Compile Data Set for Download or QSAR
maximum 50k data
Found 67 with Last Name = 'guzikowski' and Initial = 'ap'
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50369783(CHEMBL1203902)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50085922(4-(4-Hydroxy-phenyl)-1-(4-phenyl-butyl)-piperidin-...)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50054631(8-Chloro-3-hydroxy-1H-benzo[b]azepine-2,5-dione | ...)
Affinity DataIC50:  13nMAssay Description:Tested for the inhibition of [3H]5,7-dichlorokynurenic acid (DCKA) binding to NMDA receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50085933(4-[1-(5-Phenyl-pentyl)-pyrrolidin-3-yl]-phenol | C...)
Affinity DataIC50:  17nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50085927(4-[1-(2-Hydroxy-4-phenyl-butyl)-piperidin-4-yl]-ph...)
Affinity DataIC50:  19nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50369786(CHEMBL1201889)
Affinity DataIC50:  19nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50369791(CHEMBL1202296)
Affinity DataIC50:  22nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50085929(4-(4-Hydroxy-phenyl)-1-(2-hydroxy-4-phenyl-butyl)-...)
Affinity DataIC50:  26nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50085921(4-[1-(3-Phenyl-propyl)-piperidin-4-ylmethyl]-pheno...)
Affinity DataIC50:  59nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50369784(CHEMBL1202295)
Affinity DataIC50:  71nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50369782(CHEMBL1203909)
Affinity DataIC50:  74nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50369787(CHEMBL1203901)
Affinity DataIC50:  75nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50059247((7S,8S)-7,8-Dichloro-3-hydroxy-6,7,8,9-tetrahydro-...)
Affinity DataIC50:  130nMAssay Description:Antagonism of N-methyl-D-aspartate glutamate receptor 1 sites using [3H]-DCKA as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50085923(4-[1-(4-Phenyl-butyl)-pyrrolidin-3-yl]-phenol | CH...)
Affinity DataIC50:  130nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50059247((7S,8S)-7,8-Dichloro-3-hydroxy-6,7,8,9-tetrahydro-...)
Affinity DataIC50:  131nMAssay Description:Tested for the inhibition of [3H]5,7-dichlorokynurenic acid (DCKA) binding to NMDA receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50085930(4-[1-(3-Phenyl-prop-2-ynyl)-piperidin-4-ylmethyl]-...)
Affinity DataIC50:  180nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50059246(3-Hydroxy-7,8-dimethyl-6,7,8,9-tetrahydro-1H-benzo...)
Affinity DataIC50:  228nMAssay Description:Tested for the inhibition of [3H]5,7-dichlorokynurenic acid (DCKA) binding to NMDA receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50059246(3-Hydroxy-7,8-dimethyl-6,7,8,9-tetrahydro-1H-benzo...)
Affinity DataIC50:  230nMAssay Description:Antagonism of N-methyl-D-aspartate glutamate receptor 1 glycine sites using [3H]-DCKA as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50369790(CHEMBL1203914)
Affinity DataIC50:  230nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50369789(CHEMBL1203894)
Affinity DataIC50:  410nMAssay Description:Inhibition of [3H]-raclopride binding at Dopamine receptor D2 in rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50085925(4-[1-(4-Phenyl-but-3-ynyl)-piperidin-4-ylmethyl]-p...)
Affinity DataIC50:  800nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50054638(3-Hydroxy-1H-benzo[b]azepine-2,5-dione | CHEMBL917...)
Affinity DataIC50:  827nMAssay Description:Tested for the inhibition of [3H]5,7-dichlorokynurenic acid (DCKA) binding to NMDA receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50369791(CHEMBL1202296)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of [3H]-raclopride binding at Dopamine receptor D2 in rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50007400(4-Phenyl-1-(4-phenyl-butyl)-piperidine | 4-Phenyl-...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50059245(3-Hydroxy-6,7,8,9-tetrahydro-1H-benzo[b]azepine-2,...)
Affinity DataIC50:  3.20E+3nMAssay Description:Antagonism of N-methyl-D-aspartate glutamate receptor 1 glycine sites using [3H]-DCKA as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50059245(3-Hydroxy-6,7,8,9-tetrahydro-1H-benzo[b]azepine-2,...)
Affinity DataIC50:  3.21E+3nMAssay Description:Tested for the inhibition of [3H]5,7-dichlorokynurenic acid (DCKA) binding to NMDA receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50085927(4-[1-(2-Hydroxy-4-phenyl-butyl)-piperidin-4-yl]-ph...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of [3H]-raclopride binding at Dopamine receptor D2 in rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50085922(4-(4-Hydroxy-phenyl)-1-(4-phenyl-butyl)-piperidin-...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of [3H]-raclopride binding at Dopamine receptor D2 in rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50085933(4-[1-(5-Phenyl-pentyl)-pyrrolidin-3-yl]-phenol | C...)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2A) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50369790(CHEMBL1203914)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2A) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50369782(CHEMBL1203909)
Affinity DataIC50:  5.10E+4nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2A) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50085923(4-[1-(4-Phenyl-butyl)-pyrrolidin-3-yl]-phenol | CH...)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2A) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50369786(CHEMBL1201889)
Affinity DataIC50:  5.90E+4nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2A) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50369788(CHEMBL1202294)
Affinity DataIC50:  6.10E+4nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50085922(4-(4-Hydroxy-phenyl)-1-(4-phenyl-butyl)-piperidin-...)
Affinity DataIC50:  6.20E+4nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2A) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50085929(4-(4-Hydroxy-phenyl)-1-(2-hydroxy-4-phenyl-butyl)-...)
Affinity DataIC50:  9.30E+4nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2A) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50085921(4-[1-(3-Phenyl-propyl)-piperidin-4-ylmethyl]-pheno...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2A) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50085923(4-[1-(4-Phenyl-butyl)-pyrrolidin-3-yl]-phenol | CH...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2C) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50085925(4-[1-(4-Phenyl-but-3-ynyl)-piperidin-4-ylmethyl]-p...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2A) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50369784(CHEMBL1202295)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2A) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50007400(4-Phenyl-1-(4-phenyl-butyl)-piperidine | 4-Phenyl-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2A) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50085930(4-[1-(3-Phenyl-prop-2-ynyl)-piperidin-4-ylmethyl]-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2A) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50085929(4-(4-Hydroxy-phenyl)-1-(2-hydroxy-4-phenyl-butyl)-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2C) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50369787(CHEMBL1203901)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2A) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50085925(4-[1-(4-Phenyl-but-3-ynyl)-piperidin-4-ylmethyl]-p...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2C) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50085922(4-(4-Hydroxy-phenyl)-1-(4-phenyl-butyl)-piperidin-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2C) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50085927(4-[1-(2-Hydroxy-4-phenyl-butyl)-piperidin-4-yl]-ph...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2A) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50369784(CHEMBL1202295)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2C) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50369782(CHEMBL1203909)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2C) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Cocensys

Curated by ChEMBL
LigandPNGBDBM50369788(CHEMBL1202294)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2A) Receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 67 total ) | Next | Last >>
Jump to: