Affinity DataKi: 3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 104nMAssay Description:Displacement of [3H]Win55212 form human CB2 receptor transfected in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 312nMAssay Description:Displacement of [3H]CP55940 form human CB2 receptor transfected in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.65E+3nMAssay Description:Displacement of [3H]Win55212 form human CB2 receptor transfected in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]CP55940 form human CB2 receptor transfected in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 form human CB2 receptor transfected in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Win55212 form human CB2 receptor transfected in HEK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20nMAssay Description:Antagonist activity at rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of C-terminal histidine-tagged caspase-3 using Ac-DEVD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Antagonist activity at rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of C-terminal histidine-tagged caspase-3 using Ac-DEVD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Antagonist activity at rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Antagonist activity at rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of C-terminal FLAG-tagged human caspase-3 expressed in HEK293 T17 cells using Ac-DEVD-AMC coumarin-120 as substrate pre-incubated for 2 hr...More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of C-terminal histidine-tagged caspase-3 using Ac-DEVD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of C-terminal histidine-tagged caspase-3 using Ac-DEVD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Antagonist activity at human histamine H3 receptorMore data for this Ligand-Target Pair