3H]ADT-6,7-dihydroxy-2-aminotetralin]More data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Compound was evaluated for its ability to inhibit Dopamine receptor D2 in rat striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Dopamine receptor D2 affinity was tested in vitro against corpus striatum from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Binding affinity at rat striatal Dopamine receptor D2 using [3H]- piperone radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Dopamine receptor D2 affinity was tested in vitro against corpus striatum from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Dopamine receptor D2 affinity was tested in vitro against corpus striatum from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity at rat striatal Dopamine receptor D2 using [3H]- piperone radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Compound was evaluated for its ability to inhibit dopamine receptor D2 in rat striatum using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Compound was evaluated for its ability to inhibit Dopamine receptor D2 in rat striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity at rat striatal Dopamine receptor D2 using [3H]- piperone radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Agonistic activity against calf striatal Dopamine receptor using [3H]- ADTN radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Agonistic activity against calf striatal Dopamine receptor using [3H]- ADTN radioligandMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Northeastern University
Curated by ChEMBL
Northeastern University
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Compound was evaluated for its ability to inhibit Striatal Dopamine Receptor in rat brain through radioreceptor assay carried out with agonist ligand...More data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Northeastern University
Curated by ChEMBL
Northeastern University
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Agonist activity was tested in vitro against Dopamine receptor from rat brain membranes with [3H]ADT-6,7-dihydroxy-2-aminotetralin]More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Compound was evaluated for its ability to inhibit dopamine receptor D2 in rat striatum using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Agonistic activity against calf striatal Dopamine receptor using [3H]- ADTN radioligandMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Northeastern University
Curated by ChEMBL
Northeastern University
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:Agonist activity was tested in vitro against Dopamine receptor from rat brain membranes with [3H]ADT-6,7-dihydroxy-2-aminotetralin]More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Agonistic activity against calf striatal Dopamine receptor using [3H]- ADTN radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Agonistic activity against calf striatal Dopamine receptor using [3H]- ADTN radioligandMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Northeastern University
Curated by ChEMBL
Northeastern University
Curated by ChEMBL
Affinity DataKi: 4.20nMAssay Description:Agonist activity was tested in vitro against Dopamine receptor from rat brain membranes with [3H]ADT-6,7-dihydroxy-2-aminotetralin]More data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Northeastern University
Curated by ChEMBL
Northeastern University
Curated by ChEMBL
Affinity DataKi: 4.20nMAssay Description:Compound was evaluated for its ability to inhibit Striatal Dopamine receptor in rat brain through radioreceptor assay carried out with agonist ligand...More data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Northeastern University
Curated by ChEMBL
Northeastern University
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Compound was evaluated for its ability to inhibit Striatal Dopamine receptor in rat brain through radioreceptor assay carried out with agonist ligand...More data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Northeastern University
Curated by ChEMBL
Northeastern University
Curated by ChEMBL
Affinity DataKi: 9.80nMAssay Description:Agonist activity was tested in vitro against Dopamine receptor from rat brain membranes with [3H]ADT-6,7-dihydroxy-2-aminotetralin]More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity at rat striatal Dopamine receptor D2 using [3H]- piperone radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Dopamine receptor D2 affinity was tested in vitro against corpus striatum from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Compound was evaluated for its ability to inhibit dopamine receptor D2 in rat striatum using [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Northeastern University
Curated by ChEMBL
Northeastern University
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Agonist activity was tested in vitro against Dopamine receptor from rat brain membranes with [3H]ADT-6,7-dihydroxy-2-aminotetralin]More data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Northeastern University
Curated by ChEMBL
Northeastern University
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Agonist activity was tested in vitro against Dopamine receptor from rat brain membranes with [3H]ADT-6,7-dihydroxy-2-aminotetralin]More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Agonistic activity against calf striatal Dopamine receptor using [3H]- ADTN radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity at rat striatal Dopamine receptor D2 using [3H]- piperone radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinity at rat striatal Dopamine receptor D2 using [3H]- piperone radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Binding affinity at rat striatal Dopamine receptor D2 using [3H]- piperone radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Compound was evaluated for its ability to inhibit Dopamine receptor D2 in rat striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Compound was evaluated for its ability to inhibit dopamine receptor D2 in rat striatum using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Agonistic activity against calf striatal Dopamine receptor using [3H]- ADTN radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Binding affinity at rat striatal Dopamine receptor D2 using [3H]- piperone radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Binding affinity at rat striatal Dopamine receptor D1 using [3H]- SCH-23390 radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity at rat striatal Dopamine receptor D2 using [3H]- piperone radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 106nMAssay Description:Binding affinity at rat striatal Dopamine receptor D1 using [3H]- SCH-23390 radioligandMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Northeastern University
Curated by ChEMBL
Northeastern University
Curated by ChEMBL
Affinity DataKi: 112nMAssay Description:Compound was evaluated for its ability to inhibit Striatal Dopamine Receptor in rat brain through radioreceptor assay carried out with agonist ligand...More data for this Ligand-Target Pair
Affinity DataKi: 124nMAssay Description:Dopamine receptor D1 affinity was tested in vitro against corpus striatum from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 155nMAssay Description:Compound was evaluated for its ability to inhibit dopamine receptor D2 in rat striatum using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 162nMAssay Description:Agonistic activity against calf striatal Dopamine receptor using [3H]- ADTN radioligandMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Northeastern University
Curated by ChEMBL
Northeastern University
Curated by ChEMBL
Affinity DataKi: 199nMAssay Description:Agonist activity was tested in vitro against Dopamine receptor from rat brain membranes with [3H]ADT-6,7-dihydroxy-2-aminotetralin]More data for this Ligand-Target Pair
Affinity DataKi: 236nMAssay Description:Binding affinity at rat striatal Dopamine receptor D1 using [3H]- SCH-23390 radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Dopamine receptor D1 affinity was tested in vitro against corpus striatum from rat brain membranesMore data for this Ligand-Target Pair