Affinity DataKi: 9.73nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Inhibition of [3H]R-PIA binding to Adenosine A1 receptor from rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 16.3nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 17.1nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 20.9nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 38.3nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Noncompetitive inhibition of electric eel AchE using acetylcholine as substrate preincubated for 15 mins followed by substrate addition measured for ...More data for this Ligand-Target Pair
Affinity DataKi: 54.1nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 54.1nMAssay Description:Displacement of radioligand [125I]AB-MECA binding at rat A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 77.6nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 81nMAssay Description:Mixed-type inhibition of electric eel AChE using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 89.5nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 107nMAssay Description:Displacement of radioligand [125I]AB-MECA binding at rat A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 107nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 149nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 154nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 155nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 155nMAssay Description:Displacement of radioligand [125I]AB-MECA binding at rat A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 167nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 168nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 211nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 247nMAssay Description:Inhibition of [3H]R-PIA binding to Adenosine A1 receptor from rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 251nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 292nMAssay Description:Inhibition of [3H]R-PIA binding to Adenosine A1 receptor from rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 315nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 319nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 324nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 405nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 405nMAssay Description:Displacement of radioligand [125I]AB-MECA binding at rat A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 411nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 532nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 581nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 611nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 696nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 713nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 725nMAssay Description:Inhibition of [3H]R-PIA binding to Adenosine A1 receptor from rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 754nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 824nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 837nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 901nMAssay Description:Inhibition of [3H]R-PIA binding to Adenosine A1 receptor from rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 979nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Displacement of [3H]R-N6-phenylisopropyladenosine from adenosine A1 receptor in rat cerebral cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 5.55E+3nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.70E+3nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 8.12E+3nMAssay Description:Displacement of [3H]R-N6-phenylisopropyladenosine from adenosine A1 receptor in rat cerebral cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 1.44E+4nMAssay Description:Inhibition of [3H]R-PIA binding to Adenosine A1 receptor from rat brain membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 2.55E+4nMAssay Description:Displacement of [3H]R-N6-phenylisopropyladenosine from adenosine A1 receptor in rat cerebral cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 3.23E+4nMAssay Description:Displacement of [3H]R-N6-phenylisopropyladenosine from adenosine A1 receptor in rat cerebral cortical membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Concentration required for 50% inhibition of the adenosine kinase (AK) activity.More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Concentration required for 50% inhibition of the adenosine kinase (AK) activity.More data for this Ligand-Target Pair