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Found 35 with Last Name = 'gustafson' and Initial = 'jl'
TargetSerine/threonine-protein kinase LMTK3(Homo sapiens)
San Diego State University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  0.00200nMAssay Description:Inhibition of LMTK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))TBA
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of BLK (unknown origin) incubated for 1 hr in presence of ATP by Z'LYTE assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))TBA
LigandPNGBDBM50614535(CHEMBL5271284)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of BTK (unknown origin) by Z'LYTE assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytoplasmic tyrosine-protein kinase BMX(Homo sapiens (Human))TBA
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of BMX (unknown origin) incubated for 1 hr in presence of ATP by Z'LYTE assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytoplasmic tyrosine-protein kinase BMX(Homo sapiens (Human))TBA
LigandPNGBDBM50614535(CHEMBL5271284)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of BMX (unknown origin) by Z'LYTE assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))TBA
LigandPNGBDBM50614535(CHEMBL5271284)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of BLK (unknown origin) by Z'LYTE assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))TBA
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of BTK (unknown origin) using Blk/Lyntide as substrate preincubated for 1 hr followed by substrate addition and measured after 2 hrs in pr...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))TBA
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of ITK (unknown origin) using Blk/Lyntide as substrate preincubated for 1 hr followed by substrate addition and measured after 2 hrs in pr...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of EGFR (unknown origin) incubated for 1 hr in presence of ATP by Z'LYTE assayMore data for this Ligand-Target Pair
TargetCytoplasmic tyrosine-protein kinase BMX(Homo sapiens (Human))TBA
LigandPNGBDBM50614536(CHEMBL5278149)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of BMX (unknown origin) by Z'LYTE assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))TBA
LigandPNGBDBM50614536(CHEMBL5278149)
Affinity DataIC50:  13nMAssay Description:Inhibition of BTK (unknown origin) by Z'LYTE assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetTyrosine-protein kinase HCK(Homo sapiens (Human))TBA
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)
Affinity DataIC50:  29nMAssay Description:Inhibition of HCK (unknown origin) incubated for 1 hr in presence of ATP by Z'LYTE assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTyrosine-protein kinase HCK(Homo sapiens (Human))TBA
LigandPNGBDBM50614535(CHEMBL5271284)
Affinity DataIC50:  30nMAssay Description:Inhibition of HCK (unknown origin) by Z'LYTE assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))TBA
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)
Affinity DataIC50:  33nMAssay Description:Inhibition of JAK3 (unknown origin) incubated for 1 hr in presence of ATP by Z'LYTE assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))TBA
LigandPNGBDBM50614535(CHEMBL5271284)
Affinity DataIC50:  34nMAssay Description:Inhibition of SRC (unknown origin) by Z'LYTE assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))TBA
LigandPNGBDBM50614536(CHEMBL5278149)
Affinity DataIC50:  36nMAssay Description:Inhibition of BLK (unknown origin) by Z'LYTE assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))TBA
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)
Affinity DataIC50:  44nMAssay Description:Covalent inhibition of NanoLuc fused BTK (unknown origin) expressed in HEK293 cells incubated for 90 mins by NanoBRET assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))TBA
LigandPNGBDBM50614535(CHEMBL5271284)
Affinity DataIC50:  109nMAssay Description:Covalent inhibition of NanoLuc fused BTK (unknown origin) expressed in HEK293 cells incubated for 90 mins by NanoBRET assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50614535(CHEMBL5271284)
Affinity DataIC50:  197nMAssay Description:Inhibition of EGFR (unknown origin) by Z'LYTE assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSerine/threonine-protein kinase LMTK3(Homo sapiens)
San Diego State University

Curated by ChEMBL
LigandPNGBDBM50542351(CHEMBL4637017)
Affinity DataIC50:  210nMAssay Description:Inhibition of LMTK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase LMTK3(Homo sapiens)
San Diego State University

Curated by ChEMBL
LigandPNGBDBM50542348(CHEMBL4647760)
Affinity DataIC50:  226nMAssay Description:Inhibition of LMTK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase LMTK3(Homo sapiens)
San Diego State University

Curated by ChEMBL
LigandPNGBDBM50542350(CHEMBL4635320)
Affinity DataIC50:  308nMAssay Description:Inhibition of LMTK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))TBA
LigandPNGBDBM50614536(CHEMBL5278149)
Affinity DataIC50:  314nMAssay Description:Covalent inhibition of NanoLuc fused BTK (unknown origin) expressed in HEK293 cells incubated for 90 mins by NanoBRET assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSerine/threonine-protein kinase LMTK3(Homo sapiens)
San Diego State University

Curated by ChEMBL
LigandPNGBDBM50542349(CHEMBL4649625)
Affinity DataIC50:  318nMAssay Description:Inhibition of LMTK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))TBA
LigandPNGBDBM50614535(CHEMBL5271284)
Affinity DataIC50:  344nMAssay Description:Inhibition of ITK (unknown origin) by Z'LYTE assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSerine/threonine-protein kinase LMTK3(Homo sapiens)
San Diego State University

Curated by ChEMBL
LigandPNGBDBM50542347(CHEMBL4638119)
Affinity DataIC50:  654nMAssay Description:Inhibition of LMTK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))TBA
LigandPNGBDBM50614535(CHEMBL5271284)
Affinity DataIC50:  874nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'LYTE assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSerine/threonine-protein kinase LMTK3(Homo sapiens)
San Diego State University

Curated by ChEMBL
LigandPNGBDBM50542346(CHEMBL4649046)
Affinity DataIC50:  1.61E+3nMAssay Description:Inhibition of LMTK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))TBA
LigandPNGBDBM50614536(CHEMBL5278149)
Affinity DataIC50:  1.71E+3nMAssay Description:Inhibition of SRC (unknown origin) by Z'LYTE assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetTyrosine-protein kinase HCK(Homo sapiens (Human))TBA
LigandPNGBDBM50614536(CHEMBL5278149)
Affinity DataIC50:  2.31E+3nMAssay Description:Inhibition of HCK (unknown origin) by Z'LYTE assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSerine/threonine-protein kinase LMTK3(Homo sapiens)
San Diego State University

Curated by ChEMBL
LigandPNGBDBM50299148((S)-1-(4-(5-cyclopropyl-1H-pyrazol-3-ylamino)pyrro...)
Affinity DataIC50:  3.16E+3nMAssay Description:Inhibition of LMTK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase LMTK3(Homo sapiens)
San Diego State University

Curated by ChEMBL
LigandPNGBDBM158154(US10081622, Compound 11 | US10370379, Entrectinib ...)
Affinity DataIC50:  4.65E+3nMAssay Description:Inhibition of LMTK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50614536(CHEMBL5278149)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of EGFR (unknown origin) by Z'LYTE assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))TBA
LigandPNGBDBM50614536(CHEMBL5278149)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ITK (unknown origin) by Z'LYTE assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))TBA
LigandPNGBDBM50614536(CHEMBL5278149)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'LYTE assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed