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Found 216 with Last Name = 'giupponi' and Initial = 'l'
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371684(CHEMBL270666)
Affinity DataKi:  5.70nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371688(CHEMBL404545)
Affinity DataKi:  7.5nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371686(CHEMBL271876)
Affinity DataKi:  40nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222142((S,E)-2-amino-N-(2-(benzyloxy)-1-(1-cinnamyl-1H-te...)
Affinity DataKi:  190nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371687(CHEMBL272085)
Affinity DataKi:  197nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222164((S)-2-amino-N-(2-(benzyloxy)-1-(1-(3-phenylpropyl)...)
Affinity DataKi:  200nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222164((S)-2-amino-N-(2-(benzyloxy)-1-(1-(3-phenylpropyl)...)
Affinity DataKi:  200nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371683(CHEMBL410060)
Affinity DataKi:  240nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371693(CHEMBL402086)
Affinity DataKi:  298nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222147((S)-benzyl 5-(5-(1-(2-amino-2-methylpropanamido)-2...)
Affinity DataKi:  320nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222136(CHEMBL235793 | methyl 2-(5-((S)-1-(2-amino-2-methy...)
Affinity DataKi:  470nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371685(CHEMBL270876)
Affinity DataKi:  503nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371691(CHEMBL270851)
Affinity DataKi:  611nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371689(CHEMBL256235)
Affinity DataKi:  696nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371689(CHEMBL256235)
Affinity DataKi:  696nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371697(CHEMBL404336)
Affinity DataKi:  737nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371697(CHEMBL404336)
Affinity DataKi:  737nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222157(2-amino-N-{(S)-2-benzyloxy-1-[1-(2-phenethylcarbam...)
Affinity DataKi:  780nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222166(2-amino-N-((S)-2-benzyloxy-1-{1-[2-(3-phenyl-propy...)
Affinity DataKi:  820nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222162((S)-2-amino-N-(2-(benzyloxy)-1-(1-(2-(1-(methylsul...)
Affinity DataKi:  970nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222167(2-amino-N-{(S)-1-[1-(2-benzylcarbamoyl-ethyl)-1H-t...)
Affinity DataKi:  1.07E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222173((S)-2-amino-N-(2-(benzyloxy)-1-(2-(2-(1-(methylsul...)
Affinity DataKi:  1.27E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222150(2-amino-N-{(R)-1-[1-(2-butylcarbamoyl-ethyl)-1H-te...)
Affinity DataKi:  1.37E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371695(CHEMBL403180)
Affinity DataKi:  1.38E+3nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371695(CHEMBL403180)
Affinity DataKi:  1.38E+3nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222151(2-amino-N-((S)-2-(benzyloxy)-1-(1-((1-(methylsulfo...)
Affinity DataKi:  1.59E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222161((S)-2-amino-N-(2-(benzyloxy)-1-(1-(3-(2-(N-methylm...)
Affinity DataKi:  1.72E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222146((S)-4-(5-(1-(2-amino-2-methylpropanamido)-2-(benzy...)
Affinity DataKi:  1.78E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222153((S)-2-amino-N-(1-(1-benzyl-1H-tetrazol-5-yl)-2-(be...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222165(2-amino-N-{(S)-2-benzyloxy-1-[1-(2-butylcarbamoyl-...)
Affinity DataKi:  2.19E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222143((S)-N-(1-(1-(2-(methylsulfonamido)phenethyl)-1H-te...)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222172((S)-methyl 4-(5-(1-(2-amino-2-methylpropanamido)-2...)
Affinity DataKi:  2.38E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222158((S)-2-amino-N-(2-(benzyloxy)-1-(2-(3-(2-(methylsul...)
Affinity DataKi:  2.39E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371696(CHEMBL271082)
Affinity DataKi:  2.51E+3nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371696(CHEMBL271082)
Affinity DataKi:  2.51E+3nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222139((S)-N-(1-(2-(2-(methylsulfonamido)phenethyl)-2H-te...)
Affinity DataKi:  2.66E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222148((S)-2-amino-N-(2-(benzyloxy)-1-(1-(2-cyanoethyl)-1...)
Affinity DataKi:  2.94E+3nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222148((S)-2-amino-N-(2-(benzyloxy)-1-(1-(2-cyanoethyl)-1...)
Affinity DataKi:  2.94E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222156((S)-2-amino-N-(2-(benzyloxy)-1-(1-(4-cyanobutyl)-1...)
Affinity DataKi:  3.12E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222171((S)-methyl 3-(5-(1-(2-amino-2-methylpropanamido)-2...)
Affinity DataKi:  3.38E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371694(CHEMBL402808)
Affinity DataKi:  3.94E+3nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371694(CHEMBL402808)
Affinity DataKi:  3.94E+3nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222149((S)-2-amino-N-(2-(benzyloxy)-1-(1-(cyanomethyl)-1H...)
Affinity DataKi:  4.17E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222141((S)-N-(1-(1-(2-(methylsulfonamido)benzyl)-1H-tetra...)
Affinity DataKi:  4.45E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222168((S)-2-amino-N-(1-(2-benzyl-2H-tetrazol-5-yl)-2-(be...)
Affinity DataKi:  4.75E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222144((S)-N-(1-(2-(3-(methylsulfonamido)benzyl)-2H-tetra...)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222152(2-amino-N-((S)-2-(benzyloxy)-1-(2-((1-(methylsulfo...)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371692(CHEMBL404227)
Affinity DataKi: >5.00E+3nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50222154((S)-N-(1-(1-(4-(methylsulfonamido)benzyl)-1H-tetra...)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50371690(CHEMBL256236)
Affinity DataKi: >5.00E+3nMAssay Description:Agonist activity at human GHS receptor expressed in H4 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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