Compile Data Set for Download or QSAR
maximum 50k data
Found 57 with Last Name = 'guillard' and Initial = 'j'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM28798((2S)-2-ethoxy-3-(4-{2-[4-(methanesulfonyloxy)pheny...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234375((S)-2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)met...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294690((S)-2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)met...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294688((S)-3-(4-(2-(6-((benzyloxyimino)(phenyl)methyl)-4,...)
Affinity DataKi:  18.4nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294692((S)-3-(4-(2-(6-((methoxyimino)(phenyl)methyl)-4,4-...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234377(2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)methyl)...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294691((S)-2-(2-benzoylphenylamino)-3-(4-(2-(6-((methoxyi...)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294689((S)-3-(4-(2-(6-((allyloxyimino)(phenyl)methyl)-4,4...)
Affinity DataKi:  54.2nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234372((R)-2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)met...)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294693((S)-3-(4-(2-(6-((cyclopropylmethoxyimino)(phenyl)m...)
Affinity DataKi:  254nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234373(CHEMBL253851 | ethyl 2-ethoxy-3-(4-(2-(6-((hydroxy...)
Affinity DataKi:  618nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50437446(CHEMBL2409341)
Affinity DataKi:  4.60E+3nMAssay Description:Inhibition of bovine kidney alpha-L-fucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234376(CHEMBL252996 | dimethyl 2-(4-(2-(6-((hydroxyimino)...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234374((S)-ethyl 2-ethoxy-3-(4-(2-(6-((methoxyimino)(phen...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294695((S)-2-acetoxy-3-(4-(2-(6-((methoxyimino)(phenyl)me...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294694((S)-2-(2-ethoxy-2-oxoethylamino)-3-(4-(2-(6-((hydr...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234379(CHEMBL252995 | dimethyl 2-(4-(2-(6-benzoyl-4,4-dim...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234378(CHEMBL399629 | ethyl 2-ethoxy-3-(4-(2-(6-((methoxy...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-galactosidase(Coffea arabica (Coffee beans))
Universit£

Curated by ChEMBL
LigandPNGBDBM50437446(CHEMBL2409341)
Affinity DataKi:  5.40E+4nMAssay Description:Inhibition of coffee bean alpha-galactosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50437448(CHEMBL2409344)
Affinity DataIC50:  7.20E+4nMAssay Description:Inhibition of bovine kidney alpha-L-fucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50437447(CHEMBL2409343)
Affinity DataIC50:  2.08E+5nMAssay Description:Inhibition of bovine kidney alpha-L-fucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50437451(CHEMBL2409348)
Affinity DataIC50:  4.87E+5nMAssay Description:Inhibition of bovine liver beta-glucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-galactosidase(Bos taurus (Bovine))
Universit£

Curated by ChEMBL
LigandPNGBDBM50437451(CHEMBL2409348)
Affinity DataIC50:  5.26E+5nMAssay Description:Inhibition of bovine liver beta-galactosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-galactosidase(Bos taurus (Bovine))
Universit£

Curated by ChEMBL
LigandPNGBDBM50437450(CHEMBL2409346)
Affinity DataIC50:  5.41E+5nMAssay Description:Inhibition of bovine liver beta-galactosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50437449(CHEMBL2409342)
Affinity DataIC50:  7.13E+5nMAssay Description:Inhibition of bovine kidney alpha-L-fucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234375((S)-2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)met...)
Affinity DataEC50:  114nMAssay Description:Agonist activity at human PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM28798((2S)-2-ethoxy-3-(4-{2-[4-(methanesulfonyloxy)pheny...)
Affinity DataEC50:  37nMAssay Description:Agonist activity at human PPARalpha at 100 uM by GAL4 transactivation assay relative to WY 14,643More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234377(2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)methyl)...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294691((S)-2-(2-benzoylphenylamino)-3-(4-(2-(6-((methoxyi...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human PPARalpha by Gal4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294692((S)-3-(4-(2-(6-((methoxyimino)(phenyl)methyl)-4,4-...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARalpha by Gal4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294693((S)-3-(4-(2-(6-((cyclopropylmethoxyimino)(phenyl)m...)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human PPARalpha by Gal4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294688((S)-3-(4-(2-(6-((benzyloxyimino)(phenyl)methyl)-4,...)
Affinity DataEC50:  34nMAssay Description:Agonist activity at human PPARalpha by Gal4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294689((S)-3-(4-(2-(6-((allyloxyimino)(phenyl)methyl)-4,4...)
Affinity DataEC50:  73nMAssay Description:Agonist activity at human PPARalpha by Gal4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294690((S)-2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)met...)
Affinity DataEC50:  114nMAssay Description:Agonist activity at human PPARalpha by Gal4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294694((S)-2-(2-ethoxy-2-oxoethylamino)-3-(4-(2-(6-((hydr...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human PPARgamma by Gal4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294691((S)-2-(2-benzoylphenylamino)-3-(4-(2-(6-((methoxyi...)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human PPARgamma by Gal4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294692((S)-3-(4-(2-(6-((methoxyimino)(phenyl)methyl)-4,4-...)
Affinity DataEC50:  125nMAssay Description:Agonist activity at human PPARgamma by Gal4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294693((S)-3-(4-(2-(6-((cyclopropylmethoxyimino)(phenyl)m...)
Affinity DataEC50:  7.52nMAssay Description:Agonist activity at human PPARgamma by Gal4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294688((S)-3-(4-(2-(6-((benzyloxyimino)(phenyl)methyl)-4,...)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human PPARgamma by Gal4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294689((S)-3-(4-(2-(6-((allyloxyimino)(phenyl)methyl)-4,4...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human PPARgamma by Gal4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50294690((S)-2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)met...)
Affinity DataEC50:  7.85nMAssay Description:Agonist activity at human PPARgamma by Gal4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234375((S)-2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)met...)
Affinity DataEC50:  7.90nMAssay Description:Agonist activity at human PPARalpha at 100 uM by GAL4 transactivation assay relative to WY 14,643More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM28798((2S)-2-ethoxy-3-(4-{2-[4-(methanesulfonyloxy)pheny...)
Affinity DataEC50:  414nMAssay Description:Agonist activity at human PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234373(CHEMBL253851 | ethyl 2-ethoxy-3-(4-(2-(6-((hydroxy...)
Affinity DataEC50:  189nMAssay Description:Agonist activity at human PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234372((R)-2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)met...)
Affinity DataEC50:  194nMAssay Description:Agonist activity at human PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234374((S)-ethyl 2-ethoxy-3-(4-(2-(6-((methoxyimino)(phen...)
Affinity DataEC50:  29nMAssay Description:Agonist activity at human PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234374((S)-ethyl 2-ethoxy-3-(4-(2-(6-((methoxyimino)(phen...)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human PPARalpha at 100 uM by GAL4 transactivation assay relative to WY 14,643More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234373(CHEMBL253851 | ethyl 2-ethoxy-3-(4-(2-(6-((hydroxy...)
Affinity DataEC50:  48nMAssay Description:Agonist activity at human PPARalpha at 100 uM by GAL4 transactivation assay relative to WY 14,643More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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