Affinity DataKi: 3nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago
Curated by ChEMBL
University Of Santiago
Curated by ChEMBL
Affinity DataKi: 52nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Rattus norvegicus)
Experimental Sugar Cane Station&Quot;Villa Clara-Cienfuegos&Quot
Curated by ChEMBL
Experimental Sugar Cane Station&Quot;Villa Clara-Cienfuegos&Quot
Curated by ChEMBL
Affinity DataKi: 54.1nMAssay Description:Displacement of radioligand [125I]AB-MECA binding at rat A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 81nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Rattus norvegicus)
Experimental Sugar Cane Station&Quot;Villa Clara-Cienfuegos&Quot
Curated by ChEMBL
Experimental Sugar Cane Station&Quot;Villa Clara-Cienfuegos&Quot
Curated by ChEMBL
Affinity DataKi: 107nMAssay Description:Displacement of radioligand [125I]AB-MECA binding at rat A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 129nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 135nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago
Curated by ChEMBL
University Of Santiago
Curated by ChEMBL
Affinity DataKi: 138nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Rattus norvegicus)
Experimental Sugar Cane Station&Quot;Villa Clara-Cienfuegos&Quot
Curated by ChEMBL
Experimental Sugar Cane Station&Quot;Villa Clara-Cienfuegos&Quot
Curated by ChEMBL
Affinity DataKi: 155nMAssay Description:Displacement of radioligand [125I]AB-MECA binding at rat A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 165nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago
Curated by ChEMBL
University Of Santiago
Curated by ChEMBL
Affinity DataKi: 174nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 175nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 194nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 215nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 266nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 324nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Rattus norvegicus)
Experimental Sugar Cane Station&Quot;Villa Clara-Cienfuegos&Quot
Curated by ChEMBL
Experimental Sugar Cane Station&Quot;Villa Clara-Cienfuegos&Quot
Curated by ChEMBL
Affinity DataKi: 405nMAssay Description:Displacement of radioligand [125I]AB-MECA binding at rat A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 447nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 523nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago
Curated by ChEMBL
University Of Santiago
Curated by ChEMBL
Affinity DataKi: 537nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 554nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 562nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 741nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 747nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago
Curated by ChEMBL
University Of Santiago
Curated by ChEMBL
Affinity DataKi: 933nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago
Curated by ChEMBL
University Of Santiago
Curated by ChEMBL
Affinity DataKi: 1.07E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago
Curated by ChEMBL
University Of Santiago
Curated by ChEMBL
Affinity DataKi: 1.95E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago
Curated by ChEMBL
University Of Santiago
Curated by ChEMBL
Affinity DataKi: 2.34E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Central University Of Las Villas
Curated by ChEMBL
Central University Of Las Villas
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Displacement of [3H]R-N6-phenylisopropyladenosine from adenosine A1 receptor in rat cerebral cortical membraneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago
Curated by ChEMBL
University Of Santiago
Curated by ChEMBL
Affinity DataKi: 3.09E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Central University Of Las Villas
Curated by ChEMBL
Central University Of Las Villas
Curated by ChEMBL
Affinity DataKi: 8.12E+3nMAssay Description:Displacement of [3H]R-N6-phenylisopropyladenosine from adenosine A1 receptor in rat cerebral cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Central University Of Las Villas
Curated by ChEMBL
Central University Of Las Villas
Curated by ChEMBL
Affinity DataKi: 2.55E+4nMAssay Description:Displacement of [3H]R-N6-phenylisopropyladenosine from adenosine A1 receptor in rat cerebral cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Central University Of Las Villas
Curated by ChEMBL
Central University Of Las Villas
Curated by ChEMBL
Affinity DataKi: 3.23E+4nMAssay Description:Displacement of [3H]R-N6-phenylisopropyladenosine from adenosine A1 receptor in rat cerebral cortical membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of human p38alpha using biotinylated ATF2 as substrate preincubated for 1 hr measured after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of human p38alpha using biotinylated ATF2 substrate by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of human p38alpha using biotinylated ATF2 substrate by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Inhibition of human p38alpha using biotinylated ATF2 as substrate preincubated for 1 hr measured after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Inhibition of human p38alpha by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human p38alpha using biotinylated ATF2 as substrate preincubated for 1 hr measured after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.640nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human p38alpha using biotinylated ATF2 substrate by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.830nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibition of human p38alpha by FRET assayMore data for this Ligand-Target Pair