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Found 8 with Last Name = 'guiffant' and Initial = 'd'
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Cnrs Usr-3151

Curated by ChEMBL
LigandPNGBDBM7377(4-{7-butyl-5H-pyrrolo[2,3-b]pyrazin-6-yl}phenol | ...)
Affinity DataIC50:  200nMAssay Description:Inhibition of GST-fused recombinant CDK5/p25 expressed in Escherichia coli after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Cnrs Usr-3151

Curated by ChEMBL
LigandPNGBDBM50295352(2-(2-{2-[4-(7-Butyl-5H-pyrrolo[2,3-b]pyrazin-6-yl)...)
Affinity DataIC50:  660nMAssay Description:Inhibition of GST-fused recombinant CDK5/p25 expressed in Escherichia coli after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Saccharomyces cerevisiae)
Cnrs Usr-3151

Curated by ChEMBL
LigandPNGBDBM7377(4-{7-butyl-5H-pyrrolo[2,3-b]pyrazin-6-yl}phenol | ...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of hemagglutinin-tagged Saccharomyces cerevisiae MNY629 Cdc28/Clb2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Cnrs Usr-3151

Curated by ChEMBL
LigandPNGBDBM50295354(2-(1-{2-[2-(2-Aminoethoxy)ethoxy]ethyl}-1H-[1,2,3]...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-fused recombinant CDK5/p25 expressed in Escherichia coli after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Cnrs Usr-3151

Curated by ChEMBL
LigandPNGBDBM50295355(2-(1-{2-[2-(2-Aminoethoxy)ethoxy]ethyl}-1H-[1,2,3]...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-fused recombinant CDK5/p25 expressed in Escherichia coli after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Saccharomyces cerevisiae)
Cnrs Usr-3151

Curated by ChEMBL
LigandPNGBDBM50295351(CHEMBL560452 | N-methyl-aloisine A)
Affinity DataIC50: >3.30E+4nMAssay Description:Inhibition of hemagglutinin-tagged Saccharomyces cerevisiae MNY629 Cdc28/Clb2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Cnrs Usr-3151

Curated by ChEMBL
LigandPNGBDBM50295353(2-(2-{2-[4-(7-Butyl-5-methyl-5H-pyrrolo[2,3-b]pyra...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of GST-fused recombinant CDK5/p25 expressed in Escherichia coli after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Cnrs Usr-3151

Curated by ChEMBL
LigandPNGBDBM50295351(CHEMBL560452 | N-methyl-aloisine A)
Affinity DataIC50:  1.60E+5nMAssay Description:Inhibition of GST-fused recombinant CDK5/p25 expressed in Escherichia coli after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed