Compile Data Set for Download or QSAR
maximum 50k data
Found 74 with Last Name = 'graves' and Initial = 'd'
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM10759(2-acetoxyethyl(trimethyl)ammonium;bromide | 2-acet...)
Affinity DataIC50:  12nMAssay Description:Compound was tested in vitro for its binding affinity to muscarinic acetylcholine receptor from rat cortical homogenates using [3H]OXO-M as radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50005677(CHEMBL23957 | OXO-M | Trimethyl-[4-(2-oxo-pyrrolid...)
Affinity DataIC50:  13nMAssay Description:Compound was tested in vitro for its binding affinity to muscarinic acetylcholine receptor from rat cortical homogenates using [3H]OXO-M as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50229526(CHEMBL279356)
Affinity DataIC50:  14nMAssay Description:In vitro inhibition of [3H]OXO-M binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004665((oxotremorine)1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyr...)
Affinity DataIC50:  17nMAssay Description:In vitro inhibition of [3H]OXO-M binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50229691(CHEMBL23118)
Affinity DataIC50:  30nMAssay Description:Compound was tested in vitro for its binding affinity to muscarinic acetylcholine receptor from rat cortical homogenates using [3H]OXO-M as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50229697(CHEMBL23721)
Affinity DataIC50:  48nMAssay Description:In vitro inhibition of [3H]OXO-M binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50229618(CHEMBL23335)
Affinity DataIC50:  75nMAssay Description:In vitro inhibition of [3H]OXO-M binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM46858(1-methyl-3,6-dihydro-2H-pyridine-5-carboxylic acid...)
Affinity DataIC50:  115nMAssay Description:In vitro inhibition of [3H]OXO-M binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50229688(CHEMBL276975)
Affinity DataIC50:  140nMAssay Description:In vitro inhibition of [3H]OXO-M binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50230645(CHEMBL434772)
Affinity DataIC50:  170nMAssay Description:In vitro inhibition of [3H]OXO-M binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataIC50:  213nMAssay Description:In vitro inhibition of [3H]QNB binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50229667(CHEMBL23563)
Affinity DataIC50:  240nMAssay Description:In vitro inhibition of [3H]OXO-M binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataIC50:  322nMAssay Description:In vitro inhibition of [3H]OXO-M binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50230639(CHEMBL23172)
Affinity DataIC50:  430nMAssay Description:Compound was tested in vitro for its binding affinity to muscarinic acetylcholine receptor from rat cortical homogenates using [3H]OXO-M as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataIC50:  670nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50230644(CHEMBL429230)
Affinity DataIC50:  930nMAssay Description:In vitro inhibition of [3H]OXO-M binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
CSIR, Pretoria (Za)

US Patent
LigandPNGBDBM2195(SM36 | US8501787, 171)
Affinity DataIC50:  1.43E+3nMAssay Description:The assay is based on a sandwich-ELISA protocol employing the ROCHE colorimetric reverse transcriptase kit (cat # 1468120910).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
CSIR, Pretoria (Za)

US Patent
LigandPNGBDBM2184(SM30 | US8501787, 166)
Affinity DataIC50:  1.55E+3nMAssay Description:The assay is based on a sandwich-ELISA protocol employing the ROCHE colorimetric reverse transcriptase kit (cat # 1468120910).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetReverse transcriptase(Human immunodeficiency virus 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM2184(SM30 | US8501787, 166)
Affinity DataIC50:  1.55E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50230645(CHEMBL434772)
Affinity DataIC50:  1.60E+3nMAssay Description:In vitro inhibition of [3H]QNB binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50229526(CHEMBL279356)
Affinity DataIC50:  1.80E+3nMAssay Description:In vitro inhibition of [3H]QNB binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50230642(CHEMBL282490)
Affinity DataIC50:  2.30E+3nMAssay Description:Compound was tested in vitro for its binding affinity to muscarinic acetylcholine receptor from rat cortical homogenates using [3H]OXO-M as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50229691(CHEMBL23118)
Affinity DataIC50:  2.80E+3nMAssay Description:Compound was tested in vitro for its binding affinity to muscarinic acetylcholine receptor from rat cortical homogenates using [3H]QNB as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004665((oxotremorine)1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyr...)
Affinity DataIC50:  3.30E+3nMAssay Description:In vitro inhibition of [3H]QNB binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50230640(CHEMBL22926)
Affinity DataIC50:  3.40E+3nMAssay Description:In vitro inhibition of [3H]OXO-M binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM2173(CW23836 | US8501787, 116)
Affinity DataIC50:  3.47E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
CSIR, Pretoria (Za)

US Patent
LigandPNGBDBM2173(CW23836 | US8501787, 116)
Affinity DataIC50:  3.47E+3nMAssay Description:The assay is based on a sandwich-ELISA protocol employing the ROCHE colorimetric reverse transcriptase kit (cat # 1468120910).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
CSIR, Pretoria (Za)

US Patent
LigandPNGBDBM2172(DG 402-49748 | US8501787, 104)
Affinity DataIC50:  3.74E+3nMAssay Description:The assay is based on a sandwich-ELISA protocol employing the ROCHE colorimetric reverse transcriptase kit (cat # 1468120910).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetReverse transcriptase(Human immunodeficiency virus 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM2172(DG 402-49748 | US8501787, 104)
Affinity DataIC50:  3.74E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
CSIR, Pretoria (Za)

US Patent
LigandPNGBDBM2115(MLB133-641A | US8501787, 8)
Affinity DataIC50:  4.39E+3nMAssay Description:The assay is based on a sandwich-ELISA protocol employing the ROCHE colorimetric reverse transcriptase kit (cat # 1468120910).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetReverse transcriptase(Human immunodeficiency virus 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM2115(MLB133-641A | US8501787, 8)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50229697(CHEMBL23721)
Affinity DataIC50:  4.50E+3nMAssay Description:In vitro inhibition of [3H]QNB binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50229618(CHEMBL23335)
Affinity DataIC50:  4.50E+3nMAssay Description:In vitro inhibition of [3H]QNB binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50230638(CHEMBL278352)
Affinity DataIC50:  4.60E+3nMAssay Description:In vitro inhibition of [3H]OXO-M binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
CSIR, Pretoria (Za)

US Patent
LigandPNGBDBM2116(DG 402-49706 | US8501787, 42)
Affinity DataIC50:  4.62E+3nMAssay Description:The assay is based on a sandwich-ELISA protocol employing the ROCHE colorimetric reverse transcriptase kit (cat # 1468120910).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetReverse transcriptase(Human immunodeficiency virus 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM2116(DG 402-49706 | US8501787, 42)
Affinity DataIC50:  4.62E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50230641(CHEMBL23222)
Affinity DataIC50:  5.00E+3nMAssay Description:In vitro inhibition of [3H]OXO-M binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50229688(CHEMBL276975)
Affinity DataIC50:  5.10E+3nMAssay Description:In vitro inhibition of [3H]QNB binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
CSIR, Pretoria (Za)

US Patent
LigandPNGBDBM2126(DG 402-49760 | US8501787, 48)
Affinity DataIC50:  5.14E+3nMAssay Description:The assay is based on a sandwich-ELISA protocol employing the ROCHE colorimetric reverse transcriptase kit (cat # 1468120910).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetReverse transcriptase(Human immunodeficiency virus 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM2177(SM27 | US8501787, 163)
Affinity DataIC50:  5.39E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
CSIR, Pretoria (Za)

US Patent
LigandPNGBDBM2177(SM27 | US8501787, 163)
Affinity DataIC50:  5.39E+3nMAssay Description:The assay is based on a sandwich-ELISA protocol employing the ROCHE colorimetric reverse transcriptase kit (cat # 1468120910).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50230637(CHEMBL23962)
Affinity DataIC50:  6.50E+3nMAssay Description:In vitro inhibition of [3H]OXO-M binding to Muscarinic receptor from rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
CSIR, Pretoria (Za)

US Patent
LigandPNGBDBM99893(US8501767, 96)
Affinity DataIC50:  6.60E+3nMAssay Description:The assay is based on a sandwich-ELISA protocol employing the ROCHE colorimetric reverse transcriptase kit (cat # 1468120910).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetReverse transcriptase(Human immunodeficiency virus 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM99893(US8501767, 96)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50230636(CHEMBL23901)
Affinity DataIC50:  6.70E+3nMAssay Description:Compound was tested in vitro for its binding affinity to muscarinic acetylcholine receptor from rat cortical homogenates using [3H]OXO-M as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
CSIR, Pretoria (Za)

US Patent
LigandPNGBDBM2182(SM29 | US8501787, 165)
Affinity DataIC50:  7.18E+3nMAssay Description:The assay is based on a sandwich-ELISA protocol employing the ROCHE colorimetric reverse transcriptase kit (cat # 1468120910).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetReverse transcriptase(Human immunodeficiency virus 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM2182(SM29 | US8501787, 165)
Affinity DataIC50:  7.18E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
CSIR, Pretoria (Za)

US Patent
LigandPNGBDBM2162(DG 402-49754 | US8501787, 97)
Affinity DataIC50:  7.52E+3nMAssay Description:The assay is based on a sandwich-ELISA protocol employing the ROCHE colorimetric reverse transcriptase kit (cat # 1468120910).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetReverse transcriptase(Human immunodeficiency virus 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM2162(DG 402-49754 | US8501787, 97)
Affinity DataIC50:  7.52E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
CSIR, Pretoria (Za)

US Patent
LigandPNGBDBM2117(DG 402-49651 | US8501787, 43)
Affinity DataIC50:  1.00E+4nMAssay Description:The assay is based on a sandwich-ELISA protocol employing the ROCHE colorimetric reverse transcriptase kit (cat # 1468120910).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 74 total ) | Next | Last >>
Jump to: