TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Ability to inhibit [3H]DA uptake through DAT in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
Affinity DataKi: 7.36nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 8.80nMAssay Description:Ability to inhibit [3H]5HT uptake through SERT in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 8.80nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Ability to inhibit [3H]DA uptake through DAT in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Ability to inhibit [3H]DA uptake through DAT in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Ability to inhibit [3H]5HT uptake through SERT in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Inhibitory constant for [3H]-NE reuptake at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Ability to inhibit [3H]5HT uptake through SERT in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Ability to inhibit [3H]DA uptake through DAT in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Ability to inhibit [3H]5HT uptake through SERT in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 34nMAssay Description:Ability to inhibit [3H]DA uptake through DAT in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Ability to inhibit [3H]5HT uptake through SERT in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Ability to inhibit [3H]DA uptake through DAT in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Ability to inhibit [3H]DA uptake through DAT in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Ability to inhibit [3H]5HT uptake through SERT in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Ability to inhibit [3H]DA uptake through DAT in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 54nMAssay Description:Ability to inhibit [3H]DA uptake through DAT in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 56nMAssay Description:Ability to inhibit [3H]5HT uptake through SERT in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 67nMAssay Description:Ability to inhibit [3H]NE uptake through NET in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 68nMAssay Description:Ability to inhibit [3H]5HT uptake through SERT in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 69nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair