Affinity DataKi: 6.10nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 410nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 710nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 940nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:In vitro inhibition of human fibroblast collagenase.More data for this Ligand-Target Pair
Affinity DataKi: 4.60E+3nMAssay Description:In vitro inhibition of human recombinant stromelysin-1.More data for this Ligand-Target Pair
Affinity DataKi: 5.10E+3nMAssay Description:In vitro inhibition of human fibroblast collagenase.More data for this Ligand-Target Pair
Affinity DataKi: 7.50E+3nMAssay Description:In vitro inhibition of human fibroblast collagenase.More data for this Ligand-Target Pair
Affinity DataKi: 1.59E+4nMAssay Description:In vitro inhibition of human fibroblast collagenase.More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of DiTc binding to Kv1.3 channel in human brain membranesMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of DiTc binding to Kv1.3 channel in human brain membranesMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of Kv1.3 ion channel. Measured in the Rb_Kv assay: [86Rb+] efflux from CHO cells stably transfected with Kv1.3 channel.More data for this Ligand-Target Pair