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Found 156 with Last Name = 'giberson' and Initial = 'km'
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50178679(2-[[(3S,4S)-4-(4-chlorophenyl)-1-methylpiperidin-3...)
Affinity DataKi:  3.90nMAssay Description:Ability to inhibit [3H]DA uptake through DAT in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166332(9-[1-(3'-Fluoro-biphenyl-4-yl)-meth-(Z)-ylidene]-7...)
Affinity DataKi:  5nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166328(9-[3-(2,6-Difluoro-phenyl)-prop-2-yn-(Z)-ylidene]-...)
Affinity DataKi:  5.30nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50178663(2-[(3R,4R)-4-(4-chlorophenyl)-1-methylpiperidin-3-...)
Affinity DataKi:  5.5nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166336(9-[1-[2,3']Bithiophenyl-5-yl-meth-(Z)-ylidene]-7-a...)
Affinity DataKi:  5.90nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166339(9-[1-(2'-Methoxy-biphenyl-4-yl)-meth-(Z)-ylidene]-...)
Affinity DataKi:  6.5nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM35229(3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-met...)
Affinity DataKi:  7.36nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50178665(2-[(3S,4S)-4-(4-chlorophenyl)-1-methylpiperidin-3-...)
Affinity DataKi:  8.80nMAssay Description:Ability to inhibit [3H]5HT uptake through SERT in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166333(9-[1-(3'-Trifluoromethyl-biphenyl-4-yl)-meth-(Z)-y...)
Affinity DataKi:  8.80nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166334(9-[1-(3'-Methoxy-biphenyl-4-yl)-meth-(Z)-ylidene]-...)
Affinity DataKi:  9.40nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50178661(2-[(3R,4R)-4-(4-chlorophenyl)-1-methylpiperidin-3-...)
Affinity DataKi:  11nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50178667(2-[(3S,4S)-4-(4-chlorophenyl)-1-methylpiperidin-3-...)
Affinity DataKi:  13nMAssay Description:Ability to inhibit [3H]DA uptake through DAT in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50178657(2-[(3S,4S)-4-(4-chlorophenyl)-1-methylpiperidin-3-...)
Affinity DataKi:  13nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50178667(2-[(3S,4S)-4-(4-chlorophenyl)-1-methylpiperidin-3-...)
Affinity DataKi:  16nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50166341(9-[3-(4-Fluoro-phenyl)-prop-2-yn-(Z)-ylidene]-7-az...)
Affinity DataKi:  17nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50178665(2-[(3S,4S)-4-(4-chlorophenyl)-1-methylpiperidin-3-...)
Affinity DataKi:  17nMAssay Description:Ability to inhibit [3H]DA uptake through DAT in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50178653(2-[(3S,4S)-4-(4-chlorophenyl)-1-methylpiperidin-3-...)
Affinity DataKi:  18nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50178655(2-[[(3S,4S)-4-(4-chlorophenyl)-1-methylpiperidin-3...)
Affinity DataKi:  21nMAssay Description:Ability to inhibit [3H]5HT uptake through SERT in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166329(9-[3-Thiophen-3-yl-prop-2-yn-(Z)-ylidene]-7-aza-tr...)
Affinity DataKi:  22nMAssay Description:Inhibitory constant for [3H]-NE reuptake at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50178669(2-[[(3R,4R)-4-(4-chlorophenyl)-1-methylpiperidin-3...)
Affinity DataKi:  22nMAssay Description:Ability to inhibit [3H]5HT uptake through SERT in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50178668(CHEMBL370401 | [(3S,4S)-4-(4-chlorophenyl)-1-methy...)
Affinity DataKi:  22nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50178658(2-[[(3S,4R)-4-(4-chlorophenyl)-1-methylpiperidin-3...)
Affinity DataKi:  23nMAssay Description:Ability to inhibit [3H]DA uptake through DAT in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50178679(2-[[(3S,4S)-4-(4-chlorophenyl)-1-methylpiperidin-3...)
Affinity DataKi:  23nMAssay Description:Ability to inhibit [3H]5HT uptake through SERT in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50178664(2-[[(3S,4S)-4-(4-chlorophenyl)-1-methylpiperidin-3...)
Affinity DataKi:  26nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50178662(CHEMBL200056 | acetic acid 2-[[(3S,4S)-4-(4-chloro...)
Affinity DataKi:  30nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50166328(9-[3-(2,6-Difluoro-phenyl)-prop-2-yn-(Z)-ylidene]-...)
Affinity DataKi:  32nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50178659(2-[[(3S,4R)-4-(4-chlorophenyl)-1-methylpiperidin-3...)
Affinity DataKi:  32nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50166336(9-[1-[2,3']Bithiophenyl-5-yl-meth-(Z)-ylidene]-7-a...)
Affinity DataKi:  32nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50178657(2-[(3S,4S)-4-(4-chlorophenyl)-1-methylpiperidin-3-...)
Affinity DataKi:  34nMAssay Description:Ability to inhibit [3H]DA uptake through DAT in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50178661(2-[(3R,4R)-4-(4-chlorophenyl)-1-methylpiperidin-3-...)
Affinity DataKi:  36nMAssay Description:Ability to inhibit [3H]5HT uptake through SERT in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50178664(2-[[(3S,4S)-4-(4-chlorophenyl)-1-methylpiperidin-3...)
Affinity DataKi:  37nMAssay Description:Ability to inhibit [3H]DA uptake through DAT in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50178668(CHEMBL370401 | [(3S,4S)-4-(4-chlorophenyl)-1-methy...)
Affinity DataKi:  38nMAssay Description:Ability to inhibit [3H]DA uptake through DAT in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50178657(2-[(3S,4S)-4-(4-chlorophenyl)-1-methylpiperidin-3-...)
Affinity DataKi:  42nMAssay Description:Ability to inhibit [3H]5HT uptake through SERT in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50178652(2-[[(3S,4R)-4-(4-chlorophenyl)-1-methylpiperidin-3...)
Affinity DataKi:  44nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50178662(CHEMBL200056 | acetic acid 2-[[(3S,4S)-4-(4-chloro...)
Affinity DataKi:  46nMAssay Description:Ability to inhibit [3H]DA uptake through DAT in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50178654(2-[(3R,4R)-4-(4-chlorophenyl)-1-methylpiperidin-3-...)
Affinity DataKi:  47nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166330(9-[3-(3-Fluoro-4-methyl-phenyl)-prop-2-yn-(Z)-ylid...)
Affinity DataKi:  52nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50178656(CHEMBL197013 | acetic acid 2-[[(3S,4R)-4-(4-chloro...)
Affinity DataKi:  52nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50178680(2-[[(3S,4R)-4-(4-chlorophenyl)-1-methylpiperidin-3...)
Affinity DataKi:  53nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166326(9-[1-(4'-Fluoro-biphenyl-4-yl)-meth-(Z)-ylidene]-7...)
Affinity DataKi:  53nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50178655(2-[[(3S,4S)-4-(4-chlorophenyl)-1-methylpiperidin-3...)
Affinity DataKi:  54nMAssay Description:Ability to inhibit [3H]DA uptake through DAT in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50178669(2-[[(3R,4R)-4-(4-chlorophenyl)-1-methylpiperidin-3...)
Affinity DataKi:  54nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50178672((3R,4R)-methyl 4-(4-chlorophenyl)-1-methylpiperidi...)
Affinity DataKi:  56nMAssay Description:Ability to inhibit [3H]5HT uptake through SERT in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50178650(CHEMBL200713 | benzoic acid 2-[[(3S,4R)-4-(4-chlor...)
Affinity DataKi:  56nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50178676(CHEMBL198641 | [(3S,4R)-4-(4-chlorophenyl)-1-methy...)
Affinity DataKi:  57nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166327(9-[1-(4'-Methylsulfanyl-biphenyl-4-yl)-meth-(Z)-yl...)
Affinity DataKi:  62nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50178665(2-[(3S,4S)-4-(4-chlorophenyl)-1-methylpiperidin-3-...)
Affinity DataKi:  63nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50178678(2-[[(3S,4R)-4-(4-chlorophenyl)-1-methylpiperidin-3...)
Affinity DataKi:  67nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50178658(2-[[(3S,4R)-4-(4-chlorophenyl)-1-methylpiperidin-3...)
Affinity DataKi:  68nMAssay Description:Ability to inhibit [3H]5HT uptake through SERT in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50166337(9-[3-(3,4-Difluoro-phenyl)-prop-2-yn-(Z)-ylidene]-...)
Affinity DataKi:  69nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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