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Found 67 with Last Name = 'gil' and Initial = 'mj'
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120056(15-Amino-1-methyl-10-thia-tricyclo[7.5.1.0*2,7*]pe...)
Affinity DataKi:  0.790nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120057(7-Amino-8,8-dimethyl-6-methylsulfanyl-5,6,7,8-tetr...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120058(7-Amino-6-methoxy-8,8-dimethyl-5,6,7,8-tetrahydro-...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173870(3-Benzyloxy-1,1-dioxo-2,3-dihydro-1H-1lambda*6*-be...)
Affinity DataKi:  2.80nMAssay Description:Inhibitory activity against catalytic domain of human cloned Carbonic anhydrase IX by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173865(3-Butoxy-1,1-dioxo-2,3-dihydro-1H-1lambda*6*-benzo...)
Affinity DataKi:  3.10nMAssay Description:Inhibitory activity against catalytic domain of human cloned Carbonic anhydrase IX by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  4nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173865(3-Butoxy-1,1-dioxo-2,3-dihydro-1H-1lambda*6*-benzo...)
Affinity DataKi:  6.30nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase II by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173871(1,1-Dioxo-1H-1lambda*6*-benzo[b]thiophene-5-sulfon...)
Affinity DataKi:  7.40nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase II by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173862(1,1-Dioxo-1H-1lambda*6*-benzo[b]thiophene-6-sulfon...)
Affinity DataKi:  7.5nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase II by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173870(3-Benzyloxy-1,1-dioxo-2,3-dihydro-1H-1lambda*6*-be...)
Affinity DataKi:  7.90nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase II by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM10882(6-ethoxy-1,3-benzothiazole-2-sulfonamide | CHEMBL1...)
Affinity DataKi:  8nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase II by the CO2 hydration methodMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173867(3-Methyl-1,1-dioxo-1H-1lambda*6*-benzo[b]thiophene...)
Affinity DataKi:  8.30nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase II by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173864(1,1-Dioxo-2,3-dihydro-1H-1lambda*6*-benzo[b]thioph...)
Affinity DataKi:  8.80nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase II by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173864(1,1-Dioxo-2,3-dihydro-1H-1lambda*6*-benzo[b]thioph...)
Affinity DataKi:  10nMAssay Description:Inhibitory activity against catalytic domain of human cloned Carbonic anhydrase IX by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  12nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase II by the CO2 hydration methodMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173871(1,1-Dioxo-1H-1lambda*6*-benzo[b]thiophene-5-sulfon...)
Affinity DataKi:  13nMAssay Description:Inhibitory activity against catalytic domain of human cloned Carbonic anhydrase IX by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173867(3-Methyl-1,1-dioxo-1H-1lambda*6*-benzo[b]thiophene...)
Affinity DataKi:  13nMAssay Description:Inhibitory activity against catalytic domain of human cloned Carbonic anhydrase IX by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM10881(CHEMBL288100 | MZA3 | Methazolamide | Methazolamid...)
Affinity DataKi:  14nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase II by the CO2 hydration methodMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173862(1,1-Dioxo-1H-1lambda*6*-benzo[b]thiophene-6-sulfon...)
Affinity DataKi:  15nMAssay Description:Inhibitory activity against catalytic domain of human cloned Carbonic anhydrase IX by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM10890(1-N-(3-chloro-1H-indol-7-yl)benzene-1,4-disulfonam...)
Affinity DataKi:  15nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase II by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120053(7-Amino-6-ethyl-8,8-dimethyl-5,6,7,8-tetrahydro-na...)
Affinity DataKi:  21nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM10890(1-N-(3-chloro-1H-indol-7-yl)benzene-1,4-disulfonam...)
Affinity DataKi:  24nMAssay Description:Inhibitory activity against catalytic domain of human cloned Carbonic anhydrase IX by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  25nMAssay Description:Inhibitory activity against catalytic domain of human cloned Carbonic anhydrase IX by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM10882(6-ethoxy-1,3-benzothiazole-2-sulfonamide | CHEMBL1...)
Affinity DataKi:  25nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase I by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM10881(CHEMBL288100 | MZA3 | Methazolamide | Methazolamid...)
Affinity DataKi:  27nMAssay Description:Inhibitory activity against catalytic domain of human cloned Carbonic anhydrase IX by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM10890(1-N-(3-chloro-1H-indol-7-yl)benzene-1,4-disulfonam...)
Affinity DataKi:  31nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase I by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM10882(6-ethoxy-1,3-benzothiazole-2-sulfonamide | CHEMBL1...)
Affinity DataKi:  34nMAssay Description:Inhibitory activity against catalytic domain of human cloned Carbonic anhydrase IX by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM10883(4,5-dichlorobenzene-1,3-disulfonamide | CHEMBL17 |...)
Affinity DataKi:  38nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase II by the CO2 hydration methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120056(15-Amino-1-methyl-10-thia-tricyclo[7.5.1.0*2,7*]pe...)
Affinity DataKi:  43nMAssay Description:Binding affinity of the compound for Opioid receptor kappa 1 was determined.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM10883(4,5-dichlorobenzene-1,3-disulfonamide | CHEMBL17 |...)
Affinity DataKi:  50nMAssay Description:Inhibitory activity against catalytic domain of human cloned Carbonic anhydrase IX by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  52nMAssay Description:Binding affinity of the compound for Opioid receptor kappa 1 was determined.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCarbonic anhydrase 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173862(1,1-Dioxo-1H-1lambda*6*-benzo[b]thiophene-6-sulfon...)
Affinity DataKi:  63nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase I by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120057(7-Amino-8,8-dimethyl-6-methylsulfanyl-5,6,7,8-tetr...)
Affinity DataKi:  66nMAssay Description:Binding affinity of the compound for Opioid receptor kappa 1 was determined.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173864(1,1-Dioxo-2,3-dihydro-1H-1lambda*6*-benzo[b]thioph...)
Affinity DataKi:  72nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase I by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173871(1,1-Dioxo-1H-1lambda*6*-benzo[b]thiophene-5-sulfon...)
Affinity DataKi:  75nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase I by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173869(1,1-Dioxo-1H-1lambda*6*-benzo[b]thiophene-6-sulfon...)
Affinity DataKi:  76nMAssay Description:Inhibitory activity against catalytic domain of human cloned Carbonic anhydrase IX by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173867(3-Methyl-1,1-dioxo-1H-1lambda*6*-benzo[b]thiophene...)
Affinity DataKi:  85nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase I by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173865(3-Butoxy-1,1-dioxo-2,3-dihydro-1H-1lambda*6*-benzo...)
Affinity DataKi:  104nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase I by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  113nMAssay Description:Binding affinity of the compound for Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120061(7-Amino-6-ethyl-8,8-dimethyl-5,6,7,8-tetrahydro-na...)
Affinity DataKi:  135nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173870(3-Benzyloxy-1,1-dioxo-2,3-dihydro-1H-1lambda*6*-be...)
Affinity DataKi:  138nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase I by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120062(7-Amino-6-mercapto-8,8-dimethyl-5,6,7,8-tetrahydro...)
Affinity DataKi:  163nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120058(7-Amino-6-methoxy-8,8-dimethyl-5,6,7,8-tetrahydro-...)
Affinity DataKi:  184nMAssay Description:Binding affinity of the compound for Opioid receptor kappa 1 was determined.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120054(3-Amino-4,4-dimethyl-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataKi:  204nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120059(7-Amino-8,8-dimethyl-6-methylsulfanyl-5,6,7,8-tetr...)
Affinity DataKi:  286nMAssay Description:Binding affinity for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120053(7-Amino-6-ethyl-8,8-dimethyl-5,6,7,8-tetrahydro-na...)
Affinity DataKi:  345nMAssay Description:Binding affinity of the compound for Opioid receptor kappa 1 was determined.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120057(7-Amino-8,8-dimethyl-6-methylsulfanyl-5,6,7,8-tetr...)
Affinity DataKi:  349nMAssay Description:Binding affinity of the compound for Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173868(1,1-Dioxo-1H-1lambda*6*-benzo[b]thiophene-6-sulfon...)
Affinity DataKi:  362nMAssay Description:Inhibitory activity against catalytic domain of human cloned Carbonic anhydrase IX by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50120056(15-Amino-1-methyl-10-thia-tricyclo[7.5.1.0*2,7*]pe...)
Affinity DataKi:  420nMAssay Description:Binding affinity of the compound for Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50173868(1,1-Dioxo-1H-1lambda*6*-benzo[b]thiophene-6-sulfon...)
Affinity DataKi:  436nMAssay Description:Inhibitory activity against human cloned Carbonic anhydrase II by the CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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