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Found 25 with Last Name = 'gunatilaka' and Initial = 'aa'
TargetAndrogen receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM18161((1S,2S,7S,10R,11S,14S,15S)-14-hydroxy-2,15-dimethy...)
Affinity DataIC50:  13nMAssay Description:Competitive inhibition of androgen binding to androgen receptor (unknown origin) by invitrogen polar screen assayMore data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50114395(CHEMBL3605564)
Affinity DataIC50:  580nMAssay Description:Inhibition of androgen receptor in human LNCAP cells assessed as inhibition of DHT-induced KLK2 gene expression by Array Plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50114397(CHEMBL3605563)
Affinity DataIC50:  620nMAssay Description:Inhibition of androgen receptor in human LNCAP cells assessed as inhibition of DHT-induced KLK2 gene expression by Array Plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50114395(CHEMBL3605564)
Affinity DataIC50:  750nMAssay Description:Inhibition of androgen receptor in human LNCAP cells assessed as inhibition of DHT-induced KLK3 gene expression by Array Plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50114395(CHEMBL3605564)
Affinity DataIC50:  770nMAssay Description:Inhibition of androgen receptor in human LNCAP cells assessed as inhibition of DHT-induced SPDEF gene expression by Array Plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50114397(CHEMBL3605563)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of androgen receptor in human LNCAP cells assessed as inhibition of DHT-induced SPDEF gene expression by Array Plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50114397(CHEMBL3605563)
Affinity DataIC50:  1.42E+3nMAssay Description:Inhibition of androgen receptor in human LNCAP cells assessed as inhibition of DHT-induced KLK3 gene expression by Array Plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50112125(CHEMBL3605562)
Affinity DataIC50:  1.79E+3nMAssay Description:Inhibition of androgen receptor in human LNCAP cells assessed as inhibition of DHT-induced KLK2 gene expression by Array Plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50114392(CHEMBL3605560)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of androgen receptor in human LNCAP cells assessed as inhibition of DHT-induced KLK2 gene expression by Array Plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50112125(CHEMBL3605562)
Affinity DataIC50:  2.72E+3nMAssay Description:Inhibition of androgen receptor in human LNCAP cells assessed as inhibition of DHT-induced SPDEF gene expression by Array Plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50114392(CHEMBL3605560)
Affinity DataIC50:  3.28E+3nMAssay Description:Inhibition of androgen receptor in human LNCAP cells assessed as inhibition of DHT-induced SPDEF gene expression by Array Plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50114392(CHEMBL3605560)
Affinity DataIC50:  3.52E+3nMAssay Description:Inhibition of androgen receptor in human LNCAP cells assessed as inhibition of DHT-induced KLK3 gene expression by Array Plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50112125(CHEMBL3605562)
Affinity DataIC50:  3.58E+3nMAssay Description:Inhibition of androgen receptor in human LNCAP cells assessed as inhibition of DHT-induced KLK3 gene expression by Array Plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 6(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50231326(CHEMBL4073317)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of SHP1 (unknown origin) expressed in Escherichia coli BL21(DE3) using pNPP as substrate preincubated for 15 mins followed by substrate ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50231326(CHEMBL4073317)
Affinity DataIC50:  1.37E+4nMAssay Description:Inhibition of PTP1B (unknown origin) expressed in Escherichia coli BL21(DE3) using pNPP as substrate preincubated for 15 mins followed by substrate a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50231326(CHEMBL4073317)
Affinity DataIC50:  1.66E+4nMAssay Description:Inhibition of TCPTP (unknown origin) expressed in Escherichia coli BL21(DE3) using pNPP as substrate preincubated for 15 mins followed by substrate a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50250932(CHEMBL465251 | demethylzeylasterone)
Affinity DataIC50:  1.76E+4nMAssay Description:Inhibition of human topoisomerase 2 p170alpha assessed as relaxation of lambda ZAPII plasmid Bluescript KS+ DNA by SDS electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50163869(CHEMBL3800252)
Affinity DataIC50:  3.12E+4nMAssay Description:Inhibition of p97 (unknown origin) ATPase activity after 10 mins by malachite green dye based visible spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50478501(10-Hydroxyliriodenine | CHEMBL499126)
Affinity DataIC50:  4.46E+4nMAssay Description:Inhibition of DNA topoisomerase 2 assessed as bacteriophage P4 DNA unknotting after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50478502(10-Methoxyliriodenine | CHEMBL471281)
Affinity DataIC50:  8.18E+4nMAssay Description:Inhibition of DNA topoisomerase 2 assessed as bacteriophage P4 DNA unknotting after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50493008(CHEMBL1797186)
Affinity DataEC50:  2.40E+4nMAssay Description:Inhibition of HSP90 in human MCF7 cells assessed as depletion of cell surface HER2 protein level after 18 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50493009(CHEMBL2420692)
Affinity DataEC50:  4.10E+4nMAssay Description:Inhibition of HSP90 in human MCF7 cells assessed as depletion of cell surface HER2 protein level after 18 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50493010(CHEMBL2420690)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of HSP90 in human MCF7 cells assessed as depletion of cell surface HER2 protein level after 18 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50493011(CHEMBL2420691)
Affinity DataEC50:  3.80E+4nMAssay Description:Inhibition of HSP90 in human MCF7 cells assessed as depletion of cell surface HER2 protein level after 18 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50493012(CHEMBL2420689)
Affinity DataEC50:  2.00E+4nMAssay Description:Inhibition of HSP90 in human MCF7 cells assessed as depletion of cell surface HER2 protein level after 18 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed